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N-{[3-(2-chlorophenyl)-1,2-oxazol-5-yl]methyl}-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
2-(2-methoxyquinolin-3-yl)-N-(propan-2-yl)pyrimidin-4-amine
1-({1-[6-(4-methylphenyl)pyridine-3-carbonyl]piperidin-4-yl}methyl)pyrrolidin-2-one
4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1H-pyrrole-2-carbonyl)piperidine
2,6-dihydroxy-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]benzamide
1-ethyl-4-{[1-(4-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}-3-methyl-1H-pyrazole
3-{5H,6H,7H-pyrrolo[2,1-c][1,2,4]triazol-3-ylmethyl}-1-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
3-methoxy-N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]propanamide
3-[(1S,5R)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1H-indazole
2-methoxy-4-(2-methoxypyridin-3-yl)pyridine-3-carbonitrile
5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-N-ethyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3-carboxamide
1-{2-methylthieno[2,3-d]pyrimidin-4-yl}-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
(3R,4R)-1-(5-fluoro-2-methylbenzoyl)-3-methyl-4-(oxan-4-yl)piperidin-4-ol
3-chloro-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-4-propoxybenzamide
1-methyl-3-propyl-N-[(1R)-2,2,2-trifluoro-1-phenylethyl]-1H-pyrazole-5-carboxamide
4-({2-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}methyl)-1-phenyl-1H-1,2,3-triazole
2-(dimethyl-1,2-oxazol-4-yl)-6,8-dimethoxy-4-methylquinoline
2-[2-(1H-indol-4-yl)-4-methylphenoxy]acetamide
(2S,4S)-4-amino-1-[3-(3-hydroxyquinoxalin-2-yl)propanoyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]piperidin-3-amine
2-oxo-6-phenyl-N-(2,3,4,5-tetrahydro-1-benzoxepin-4-ylmethyl)-1,2-dihydropyridine-3-carboxamide
1-cyclopentyl-5-{[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1H-imidazole
3-{[1-({7-oxo-4H,7H-[1,2,4]triazolo[1,5-a]pyrimidin-5-yl}methyl)pyrrolidin-3-yl]methyl}benzoic acid
propan-2-yl 4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carboxylate
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-ethyl-1,2-oxazole-5-carboxamide
4-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]-N-(3-methoxyphenyl)piperidine-1-carboxamide
1-{2-[2-(2-methylphenyl)pyrrolidine-1-carbonyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl}ethan-1-one
3-(2-chlorophenyl)-1-(4-methoxyphenyl)-4-(pyrrolidin-1-ylmethyl)-1H-pyrazole
{3-[(4-chlorophenyl)methyl]-9-(oxan-4-yl)-3,9-diazaspiro[5.5]undecan-1-yl}methanol
5-{[(3S,4R)-3-(dimethylamino)-4-(propan-2-yl)pyrrolidin-1-yl]methyl}-N-propylpyrimidin-2-amine
N-[4-(2,2-dimethylpropanamido)-3-methoxyphenyl]-2-methoxypyridine-4-carboxamide
N-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)-3-(piperidin-3-yl)benzamide
3-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-1-[4-(propylsulfamoyl)phenyl]urea
N,N-dimethyl-4-(4-{[2-(3-phenylpiperidin-1-yl)ethyl]amino}piperidin-1-yl)benzamide
[2-(1H-1,3-benzodiazol-2-yl)ethyl]({[2-(3,4-dimethoxyphenyl)-7-methoxyquinolin-3-yl]methyl})amine
(1S,4S)-N-[4-(4-chlorophenoxy)phenyl]-5-methyl-2,5-diazabicyclo[2.2.1]heptane-2-carboxamide
N-[1-(2,3-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-methylpiperidine-4-carboxamide
1-tert-butyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)-5-oxopyrrolidine-3-carboxamide
(3S,4R)-4-(4-methoxyphenyl)-N,N-dimethyl-1-(6-methylpyridine-2-carbonyl)pyrrolidin-3-amine
N-[(4-methyl-2-propyl-1,3-thiazol-5-yl)methyl]-2-oxo-1,2-dihydroquinoline-4-carboxamide
7,8-dimethyl-3-{[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]methyl}-3,4-dihydroquinazolin-4-one
2-[1-(4-chlorophenyl)-3-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-[(5-methylpyrazin-2-yl)methyl]acetamide
(3S,9aR)-8-(4-chlorobenzoyl)-3-[(4-chlorophenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
(3R,4S)-4-[4-(4-{[(4-methylphenyl)amino]methyl}benzoyl)-1,4-diazepan-1-yl]oxolan-3-ol
N-[(2-methoxyphenyl)methyl]-1,3,5-trimethyl-N-(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
2-(2-fluorophenyl)-2-hydroxy-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethan-1-one
9-[3-(4-chloro-1H-pyrazol-1-yl)propanoyl]-2-[2-(dimethylamino)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
[(2S,6S)-4-[(4-chloro-3-fluorophenyl)methyl]-11-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-6-yl]methanol
5-hydroxy-N-[(3R,5S)-5-[(propan-2-yl)carbamoyl]-1-(pyrimidin-2-yl)pyrrolidin-3-yl]pyrazine-2-carboxamide
2-[(3R,4R)-3-{[ethyl(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4,6-bis(propan-2-yl)phenol