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2-{1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}ethan-1-ol
(2R,3R,6R)-3-(4-methylphenyl)-5-(1-methylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[(2R,3R,6R)-3-(2-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(1-ethyl-3-methyl-1H-pyrazol-4-yl)methyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
1-(2-aminoethyl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
1-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-4-(3-methylpyridin-2-yl)piperazine
(2S,4S)-4-amino-N-ethyl-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidine-2-carboxamide
ethyl 1-[2-(3-methylpyridin-2-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
4-(2-phenylethyl)-1-(quinoxalin-2-yl)piperidine-4-carboxylic acid
4-[(3-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}phenyl)methyl]piperidine
3-(3-methyl-2-oxo-2,3-dihydro-1,3-benzoxazol-6-yl)-1-[2-(1,2,3,4-tetrahydroquinolin-1-yl)ethyl]urea
(2S)-2-(dimethylamino)-1-[(3S)-3-ethylmorpholin-4-yl]-3-phenylpropan-1-one
N-[2-(2-oxo-1,3-oxazolidin-3-yl)phenyl]-3-(1H-pyrazol-3-yl)piperidine-1-carboxamide
2-[3-(methoxymethyl)piperidin-1-yl]-4-(4-methylphenyl)-5-(pyridin-3-yl)pyrimidine
2-(5-chloro-1H-1,3-benzodiazol-2-yl)-N-[1-(pyridin-4-yl)propyl]acetamide
2-(pyridin-4-yl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]quinoline-4-carboxamide
2-butyl-5-[5-(1,3-dimethyl-1H-pyrazol-5-yl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
5-(3-acetylphenoxymethyl)-N-methyl-N-(pyridin-3-ylmethyl)-1H-pyrazole-3-carboxamide
5-({5-[2-(methylsulfanyl)ethyl]-4-phenyl-1H-imidazol-1-yl}methyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-cyclopropanecarbonyl-N-[1-(4-fluorophenyl)piperidin-4-yl]piperidine-4-carboxamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-methyl-2-oxo-4-(pyridin-3-yl)-1,2,3,4-tetrahydropyrimidine-5-carboxamide
5-(4-hydroxy-4-phenylpiperidine-1-carbonyl)-2,3-dimethylbenzene-1-sulfonamide
3-{5-[2-(1H-indol-3-yl)ethyl]-1,3,4-oxadiazol-2-yl}-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]propan-1-one
(1R,5R)-6-(1H-imidazol-4-ylmethyl)-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
(2S,3R)-2-amino-3-hydroxy-N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)butanamide
ethyl 1-(7-chloroquinolin-4-yl)-5-({[3-(morpholin-4-yl)propyl]amino}methyl)-1H-pyrazole-4-carboxylate
3-{5-[(2,3-difluorophenyl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
5-[3-(methoxymethyl)piperidine-1-carbonyl]-N-methyl-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyridin-2-amine
(2R,3R,6R)-3-(4-methoxyphenyl)-5-[2-(methylsulfanyl)pyrimidin-4-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
[(3R,4R)-4-[(dimethylamino)methyl]-1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]pyrrolidin-3-yl]methanol
1-(2-methylpropyl)-4-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]-1,4-diazepane
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(2-methylphenyl)methyl]-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(dimethylamino)-N-[3-(dimethylamino)-2,2-dimethylpropyl]-2-(4-methylphenyl)acetamide
7-[(3S)-3-phenylbutanoyl]-2-(pyridin-4-yl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{1-[(4-methoxyphenyl)methyl]-1H-pyrazol-4-yl}-2-{methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}acetic acid
(3S,4S)-1-[(3-ethyl-1H-pyrazol-5-yl)methyl]-4-(naphthalen-2-yl)piperidin-3-ol
1-[3-(3-methoxyphenyl)phenyl]-3-[4-(methylamino)butyl]urea
2-[5-(piperidin-1-ylmethyl)-1,2,4-oxadiazol-3-yl]pyridine
N-ethyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-{[2-(prop-2-en-1-yloxy)phenyl]methyl}acetamide
N-(1-{1-[(2-methoxyphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)pyridine-3-carboxamide
N-benzyl-N-ethyl-3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]propanamide
[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]({1-[1-(furan-2-carbonyl)piperidin-4-yl]-2-phenylethyl})methylamine
3-{2-[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
6-(2-fluoro-4-methoxyphenyl)-7-methyl-N-[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
1-[4-(azepan-1-yl)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]-4-(4-chlorophenyl)piperidin-4-ol
N-(2-hydroxyethyl)-3-(1,2-oxazinan-2-yl)-N-[(2E)-3-phenylprop-2-en-1-yl]propanamide
1-(oxolan-2-ylmethyl)-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperazine
3-[1-(adamantan-1-yl)piperidin-4-yl]-N-(2-chlorophenyl)propanamide
8-[2-(2,5-dimethylphenyl)acetyl]-2-(2-hydroxyethyl)-2,8-diazaspiro[5.5]undecan-3-one