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4-(1-benzofuran-5-carbonyl)-1-(3-chlorophenyl)-5-methylpiperazin-2-one
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-{7,9-dioxo-8-azaspiro[4.5]decan-8-yl}-N-[2-(4-fluorophenyl)ethyl]acetamide
4-({3-[2-(propan-2-yloxy)phenyl]phenyl}methyl)morpholine
6-[4-(4-methoxyphenyl)-3,3-dimethylpiperazin-1-yl]pyrimidin-4-amine
N-{[5,8-dimethoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-(furan-2-ylmethyl)-1,2,5-thiadiazole-3-carboxamide
8-{[3-(2-hydroxyethoxy)phenyl]methyl}-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[(3R,5S)-5-({imidazo[2,1-b][1,3]thiazol-6-ylmethyl}carbamoyl)pyrrolidin-3-yl]-3,5-dimethyl-1,2-oxazole-4-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[2-methyl-4-(pyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]propan-1-one
1-[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-hydroxyethan-1-one
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(3R,4R)-1-[(2-methoxyquinolin-3-yl)methyl]-4-(morpholin-4-yl)piperidin-3-ol
ethyl 4-({[2-(2-methylphenoxy)pyridin-3-yl]methyl}amino)piperidine-1-carboxylate
3-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-6-ethyl-1,5-dimethyl-1,2-dihydropyridin-2-one
2-[3-(2-methylpropyl)-5-[2-(pyridin-3-yl)ethyl]-1H-1,2,4-triazol-1-yl]pyridine
6-(3-oxo-1,4-diazepan-1-yl)-N-propylpyridine-3-carboxamide
2-methyl-5-(2-{2-[(quinoxalin-2-yl)amino]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
7-{5-[(pyrimidin-2-ylsulfanyl)methyl]furan-2-carbonyl}-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-ethyl-8-[4-(pyrrolidin-1-ylmethyl)benzoyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(1-cyclobutanecarbonylpiperidin-3-yl)-N-(2-methylpropyl)-1H-1,2,3-triazole-4-carboxamide
N-[(5-methylfuran-2-yl)methyl]-2-(pyridazine-3-carbonyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
3-[4-(1,3-benzoxazol-2-yl)phenyl]-1-[(4-methylmorpholin-2-yl)methyl]urea
4-({5-[1-(2-fluorobenzoyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)morpholine
1-(pyrimidin-2-yl)-N-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-amine
1-(6-amino-2-{[(2-methylphenyl)methyl]sulfanyl}pyrimidin-4-yl)piperidin-3-ol
(2R,3R,6R)-3-phenyl-5-(2-phenylethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-hydroxyquinoxalin-2-yl)-N-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}ethyl)propanamide
1-benzyl-5-(2,4,5-trimethoxyphenyl)-1H,4H-pyrazolo[3,4-d]imidazole
methyl 4-{4-[(2R)-2-amino-3-methoxypropanoyl]piperazin-1-yl}benzoate
6-{4-[4-(propan-2-yl)-6-(trifluoromethyl)pyrimidin-2-yl]piperazin-1-yl}pyrimidin-4-amine
N-(dimethyl-1H-1,2,4-triazol-3-yl)-4-(1-hydroxy-2-methylpropyl)piperidine-1-carboxamide
2-(1-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-1,2,3-triazol-4-yl)-4,5,6,7-tetrahydro-1,3-benzothiazole
methyl({[5-(oxan-4-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl})(pyridin-3-ylmethyl)amine
1-(2-phenylethyl)-2-(propane-2-sulfonyl)-5-(pyrrolidin-1-ylmethyl)-1H-imidazole
N-[(3S,4R)-1-[(1-ethyl-1H-imidazol-2-yl)methyl]-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
(2S)-1-(4-{1-[3-(dimethylamino)propyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-hydroxy-2-phenylethan-1-one
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-3-(1-phenylethyl)-1,2-oxazole-5-carboxamide
1-cyclohexyl-3-[4-(1H-pyrazol-5-yl)phenyl]-1-(pyridin-3-ylmethyl)urea
N-[2-(methylsulfanyl)ethyl]-2-[3-oxo-1-(2-phenylethyl)piperazin-2-yl]acetamide
4-[(5-{1-[(dimethyl-1,2-oxazol-4-yl)methyl]piperidin-4-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
3-{[4-(cyclopropylmethyl)-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}pyridin-2-amine
[3-(2-methoxyethyl)-1-(2-methoxypyridine-3-carbonyl)piperidin-3-yl]methanol
5-{1-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}-5-propyl-3-[2-(pyridin-2-yl)ethyl]imidazolidine-2,4-dione
[(3S,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(4-methylbenzoyl)piperidin-3-yl]methanol
1-[(2R,3R,6R)-3-(4-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methylpropan-1-one
3-{1-[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]-1H-imidazol-2-yl}-1,2-dihydroquinolin-2-one
2-({3-[3-(2,4-dimethoxyphenyl)phenyl]-1H-pyrazol-1-yl}methyl)pyridine
5-(1-ethyl-1H-pyrazol-3-yl)-1-[4-(trifluoromethyl)phenyl]-1H-1,2,4-triazole
(3R,4S)-4-propyl-1-(pyridazine-3-carbonyl)pyrrolidin-3-amine
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-3-(methylsulfanyl)propanamide