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N-(2-propoxypropyl)-2-propyl-1,3-thiazole-4-carboxamide
(1S,3R)-3-amino-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]cyclopentane-1-carboxamide
2-cyclopentyl-9-[5-(propan-2-yl)-1,3,4-thiadiazol-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-hydroxyadamantan-1-yl)-N-[1-(3-methylbutan-2-yl)-1H-pyrazol-5-yl]acetamide
3-ethyl-4-{2-[(isoquinolin-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-1-methylpiperazin-2-one
4-benzyl-3-butyl-1-[2-(2-methylpyrrolidin-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-chloro-1-methyl-3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]-1H-indazole
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-4-oxo-3,4-dihydrophthalazine-1-carboxamide
N-[3-(4-methoxyphenyl)propyl]-6-[(oxan-4-yl)amino]pyridine-3-carboxamide
N-[(2-methoxyphenyl)methyl]-1-methyl-3-(piperidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-[1-(furan-2-yl)ethyl]-N-methylbenzamide
N-[(3S,4R)-1-[3-(4-fluorophenoxy)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
4-methoxy-2-{8-methyl-2,8-diazaspiro[4.5]decane-2-carbonyl}phenol
5-methyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-4-phenylthiophene-3-carboxamide
5-methanesulfonyl-N-(3-methoxypropyl)-4-(piperidin-3-yl)pyrimidin-2-amine
2-[1-({1-[(1S,2R)-2-butylcyclopropanecarbonyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]propan-2-amine
3-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1-methyl-1,2-dihydropyridin-2-one
[1-({1-[1-(3-methylphenyl)piperidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]methanol
(3S,4R)-N,N-dimethyl-1-(5-methyl-1-benzofuran-2-carbonyl)-4-propylpyrrolidin-3-amine
5-ethyl-N-{[1-(2-methoxyethyl)pyrrolidin-3-yl]methyl}-N-methylpyrimidin-2-amine
3-{5-[(1-phenyl-1H-pyrazol-5-yl)methyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-(pyrimidin-2-yloxy)-N-(4-sulfamoylphenyl)piperidine-1-carboxamide
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N'-(3,5-dimethylphenyl)propanediamide
(3aS,6aS)-2-[4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carbonyl]-5-propyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-butyl-4-[(4-fluorophenyl)methanesulfonyl]-1-methylpiperazin-2-one
6-[3-(pyrazin-2-yl)-1H-pyrazol-1-yl]pyridin-2-amine
5-methoxy-4-(1-methyl-1H-pyrazol-5-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)pyrimidin-2-amine
3-(2,3-dimethylquinoxalin-6-yl)-1-methyl-1-[1-(pyridin-2-yl)propan-2-yl]urea
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-{[methyl(1,2-oxazol-5-ylmethyl)amino]methyl}piperidin-2-one
4-(3,5-dimethyl-1-benzofuran-2-yl)-7-hydroxy-6-methoxy-1,2,3,4-tetrahydroquinolin-2-one
2-methyl-4-[4-({methyl[(1-methyl-1H-imidazol-2-yl)methyl]amino}methyl)phenyl]butan-2-ol
4-(4-fluorophenoxy)-1-(5-methyl-1,3-oxazole-4-carbonyl)piperidine
1-[4-(1H-1,2,3,4-tetrazol-1-yl)butanoyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-(2,1,3-benzoxadiazol-5-ylmethyl)-N,2,5-trimethyl-4-oxo-3H,4H-thieno[2,3-d]pyrimidine-6-carboxamide
ethyl 6-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}pyridine-3-carboxylate
(4aS,7aR)-1-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-4-(2-methoxyacetyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]benzamide
N-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-6-{octahydropyrrolo[1,2-a]piperazin-2-yl}pyridine-3-carboxamide
(1S,5R)-6-(cyclopropanesulfonyl)-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-[2-(2-fluorophenyl)-1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]ethyl]-N-methyl-3-(methylsulfanyl)propanamide
N-[4-methyl-2-(1-methylcyclopropaneamido)phenyl]benzamide
1-({3-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]phenyl}methyl)-1H-pyrazole
2-methyl-2-(methylamino)-N-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}propanamide
4-[(4-fluorophenyl)methyl]-3-[2-oxo-2-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethyl]piperazin-2-one
6-(3-phenyl-1H-pyrazole-5-carbonyl)-1-(4-phenylpiperazine-1-carbonyl)-6-azaspiro[2.5]octane
4-(2-methylphenoxy)-1-[2-(pyrrolidin-1-yl)acetyl]piperidine-4-carboxylic acid
(3S,5S,9R)-5-[(quinolin-5-ylmethyl)amino]-1,7-diazatricyclo[7.3.0.03,7]dodecane-2,8-dione
2-tert-butyl-6-{2,8-diazaspiro[4.5]decan-2-ylmethyl}phenol
N-[1-(3,4-dimethylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(2-methyl-1H-imidazol-1-yl)propanamide
(2S,4R)-4-cyclohexaneamido-N-ethyl-1-(2-phenylethyl)pyrrolidine-2-carboxamide