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4-{[propyl(pyridin-4-ylmethyl)amino]methyl}benzonitrile
4-[(2-propoxypropyl)carbamoyl]benzoic acid
3-(1H-1,3-benzodiazol-2-yl)-1-[2-(pyridin-2-yl)piperidin-1-yl]propan-1-one
3-(dimethyl-1H-1,2,4-triazol-1-yl)-1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-methylpropan-1-one
(3S)-N-tert-butyl-2-[(5-cyano-1,2-dimethyl-1H-pyrrol-3-yl)methyl]-1,2,3,4-tetrahydroisoquinoline-3-carboxamide
N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}-1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carboxamide
4-{3-[(dimethylamino)methyl]benzoyl}-3-(3-fluorophenyl)piperazin-2-one
2-{3-cyclopentyl-5-[4-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1H-1,2,4-triazol-1-yl}ethan-1-ol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2,5,6-trimethylpyrimidin-4-amine
N-({6-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]pyridin-3-yl}methyl)acetamide
3-{5-[2-hydroxy-2-(4-methoxyphenyl)acetyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
8-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propanoyl]-3-(pentan-2-yl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[2-(5-methylfuran-2-yl)-2-(morpholin-4-yl)ethyl]-4-(pyridin-2-yl)pyrimidin-2-amine
1-[1-(3-chlorobenzoyl)piperidin-4-yl]-N-cyclopentyl-1H-1,2,3-triazole-4-carboxamide
8-(2-hydroxyacetyl)-1-methyl-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
3-{[1-(2-propyl-1,3-thiazole-4-carbonyl)piperidin-4-yl]oxy}pyridine
1-cyclohexyl-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]piperidine-4-carboxamide
1-(2-{[4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-yl]amino}ethyl)pyrrolidin-2-one
5-(2,2-dimethyloxan-4-yl)-3-(ethoxymethyl)-1-methyl-1H-1,2,4-triazole
1-{2-[6-(hydroxymethyl)-1,4-oxazepan-4-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
4-hydroxy-N-{[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]methyl}-2-(thiophen-2-yl)pyrimidine-5-carboxamide
4-methyl-2-(2-{2-oxa-7-azaspiro[4.5]decan-7-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
2-{[(2-chlorophenyl)methyl]sulfanyl}-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}acetamide
3-(7-chloro-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[2-(pyridin-3-yloxy)propyl]propanamide
2-(3-fluorophenoxymethyl)-N-{[1-(hydroxymethyl)cyclopropyl]methyl}-N-methyl-1,3-oxazole-4-carboxamide
N-[(5-chloro-3-methyl-2-phenyl-1H-indol-7-yl)methyl]-3-fluoropyridine-4-carboxamide
2-{4-[(2-methylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-2-(pyridin-2-yl)pyrimidin-4-ol
5-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N,N-dimethyl-2-(2-methylquinazolin-4-yl)aniline
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-N-propylpiperidine-1-carboxamide
(3R,4R)-1-[1-(furan-2-ylmethyl)piperidine-4-carbonyl]-4-(hydroxymethyl)piperidin-3-ol
(2S,4S)-4-amino-1-(3,5-dimethylbenzenesulfonyl)-N-ethylpyrrolidine-2-carboxamide
N-[1-(dimethylsulfamoyl)azepan-3-yl]thiophene-3-carboxamide
[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl][(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]amine
4-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]-1,3-oxazole-5-carboxamide
1-{4-[4-cyclopropyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}propan-1-one
N-{1-[1-(2-methoxy-2-phenylacetyl)piperidin-4-yl]-2-phenylethyl}-N,1,3-trimethyl-1H-pyrazole-5-carboxamide
5-(1-{5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}pyrrolidin-2-yl)-3-phenyl-1,2,4-oxadiazole
2-[(1-cyclohexyl-1H-imidazol-5-yl)methyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
6-(2H-1,3-benzodioxol-5-yl)-4-methyl-1,2-dihydroquinolin-2-one
1-[(dimethyl-1,3-thiazol-2-yl)methyl]-4-ethyl-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl (1R,3S,3aR,6aS)-3-(1-benzofuran-5-yl)-1-ethyl-5-methyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
N-{1-[(4-chlorophenyl)methyl]piperidin-3-yl}pent-4-enamide
3-(3-hydroxy-3-methylbutyl)-N-[2-(pyridin-3-ylformamido)ethyl]benzamide
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-1-(2-methoxyethyl)piperidine-4-carboxamide
(3R,4S)-4-cyclopropyl-1-[1-(3-methoxybenzoyl)piperidine-4-carbonyl]pyrrolidin-3-amine
3-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-1-[5-(dimethylamino)-2-methylphenyl]urea
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-6-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
5-(4-fluorophenyl)-3-(1-hydroxybutan-2-yl)-3H,4H-thieno[2,3-d]pyrimidin-4-one