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11-{[(2,5-difluorophenyl)methyl]amino}-4-(pyridin-4-ylmethyl)-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-2-propylpyridine
1-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethan-1-one
1-ethyl-N-methyl-N-{2-[(4-methylphenyl)sulfanyl]ethyl}-1H-pyrazole-3-carboxamide
N-[1-(2-chlorophenyl)cyclopropyl]-3-methoxy-2,2-dimethylpropanamide
N-{[3-fluoro-5-(trifluoromethyl)phenyl]methyl}-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
7-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
5-{[2-(5-methyl-1,2-oxazol-3-yl)piperidin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-3-(2-methoxyphenyl)-1H-pyrazole-5-carboxamide
(1S,5R)-6-(2H-1,3-benzodioxole-5-carbonyl)-3-(pyridin-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
1-cyclohexyl-5-(furan-3-yl)-3-(oxolan-3-yl)-1H-1,2,4-triazole
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
7-(thiophen-2-yl)-4-{[2-(trifluoromethyl)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-methoxybutyl)-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
1-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]urea
2-amino-1-{5-[5-(1-methoxypropyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl}ethan-1-one
2-[(2-fluorophenyl)methyl]-6-[4-(2-methoxyethoxy)piperidine-1-carbonyl]-1,3-benzoxazole
2-(3-methoxypropyl)-8-[(2-methylphenyl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3-[(cycloheptylamino)methyl]-1-[(3,4-difluorophenyl)methyl]-3-hydroxypiperidin-2-one
3-(2H-1,3-benzodioxol-5-yl)-1-(4-hydroxypiperidin-1-yl)-3-phenylpropan-1-one
1-(3-{[4-(2,6-diaminopyrimidin-4-yl)piperazin-1-yl]methyl}-2,4,6-trimethylphenyl)ethan-1-one
5-{1-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
1-[(dimethylcarbamoyl)methyl]-4-(1H-imidazol-4-ylmethyl)-1,4-diazepane-6-carboxylic acid
N-{1-[1-(4,5,6,7-tetrahydro-1,2-benzoxazole-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-[(1R,2R)-2-hydroxycyclohexyl]-N-propyl-3-(4H-1,2,4-triazol-4-yl)benzamide
4-{5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazin-2-one
N'-(butan-2-yl)-N-(2-chlorophenyl)-N'-(pyridin-3-ylmethyl)ethanediamide
1-[7-(1-benzothiophen-3-yl)-9-(oxolan-3-yloxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-3-(3-methyl-1H-pyrazol-1-yl)propan-1-one
ethyl 1-[1-(ethoxycarbonyl)piperidin-4-yl]-4-(2-phenylethyl)piperidine-4-carboxylate
1-[(1R,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-{8-methylimidazo[1,2-a]pyridin-3-yl}ethan-1-one
N-[2-(1H-1,3-benzodiazol-2-yl)ethyl]-4-chloro-1-ethyl-1H-pyrazole-3-carboxamide
N-[(3R,4S)-1-cyclopentanecarbonyl-4-cyclopropylpyrrolidin-3-yl]-2-(2,3-dihydro-1H-indol-1-yl)acetamide
4-(4-chlorophenyl)-N-(2-oxoazepan-3-yl)butanamide
[1-(3-fluoro-4-methylbenzenesulfonyl)-3-(3-methoxypropyl)piperidin-3-yl]methanol
3-[2-(aminomethyl)-5-methyl-2,3-dihydro-1-benzofuran-7-yl]-1-benzyl-N,N-dimethyl-1H-1,2,4-triazol-5-amine
(3R,4R)-4-(azepan-1-yl)-1-[3-(1H-pyrazol-1-yl)propyl]piperidin-3-ol
3-[(3S,4R)-4-[4-(2-methoxyphenyl)piperazin-1-yl]-1-(pyridin-3-ylmethyl)piperidin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
(2R)-2-{[3-(2-hydroxyphenyl)-1H-pyrazol-5-yl]formamido}-4-methylpentanoic acid
N2-({2-[(6-methylpyridin-3-yl)oxy]pyridin-3-yl}methyl)pyrrolidine-1,2-dicarboxamide
N3-(2-methylpropyl)-4-oxo-1-(propan-2-yl)-N5-[2,2,2-trifluoro-1-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
(1S,5R)-3-(pyrimidin-2-yl)-6-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
2-[4-(1,3-benzoxazol-2-yl)piperazin-1-yl]-2-(trimethyl-1H-pyrazol-4-yl)acetic acid
2-[2-(1-{3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]propanoyl}piperidin-4-yl)-1H-imidazol-1-yl]acetamide
5-[4-({methyl[(1-methylpiperidin-2-yl)methyl]amino}methyl)phenoxymethyl]furan-2-carboxylic acid
N-[(1R,3R)-3-aminocyclopentyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
1-methyl-2-{[3-(2-methylpiperidin-1-yl)azetidin-1-yl]methyl}-1H-1,3-benzodiazole
3-(4-chloro-1H-pyrazol-1-yl)-1-[2-(morpholin-4-ylmethyl)piperidin-1-yl]propan-1-one
2-[1-(cyclohexylmethyl)-4-{[3-(ethoxymethyl)-4-methoxyphenyl]methyl}piperazin-2-yl]ethan-1-ol