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3-(5-methylfuran-2-yl)-N-[1-phenyl-2-(pyrrolidin-1-yl)ethyl]-1H-pyrazole-5-carboxamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(2-methoxyphenyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-pyrazole
N-{[7-fluoro-2-(4-hydroxypiperidin-1-yl)quinolin-3-yl]methyl}-3-(2-methoxyphenyl)-N-(oxolan-2-ylmethyl)propanamide
3-[(3S)-3-(dimethylamino)azepane-1-carbonyl]-5-fluorobenzonitrile
4-{5-[(cyclohexylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}-1-(furan-2-ylmethyl)piperidine
1-[3-(4-methylphenyl)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
6-[4-(dimethylamino)azepane-1-carbonyl]-2,5-dimethyl-3H,4H-thieno[2,3-d]pyrimidin-4-one
7-(1,3-benzothiazol-2-yl)-4-[(2,5-dimethoxyphenyl)methyl]-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-(1-{imidazo[1,2-a]pyrimidin-2-yl}propyl)-4-oxo-3,4-dihydroquinazoline-2-carboxamide
4-(2-methoxyphenoxy)-1-{[5-methyl-2-(3-methylthiophen-2-yl)-1,3-oxazol-4-yl]methyl}piperidine
[(3-{2-[4-(2H-1,3-benzodioxole-5-carbonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(naphthalen-1-ylmethyl)amine
1-(1,2,3,4-tetrahydronaphthalene-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
methyl (1R,3R,3aR,6aS)-1-butyl-5-ethyl-3-(oxan-4-yl)-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-[(2R,3R)-2-hydroxy-1'-[(3-methylthiophen-2-yl)methyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-2-phenoxyacetamide
3-[(3R,4S)-1-(1,3-benzothiazol-2-yl)-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
3-(1H-indol-3-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}propanamide
2-[4-(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)piperidin-1-yl]pyrazine
1-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidin-1-yl)-3-methylbut-2-en-1-one
1-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
1-[(3R,4S)-4-hydroxy-3,4-dimethylpiperidin-1-yl]-3-[2-(hydroxymethyl)-1H-1,3-benzodiazol-1-yl]propan-1-one
2-(2,5-dimethoxyphenyl)-N-{[6-(dimethylamino)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}-N-[2-(dimethylamino)ethyl]acetamide
4-ethyl-3-{1-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]piperidin-4-yl}-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[4-(1-cyclohexyl-1H-1,2,4-triazol-5-yl)thiophen-2-yl]ethan-1-one
[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl](methyl)({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)amine
1-[3-(2-amino-1,3-thiazol-4-yl)propanoyl]-3-(2-methoxyethyl)piperidine-3-carboxylic acid
3-methyl-4-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]-1-[(4-methylphenyl)methyl]piperazin-2-one
6-oxo-1-(propan-2-yl)-N-{[3-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidine-3-carboxamide
N-[(3S,4R)-1-(2-fluorobenzoyl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-[(3-methoxyphenyl)methyl]-6-(oxolane-3-carbonyl)-3-phenyl-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-(2,1,3-benzothiadiazol-5-ylmethyl)-4-hydroxy-N-methyl-2-(pyridin-3-yl)pyrimidine-5-carboxamide
2-[4-(4-aminopyrimidin-2-yl)-1-(3-phenylpropyl)piperazin-2-yl]ethan-1-ol
N-methyl-4-{2-[2-(morpholin-4-yl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
3-(2,3-dihydro-1H-isoindol-2-yl)-N-(2,4-dimethoxyphenyl)-3-oxopropanamide
2-{2-[(3aR,7aS)-2,3,3a,4,7,7a-hexahydro-1H-isoindol-2-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
1-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-3-[1-phenyl-3-(propan-2-yl)-1H-pyrazol-5-yl]urea
(3S)-1-[6-chloro-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]-N,N-dimethylpyrrolidin-3-amine
N-[1-(2-chlorophenyl)cyclopropyl]-1-methyl-1H-1,3-benzodiazole-5-carboxamide
1-methyl-6-(pyridin-4-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
4-({5-ethyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}carbonyl)-6-(propan-2-yl)pyrimidin-2-amine
(3aS,6aS)-2-cyclobutanecarbonyl-5-[2-(pyridin-3-yl)acetyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(carbamoylmethyl)-N-[3-(1H-indol-2-yl)phenyl]piperidine-3-carboxamide
2-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-[1-(propan-2-yl)piperidine-4-carbonyl]morpholine
(2R,6R)-1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)-6-methyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
1-[(2-oxo-2,3-dihydro-1,3-benzothiazol-6-yl)sulfonyl]-3-propylpiperidine-3-carboxylic acid
7-{[3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazol-5-yl]methoxy}-1,2-benzoxazole
(3S,4R)-1-[(3-fluoro-5-methylphenyl)methyl]-N,N-dimethyl-4-(propan-2-yl)pyrrolidin-3-amine
N-[(2,5-dimethylphenyl)(pyridin-3-yl)methyl]-1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
5-({4-[1-(4-fluorophenyl)-1H-pyrazol-4-yl]pyrimidin-2-yl}amino)pentan-1-ol