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1-{6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-4-(oxolan-2-ylmethyl)piperazine
(2S,4R)-4-amino-N-ethyl-1-{pyrazolo[1,5-a]pyridine-2-carbonyl}pyrrolidine-2-carboxamide
3-{5-[5-(1,5-dimethyl-1H-pyrazol-4-yl)-1,2-oxazol-3-yl]-3-methyl-1H-1,2,4-triazol-1-yl}-1λ6-thiolane-1,1-dione
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(1,3-dimethyl-1H-pyrazole-5-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-{1-methyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-(pyridin-4-yl)propan-1-one
5-(2H-1,3-benzodioxol-4-ylmethyl)-3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
2-[(3S,4R)-3-acetamido-4-(4-methoxyphenyl)pyrrolidin-1-yl]pyridine-3-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-(pyridin-3-yl)pyridine-3-carboxamide
8-methoxy-N-{2-[4-(trifluoromethyl)phenyl]ethyl}-3,4-dihydro-2H-1-benzopyran-3-amine
1-[4-({2-[2-hydroxy-3-(piperidin-1-yl)propoxy]phenyl}methyl)-1,4-diazepan-1-yl]ethan-1-one
5-chloro-2-{4-[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl]piperazin-1-yl}pyrimidine
3-(1-{2,6-dimethylimidazo[1,2-a]pyridine-3-carbonyl}pyrrolidin-2-yl)-4-methyl-1,2,5-oxadiazole
1-ethyl-4-[4-(pyrimidin-2-yloxy)piperidine-1-carbonyl]-1,2-dihydropyridin-2-one
N-[2-hydroxy-3-(3-methoxyphenoxy)propyl]-2-(2-phenyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
3-{5-[(4-acetyl-1-methyl-1H-pyrrol-2-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-N-cyclopropylpropanamide
3-{[4-(4-chloro-2-fluorophenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}pyridin-2-amine
1-{4-[(2-methylphenyl)sulfanyl]piperidin-1-yl}-3-(morpholin-4-yl)propan-1-one
N-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
ethyl 1-(2-methoxyethyl)-5-(5-methyl-3-phenyl-1,2-oxazole-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(4-methylpiperazine-1-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
[1-(6-methylpyridazin-3-yl)piperidin-4-yl](thiophen-2-yl)methanol
2-hydroxy-1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}ethan-1-one
(4aR,8aR)-2-{[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]methyl}-7-methanesulfonyl-decahydro-2,7-naphthyridin-4a-ol
N-(3-cyano-4-ethoxyphenyl)-8-methyl-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxamide
(4aR,7aS)-4-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
6-{4-[(3-fluorophenyl)methyl]-1,4-diazepan-1-yl}-9H-purin-2-amine
3-{2-[4-(4,6-dimethylpyrimidin-2-yl)piperazin-1-yl]-2-oxoethyl}-1,3-diazinane-2,4-dione
1-(7,7-dimethyl-5-{[6-methyl-2-(methylamino)pyrimidin-4-yl]amino}-5,6,7,8-tetrahydroquinazolin-2-yl)piperidin-4-ol
1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(methoxymethyl)-N-[2-methyl-2-(morpholin-4-yl)propyl]-1H-pyrazole-4-carboxamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2-(4-methylphenoxymethyl)furan-3-carboxamide
2-[2-(1H-imidazol-1-yl)ethyl]-1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
5-(2-aminopyrimidin-4-yl)-N-cyclopropyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
3-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}pyridin-2-ol
(1R,5R)-6-methyl-3-[3-(trifluoromethyl)benzenesulfonyl]-3,6-diazabicyclo[3.2.2]nonane
N-(cyclopropylmethyl)-2-ethyl-7-(2-methoxybenzamido)-1-methyl-N-(oxolan-2-ylmethyl)-1H-1,3-benzodiazole-5-carboxamide
2-(dimethylamino)-N-[(5-methyl-1H-pyrazol-3-yl)methyl]-2-(4-methylphenyl)acetamide
{3-[(2-methylphenyl)methyl]-1-(quinolin-2-ylmethyl)piperidin-3-yl}methanol
N-[1-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(2-phenyl-1,3-thiazol-4-yl)acetamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-2-(pyrimidin-2-ylsulfanyl)acetamide
1-[(2,3-difluorophenyl)methyl]-N-[2-(4-methoxyphenyl)phenyl]piperidine-3-carboxamide
4-{9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}-N,N-dimethylpiperazine-1-carboxamide
dimethyl[1-(4-{1-methyl-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}phenyl)ethyl]amine
2-amino-N-[(1R,2R)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-phenylpyrimidine-5-carboxamide
N-methyl-2-(1H-1,2,4-triazol-1-yl)-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
methyl (2S)-2-{[1-(4-methylquinazolin-2-yl)piperidin-4-yl]formamido}-2-phenylacetate
1-(5-methanesulfonamido-2-methylphenyl)-3-methyl-3-[3-(oxolan-2-yl)propyl]urea
4-(4-cyclopropyl-1H-1,2,3-triazol-1-yl)-1-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-2-propoxyethan-1-one
2-[(2-methoxyethyl)(methyl)amino]-1-{4-[3-(trifluoromethyl)phenoxy]piperidin-1-yl}ethan-1-one
8-methoxy-N-[(4-methyl-1,3-benzoxazol-2-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide