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1-{3-[4-(2-methylphenyl)piperazin-1-yl]piperidin-1-yl}-2-phenylethane-1,2-dione
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[2-(dimethylamino)pyrimidin-5-yl]methyl}pyrrolidin-3-yl]methanol
6-{[2-(4-hydroxypiperidin-1-yl)ethyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
1,2-dimethyl-N-{[1-(pyridin-3-ylmethyl)pyrrolidin-3-yl]methyl}-1H-imidazole-4-sulfonamide
4-[(2R)-5-oxopyrrolidine-2-carbonyl]-1-(2-phenylphenyl)piperazin-2-one
(2R,6S)-2,6-dimethyl-4-(1-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}piperidin-4-yl)morpholine
1-(3,4-dimethoxybenzoyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
3-[3-({[2-(1H-imidazol-1-yl)-1-phenylethyl]amino}methyl)-1H-indol-1-yl]propanamide
1-[cyclohexyl(methyl)amino]-3-{3-[(3,3,4-trimethylpiperazin-1-yl)methyl]phenoxy}propan-2-ol
dimethyl[(4-{1-[1-(propan-2-yl)piperidine-4-carbonyl]pyrrolidin-2-yl}phenyl)methyl]amine
3-{3-oxo-3-[3-(pyridin-3-yl)azetidin-1-yl]propyl}-3,4-dihydroquinazolin-4-one
4-chloro-2-[4-(pyrrolidin-3-yl)piperazine-1-carbonyl]phenol
2,3-difluoro-5-[4-(2-hydroxyphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]phenol
(1R,9aR)-1-{[(2-hydroxyethyl)[(2E)-3-phenylprop-2-en-1-yl]amino]methyl}-octahydro-1H-quinolizin-1-ol
3-ethoxy-N-ethyl-N-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}benzamide
2-{[6-(3-chloro-2-fluorophenyl)pyrimidin-4-yl]amino}ethan-1-ol
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-(cyclopent-3-en-1-yl)propanamide
7-cyclopropanecarbonyl-N,N-dimethyl-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
2-[9-(5-methylthiophene-3-carbonyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-{[2-(2,3-difluoro-4-methylphenoxy)pyridin-3-yl]methyl}-1-methyl-6-oxo-1,6-dihydropyridazine-3-carboxamide
2-(3-fluorophenyl)-1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]piperidine
1-cyclopentyl-N-(3,4-dimethylphenyl)piperidin-3-amine
1-[(2-ethylpyrimidin-4-yl)methyl]-4-phenylazepane
1-[4-(benzyloxy)piperidin-1-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
3-(4-chloro-1H-pyrazol-1-yl)-N-methyl-N-{[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl}propanamide
9-(2-amino-6-methylpyrimidine-4-carbonyl)-2-(3-methoxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
2-({[(3-tert-butyl-1H-pyrazol-5-yl)methyl]amino}methyl)-8-chloroquinolin-4-ol
1-(3-{[3-(dimethylamino)propyl](methyl)amino}piperidin-1-yl)-2-(phenylsulfanyl)ethan-1-one
(3-{[(furan-2-ylmethyl)(prop-2-en-1-yl)amino]methyl}-2,4,6-trimethylphenyl)methanol
5-(1-benzothiophen-3-yl)pyridine-3-carboxamide
2-(ethylsulfanyl)-1-{4-[(3-methylphenyl)methyl]piperazin-1-yl}propan-1-one
7-(3-chlorophenyl)-4-(5-hydroxypyridine-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
2-[4-(4-chlorophenyl)butanoyl]-2,7-diazaspiro[4.5]decan-6-one
N-cyclopentyl-4-{7H-pyrrolo[2,3-d]pyrimidin-4-yl}-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(3-cyclopropyl-1-methyl-1H-pyrazol-5-yl)-2-[3-(pyrimidin-5-yl)-1H-indazol-1-yl]acetamide
(2S,4S)-4-[2-(dimethylamino)acetamido]-1-(4,6-dimethylpyridine-3-carbonyl)-N-ethylpyrrolidine-2-carboxamide
N-methyl-3-(1-methyl-1H-pyrazol-4-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
methyl (2S)-2-{[1-(furan-2-ylmethyl)piperidin-4-yl]formamido}propanoate
{3-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-9-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
1-[(3-methoxyphenyl)methyl]-4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
N,N-dimethyl-2-[4-(3,4,5-trimethoxyphenyl)phenyl]acetamide
3-[(4-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}piperidin-1-yl)methyl]pyridine
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]phenyl}-3-[3-(1H-1,2,4-triazol-1-yl)propyl]urea
1-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]propane-1,2-dione
N-{2-[3-(hydroxymethyl)piperidin-1-yl]ethyl}-5-(3-methoxyphenyl)furan-2-carboxamide
5-(butylamino)-N,N-dimethyl-1-(2-methylpropyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-({1-[(2E)-2-methyl-3-phenylprop-2-en-1-yl]pyrrolidin-3-yl}methyl)-1,3-oxazole-5-carboxamide
[(3R,4R)-4-(azepan-1-ylmethyl)-1-(1-propyl-1H-pyrazole-5-carbonyl)pyrrolidin-3-yl]methanol
3-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]-1-methyl-4,5,6,7-tetrahydro-1H-indazole