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(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-(5,6-dimethylpyridine-3-carbonyl)pyrrolidine-3-carboxylic acid
N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[(2-ethoxy-3-methoxyphenyl)methyl]-1-(propan-2-yl)piperidin-4-amine
3-(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)-1-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}urea
2-ethyl-4-methyl-6-{4-[(2E)-3-phenylprop-2-en-1-yl]piperazin-1-yl}pyrimidine
2,6-dioxo-N-[2-(1-phenyl-1H-pyrazol-4-yl)ethyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-{[3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)pyrimidin-2-amine
4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
1-tert-butyl-4-(7-fluoro-1,2,3,4-tetrahydroisoquinoline-2-carbonyl)pyrrolidin-2-one
N-{[1-(morpholin-4-yl)cycloheptyl]methyl}-1-propyl-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(6-chloro-2-methylpyridin-3-yl)-4-[hydroxy(pyridin-2-yl)methyl]piperidine-1-carboxamide
8-[(1-methyl-1H-imidazol-4-yl)sulfonyl]-2-(3-methylbut-2-en-1-yl)-2,8-diazaspiro[4.5]decan-3-one
1-[1-(4-methylbenzoyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
5-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}pyrrolidin-2-yl)-3-(propan-2-yl)-1,2,4-oxadiazole
4-[5-methyl-2-oxo-4-(3-phenoxypropanoyl)piperazin-1-yl]benzonitrile
2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-2,3-dihydro-1H-isoindole
2-{[(4-hydroxyphenyl)formamido]methyl}-N,N-dimethyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carboxamide
2-[2-({[4-(dimethylamino)oxan-4-yl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
3-[(3S,7S,8aS)-1,4-dioxo-3-(propan-2-yl)-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(2,3-dichlorophenyl)urea
(2S)-4-methyl-2-{4-[2-(1H-pyrazol-1-ylmethyl)phenyl]-1H-1,2,3-triazol-1-yl}pentan-1-ol
N-[2-(2-fluorophenoxy)ethyl]-N-(2-methoxyethyl)-6,6-dimethyl-5-oxothiomorpholine-3-carboxamide
5-[2-(4,5-dimethyl-1H-pyrazol-3-yl)ethyl]-1-(2-methoxyphenyl)-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)-2-(1H-pyrazol-1-yl)acetamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-[(2-oxo-1,2-dihydroquinolin-3-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2E)-1-[4-(3-{[methyl(naphthalen-1-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-3-(thiophen-2-yl)prop-2-en-1-one
1-{3-[4-(2-phenoxyethyl)piperazine-1-carbonyl]piperidin-1-yl}ethan-1-one
2-(dimethylamino)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)acetamide
(4aS,8aR)-1-(3-aminopropyl)-6-(1H-1,2,3-benzotriazole-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-[(5-ethylpyridin-2-yl)methyl]-2,8-diazaspiro[4.5]decane
6-chloro-N,N-dimethyl-3-{[(1-phenylpiperidin-4-yl)amino]methyl}imidazo[1,2-a]pyridine-2-carboxamide
N-[2-(2-fluorophenoxy)ethyl]-3-methyl-1-propyl-1H-pyrazole-4-carboxamide
2-methoxy-1-{1'-[2-(1H-1,2,3,4-tetrazol-1-yl)acetyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl}ethan-1-one
1-methyl-5-[(2-phenyl-1,3-thiazol-4-yl)methyl]-3-(1H-1,2,4-triazol-1-ylmethyl)-1H-1,2,4-triazole
N-[2-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)ethyl]-N,1-dimethyl-1H-indole-6-carboxamide
(3S,4S)-4-cyclopropyl-1-{2-[(3-methoxyphenyl)sulfanyl]acetyl}pyrrolidine-3-carboxylic acid
N-{1-[1-(2-acetylbenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
1-{4-[(4-fluorophenyl)methyl]-1,4-diazepan-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
7,7-dimethyl-N-[(3-methylphenyl)methyl]-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-amine
1-methyl-N-[(5-methyl-2-{3-[2-(4-methylphenoxy)acetamido]phenyl}-1,3-oxazol-4-yl)methyl]-6-oxo-1,4,5,6-tetrahydropyridazine-3-carboxamide
4-[7-fluoro-2-(1H-pyrazol-4-yl)quinoline-4-carbonyl]-1λ6-thiomorpholine-1,1-dione
1-[3-(4-fluorophenoxy)azetidin-1-yl]-2-hydroxy-4-(methylsulfanyl)butan-1-one
1-[3-(2-fluorophenyl)-1H-pyrazole-5-carbonyl]-4-(hydroxymethyl)azepan-4-ol
2-chloro-4-[3-(3-ethylphenoxy)azetidine-1-carbonyl]phenol
3-(2-benzyl-1,3-thiazole-4-carbonyl)-3,9-diazaspiro[5.5]undecane
N-[(3-tert-butyl-1H-pyrazol-5-yl)methyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-(3-hydroxy-3-methylbutyl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]benzamide
(2H-1,3-benzodioxol-5-ylmethyl)({[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})amine
11-{[(3,5-difluorophenyl)methyl]amino}-4-[2-(pyridin-2-yl)ethyl]-8-thia-4,6-diazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-methyl-N-[2-(methylsulfanyl)ethyl]-3-{1-oxa-7-azaspiro[3.5]nonane-7-sulfonyl}benzamide
N-{1-[1-(3-cyclopentylpropyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide