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1-methyl-5-[3-(4-methylphenyl)propanoyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
3-(1-ethyl-5-oxopyrrolidin-3-yl)-6,7-dimethoxy-3,4-dihydroquinazolin-4-one
N-[3-(1H-imidazol-1-yl)propyl]-7-methyl-N-(pyridin-4-ylmethyl)pyrazolo[1,5-a]pyrimidine-6-carboxamide
3-{[(4-acetylphenyl)methyl](methyl)amino}-N-methylpropanamide
(2S)-N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-2-phenylacetamide
(1R,3S,5S)-8-{2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carbonyl}-8-azabicyclo[3.2.1]octan-3-ol
(2S,4S,5R)-5-(2,3-difluorophenyl)-4-[(2-hydroxyethyl)carbamoyl]-1-methylpyrrolidine-2-carboxylic acid
5-{[3-(benzyloxy)phenyl]methyl}-1-(cyclopropylmethyl)-N-ethyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[2-(1-methyl-1H-pyrazol-5-yl)ethyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
N-{[2-(2-fluoro-5-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methyloxolan-3-amine
(3R,4R)-4-(4-hydroxypiperidin-1-yl)-1-{[2-(2-phenylethynyl)phenyl]methyl}piperidin-3-ol
1-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1-methyl-1H-pyrazol-4-yl)propan-1-one
2-butoxy-1-[(1S,5R)-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
8-fluoro-2-[4-(morpholine-4-carbonyl)piperazine-1-carbonyl]quinoline
4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]-1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidine
N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-N-(pyridin-4-ylmethyl)cyclopentanecarboxamide
1-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]-2-(piperazin-1-yl)ethan-1-one
N-[(3,5-dimethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
[1-(1H-1,3-benzodiazol-2-yl)ethyl][(2-chloro-5-ethoxy-4-propoxyphenyl)methyl]amine
(2S,4R)-N-ethyl-1-[(4-fluoro-2-methylphenyl)methyl]-4-[(3E)-hex-3-enamido]pyrrolidine-2-carboxamide
4-(2-methoxy-5-methylphenyl)-7-methylthieno[3,2-d]pyrimidine
N-[(3R,4R)-3-hydroxy-1-(3-methylpyrazin-2-yl)piperidin-4-yl]pyrazine-2-carboxamide
2-[(3-amino-1H-1,2,4-triazol-5-yl)sulfanyl]-N-(1-hydroxybutan-2-yl)-N-(thiophen-3-ylmethyl)acetamide
2-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]pyrimidine-5-carboxamide
N-[3-(2,3-dihydro-1H-indol-1-yl)propyl]pyrazolo[1,5-a]pyrimidine-2-carboxamide
N-[3-(3-fluorophenyl)phenyl]-1-(pyridin-2-ylmethyl)piperidine-4-carboxamide
N-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]acetamide
2-(2,4-difluorophenyl)-2-{methyl[(2-methyl-1,3-thiazol-4-yl)methyl]amino}acetic acid
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-[3-hydroxy-3-(pyrrolidin-1-ylmethyl)piperidin-1-yl]propan-1-one
(2R,6R)-11-methoxy-4-[2-(methylamino)acetyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N-[(4-methylphenyl)methyl]acetamide
4-[3-(2-aminoethyl)phenyl]-N-(pyridin-2-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(3-methoxybenzoyl)-1-(2-methylphenyl)piperazin-2-one
[(3R,4R)-4-(azepan-1-ylmethyl)-1-[(3-chloro-4-methoxyphenyl)methyl]pyrrolidin-3-yl]methanol
1-{3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pent-4-en-1-one
1-{3-ethyl-2-oxo-1-oxa-3,8-diazaspiro[4.5]decane-8-carbonyl}cyclopropane-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-{1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}propanamide
4-{1,4-dimethyl-1,4,9-triazaspiro[5.5]undecane-9-carbonyl}-N-propylaniline
2-(3-methylphenyl)-5-({4-[2-(pyridin-4-yl)ethyl]piperazin-1-yl}methyl)pyrimidine
5-methyl-N-{[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridin-3-yl]methyl}-1,2-oxazole-3-carboxamide
2-{[benzyl(ethyl)amino]methyl}-4-(6-methoxypyridin-2-yl)phenol
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-[(3-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(3R,4S)-1-[(2-chloro-4-fluorophenyl)methyl]-4-cyclopropylpyrrolidin-3-yl]-3-hydroxypropanamide
2-{1-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-3-oxopiperazin-2-yl}-N-[2-(pyridin-3-yloxy)ethyl]acetamide
8-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2-ethyl-2,8-diazaspiro[5.5]undecan-3-one
2-(dimethylamino)-1-{4-[(dimethylamino)methyl]-4-hydroxypiperidin-1-yl}-2-(4-methylphenyl)ethan-1-one
2-[benzyl(methyl)amino]-N-[(4-hydroxy-6-methylpyrimidin-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-2-(2,5,7-trimethyl-1H-indol-3-yl)ethan-1-one
1-[1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-yl]-2,3-dihydro-1H-1,3-benzodiazol-2-one
5-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-2-phenyl-2,3-dihydro-1H-pyrazol-3-one