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3-{1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)benzoyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-[2-oxo-8-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-3-yl]acetic acid
(2R,6S)-4-[3-(1-benzothiophen-2-yl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-2,6-dimethylmorpholine
2-methyl-5-[(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)methyl]-[1,2,4]triazolo[1,5-a]pyrimidin-7-ol
2-{3-[3-(pyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1,3-thiazol-2-yl)propanamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-methyl-2-(morpholin-4-yl)propyl]propanamide
1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethan-1-one
4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]-N-methyl-N-(thian-4-yl)benzamide
2-amino-3-ethyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-3H-imidazo[4,5-b]pyridine-6-carboxamide
5-{3-[4-(2,3-dihydro-1H-inden-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}imidazolidine-2,4-dione
4-[4-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
2-({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)-1-methylpiperidine
1-[4-(3-carboxy-4-ethoxyphenyl)pyrimidin-2-yl]piperidine-4-carboxylic acid
2-{1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
2-{3-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-1,3-thiazole-4-carboxamide
1-(3-chloro-5-fluorophenyl)-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-methyl-9-{2-[methyl(pyridin-4-ylmethyl)amino]acetyl}-1,4,9-triazaspiro[5.5]undecan-5-one
1-(2-cyclohexylethyl)-3-hydroxy-3-{[methyl({[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl})amino]methyl}piperidin-2-one
2-[5-(azepan-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]-N-(2-hydroxy-2-phenylethyl)-N-methylacetamide
(3R,4S)-4-{[(6-methoxy-2H-1,3-benzodioxol-5-yl)methyl](methyl)amino}oxolan-3-ol
1-(1-{[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidin-3-yl)-3-methylbutan-1-one
5-{1H-pyrazolo[3,4-b]pyridin-1-ylmethyl}-3-(2,3,4-trimethoxyphenyl)-1,2,4-oxadiazole
2-(dimethylamino)-1-{4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]piperidin-1-yl}-2-(3-methylphenyl)ethan-1-one
ethyl[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](pyridin-4-ylmethyl)amine
2-methoxy-1-{1'-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
5-methoxy-1-methyl-N-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-1H-indole-2-carboxamide
N-[1-(3,5-difluorophenyl)ethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
(4aR,6R,8aS)-8a-(methoxymethyl)-6-(morpholin-4-yl)-2-(thiophen-2-ylmethyl)-decahydroisoquinoline
3-(2-hydroxyphenyl)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-1H-pyrazole-5-carboxamide
5-(2-{[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]amino}ethyl)-1-[3-(propan-2-yloxy)propyl]pyrrolidin-2-one
4-(2-{8-chloro-5-methyl-[1,2,4]triazolo[4,3-a]quinolin-1-yl}-2-methylpropyl)morpholine
{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}(methyl)(1H-pyrazol-3-ylmethyl)amine
1-[4-(3-butyl-4H-1,2,4-triazol-4-yl)phenyl]ethan-1-one
2-ethoxy-N-[1-(3-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]acetamide
2-(2-methylphenyl)-1-[4-(morpholin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
N-[1-(4-fluorophenyl)-4-(morpholin-4-yl)-1H-indazol-3-yl]-1,3-oxazole-4-carboxamide
5-cyclobutanecarbonyl-1'-(1-methyl-1H-pyrazole-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
[(3,5-dichloropyridin-4-yl)methyl](methyl)(oxan-4-ylmethyl)amine
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-(pyridin-4-ylmethyl)piperazin-2-yl}ethan-1-ol
1-{[3-(benzyloxy)phenyl]methyl}-1,4-diazepane-6-carboxylic acid
3-(3-chloro-1H-1,2,4-triazol-5-yl)-1-[2-(3-methoxyphenyl)pyrrolidin-1-yl]propan-1-one
(3R,4R)-1-[4-(methoxymethyl)benzoyl]-4-methyl-3-(propan-2-yl)pyrrolidin-3-ol
{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}(methyl)[(1-methyl-1H-pyrazol-4-yl)methyl]amine
N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-3-(1H-pyrazol-1-ylmethyl)benzamide
N-(3-chloro-4-fluorophenyl)-2,8-diazaspiro[4.5]decane-2-carboxamide
N-[2-(3-methoxyphenyl)phenyl]-1-(pyridin-4-yl)piperidine-4-carboxamide
N-[(1S,2R)-2-(cyclopentylamino)cyclobutyl]-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
[1-(2,3-dihydro-1,4-benzodioxine-5-sulfonyl)-3-propylpiperidin-3-yl]methanol
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[3-(methylsulfanyl)phenyl]urea
2-[4-(benzyloxy)piperidine-1-carbonyl]thiophen-3-amine