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12-[3-(1H-pyrazol-5-yl)piperidine-1-carbonyl]-8-thia-5-azatricyclo[7.4.0.02,7]trideca-1(13),2(7),9,11-tetraen-6-one
5-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazole
8-[4-(thiophen-2-yl)butanoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
(4-{[2-methoxy-1-(1-methyl-1H-pyrazol-5-yl)ethyl]amino}quinazolin-2-yl)methanol
N-[3-(1H-indol-1-yl)propyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
N-[(5-{[2-(cyclopentylmethyl)-1H-imidazol-4-yl]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl)methyl]acetamide
4-(2,4-dimethoxybenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-{3-methyl-1-[(3-methylphenyl)methyl]-1H-pyrazol-5-yl}acetamide
3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}-1-(morpholin-4-yl)propan-1-one
N-(3-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-3-oxopropyl)-4-methylbenzamide
5-[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidine-1-carbonyl]pyridine-2,4-diol
4-(2-ethylpiperidine-1-carbonyl)-7,8-dimethyl-2-(1-methyl-1H-pyrazol-4-yl)quinoline
[(3,5-dimethoxyphenyl)methyl]({1-[5-methyl-1-(naphthalen-1-yl)-1H-pyrazol-4-yl]ethyl})amine
(4aS,8aS)-2-{[3-(4-methoxyphenoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
9-{[2-(dimethylamino)pyrimidin-5-yl]methyl}-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
4-(3-{1-[2-(1H-1,2,4-triazol-1-yl)ethyl]-1H-pyrazol-3-yl}phenyl)isoquinoline
3-(2-hydroxyphenyl)-N-{3-[(pyridin-3-yl)amino]propyl}-1H-pyrazole-5-carboxamide
N-ethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carboxamide
4-(2-fluorophenoxy)-1-(1-hydroxycyclopentanecarbonyl)piperidine-4-carboxylic acid
2-amino-6-(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)-4-[2-(methylsulfanyl)pyrimidin-5-yl]pyridine-3-carbonitrile
1-(furan-2-yl)-2-[3-oxo-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethane-1,2-dione
1-[2-(2-ethoxyethoxy)benzoyl]-4-[(4-methyl-4H-1,2,4-triazol-3-yl)methyl]piperidine
N-methyl-N-[(4-phenoxyphenyl)methyl]-2-(pyrrolidin-1-yl)propanamide
N-[2-(oxan-3-yl)ethyl]-5-propylpyrazolo[1,5-a]pyrimidin-7-amine
2-({1-[(4-chloro-3-fluorophenyl)methyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
N-methyl-N-{2-[5-(2-methylprop-1-en-1-yl)-4-phenyl-1H-imidazol-1-yl]ethyl}methanesulfonamide
N4-methyl-6-(morpholin-4-yl)-N4-[(3-phenyl-1,2-oxazol-5-yl)methyl]pyrimidine-2,4-diamine
1-{[2-(3,4-dimethoxyphenoxy)phenyl]methyl}-4-methylpiperazine
methyl 2-[methyl({3-[(3-methyl-1,2-thiazol-5-yl)carbamoyl]phenyl}methyl)amino]acetate
3-[(1R,2S,6R,7S)-4-azatricyclo[5.2.2.02,6]undecane-4-carbonyl]-1-ethyl-4,6-dimethyl-1,2-dihydropyridin-2-one
2-ethyl-6-methyl-1-[(5-methylfuran-2-yl)methyl]-N-[3-(morpholin-4-yl)propyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
6-{1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}pyridine-2-carbonitrile
N-(4-fluorophenyl)-1-(oxane-4-carbonyl)piperazine-2-carboxamide
4-[4-(6-ethoxy-2,3-dihydro-1H-inden-5-yl)-1H-1,2,3-triazol-1-yl]-1-ethylpyrrolidin-2-one
1-(4-methoxy-3-{[1-(propan-2-yl)piperidin-4-yl]oxy}benzoyl)azepane
9-[2-(methylsulfanyl)propanoyl]-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-chloro-2-methylphenyl)-3-oxo-3-[2-(pyridin-3-yl)piperidin-1-yl]propanamide
1-(2-{2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl}-2-oxoethyl)-3-methoxy-1,2-dihydropyridin-2-one
5-(1H-imidazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
6-(methoxymethyl)-N-[1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-yl]pyrimidin-4-amine
2-methoxy-N,N-bis(propan-2-yl)-6-[1-(1H-1,2,3,4-tetrazol-5-yl)-1H-pyrazol-4-yl]benzamide
1-(1-cyclopropanecarbonylpiperidine-4-carbonyl)-2-(3-methoxyphenyl)piperidine
N-[1-(5-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-1-(2-methyl-5-propylpyrimidin-4-yl)piperidin-4-amine
N-(1-methylpiperidin-4-yl)-2,7-dioxo-N-(2-phenylethyl)-1,3-diazepane-4-carboxamide
1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-(morpholin-4-yl)ethan-1-one
4-methoxy-2-(8-methylquinolin-5-yl)phenol
N-[(3R,5S)-5-(ethylcarbamoyl)-1-[2-(methylsulfanyl)acetyl]pyrrolidin-3-yl]-2,6-dimethylpyrimidine-4-carboxamide
2-methyl-6-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-3-yl}pyrimidin-4-ol
N-(3,4-difluorophenyl)-1-[3-(dimethylamino)benzoyl]piperidin-3-amine
4-[(4-cyclopentylpyrimidin-2-yl)amino]-1-(4-methoxyphenyl)pyrrolidin-2-one