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8-benzyl-2-(2-methoxyethyl)-2,8-diazaspiro[5.5]undecan-3-one
1-[(2-fluorophenyl)methyl]-N-[3-(1H-pyrazol-1-yl)phenyl]piperidine-3-carboxamide
1-{4-[4-ethyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-(2H-1,2,3-triazol-2-yl)ethan-1-one
2,3-dimethyl-7-[(3-methyl-1H-pyrazol-5-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-(carbamoylmethoxy)-N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]benzamide
2-[4-(5-propyl-1,3,4-oxadiazole-2-carbonyl)piperazin-1-yl]pyridine-3-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)[1-(4-methylpyridin-2-yl)propan-2-yl]amine
3-methyl-7-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-1-oxa-3,7-diazaspiro[4.5]decan-2-one
N-[1-(oxan-4-yl)piperidin-4-yl]-4-sulfamoylbenzamide
1-[3-(4-chloro-2-methylbenzoyl)piperidin-1-yl]-3-(dimethyl-1,2-oxazol-4-yl)propan-1-one
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
2-cyclopropyl-N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)acetamide
N-(2-{[2-(cyclopropylmethyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]amino}ethyl)-N-methylmethanesulfonamide
5-[4-(4-methoxypyrimidin-2-yl)piperazine-1-carbonyl]-2-methyl-3,4-dihydropyrimidin-4-one
4-[2-(3-methoxyphenyl)-1,3-benzoxazole-6-carbonyl]morpholine-2-carboxamide
2-(4-benzyl-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]acetamide
N-(2-hydroxyethyl)-5-{[2-(prop-2-yn-1-yloxy)phenyl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]acetamide
1-ethyl-8-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-{2-[(dimethylamino)methyl]-1,3-thiazole-4-carbonyl}-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-[4-(dimethylamino)-2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-methyl-1,2-dihydroquinolin-2-one
1-[4-(2,3-dimethylphenyl)piperazin-1-yl]-3-[(3S,4R)-4-(morpholin-4-yl)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]propan-1-one
1-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
3-[1-(2-hydroxy-5-methylbenzoyl)piperidin-4-yl]-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
(8R,9aS)-8-hydroxy-2-[3-(2-methoxyphenyl)propyl]-octahydro-1H-pyrido[1,2-a]piperazine-1,4-dione
(3aR,7aS)-2-(pyridin-4-yl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole
N-({1-[ethyl(methyl)amino]cyclohexyl}methyl)pyrimidin-4-amine
1-methyl-4-[2-(pyrrolidin-3-yl)benzoyl]piperazine
N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
(1,3-benzothiazol-2-ylmethyl)(methyl)({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)amine
methyl 6-(2-chloro-4-fluorobenzoyl)-2-(pyrrolidine-1-sulfonyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
N-(5-chloro-2-methoxyphenyl)-3-[1-(1,4-dithiepan-6-yl)piperidin-3-yl]propanamide
[2-(3,4-dimethoxyphenyl)ethyl]({[3-(diphenylmethyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
N-[2-(dimethylamino)ethyl]-N,1,6-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(2r,4r)-2-(4-acetyl-4-phenylpiperidine-1-carbonyl)-5,7-diazaspiro[3.4]octane-6,8-dione
2-{1-[(9-methyl-9H-carbazol-2-yl)methyl]piperidin-2-yl}acetic acid
1-[1-(2,1,3-benzoxadiazole-5-carbonyl)piperidin-3-yl]-3-phenylpropan-1-one
6-[3-(pyridin-2-yl)azetidin-1-yl]pyridine-2-carbonitrile
3-hydroxy-N-{2-[1-(1H-imidazol-4-ylmethyl)piperidin-3-yl]ethyl}-2-methylbenzamide
5-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-3-(propan-2-yl)-4,5-dihydro-1,2-oxazole
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-N-methyl-2-(3-oxopiperazin-1-yl)acetamide
1-[2-({1-[3-(2-oxopyrrolidin-1-yl)phenyl]piperidin-4-yl}amino)ethyl]imidazolidin-2-one
N-[3-(dimethylamino)propyl]-1-[(4,5-dimethylfuran-2-yl)methyl]-N-methylpiperidin-3-amine
N3-cyclooctyl-N5-[3-(dimethylamino)-2,2-dimethylpropyl]-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-methyl-N-[1-(phenylcarbamoyl)piperidin-4-yl]-1,3-benzoxazole-6-carboxamide
1-[2-fluoro-5-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-3-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]urea
3-ethyl-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidin-1-yl)ethan-1-one
1-{1-[2-(2-chloro-4-fluorophenyl)acetyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]-1H-1,2,3-triazole-4-carboxamide