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5-[4-(furan-2-ylmethyl)-3-(2-hydroxyethyl)piperazine-1-carbonyl]pyrazin-2-ol
2-{4-[(3,4-dimethoxyphenyl)methyl]-1-[(2-methylphenyl)methyl]piperazin-2-yl}ethan-1-ol
2-ethyl-4-[2-(2-methoxy-4-methylphenoxy)ethyl]-1-(propan-2-yl)piperazine
(4aS,7aR)-4-(1H-imidazol-2-ylmethyl)-6,6-dioxo-N-phenyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
2-[5-(2,6-difluoro-4-methoxyphenyl)-3-(furan-2-yl)-1H-1,2,4-triazol-1-yl]acetic acid
N'1-[(1-cyclopentylpiperidin-3-yl)methyl]-N'1-[2-(piperidin-1-yl)ethyl]cyclopropane-1,1-dicarboxamide
5-methyl-1'-{2H,3H-thieno[3,4-b][1,4]dioxine-5-carbonyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
5-methyl-3-{3-oxo-3-[(1S,6R)-4-oxo-3,9-diazabicyclo[4.2.1]nonan-9-yl]propyl}-2,3-dihydro-1,3-benzoxazol-2-one
1-[2-(4-chlorophenyl)ethyl]-6-oxo-N-[2-(propan-2-yloxy)ethyl]piperidine-3-carboxamide
1-(1,3-dihydro-2-benzofuran-5-yl)-3-[1-(thiophen-3-yl)propan-2-yl]urea
2-[2-(2-oxopyrrolidin-1-yl)ethyl]-N-[2-(propan-2-yl)phenyl]piperidine-1-carboxamide
ethyl 1-[(5-{[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]carbamoyl}-6-oxo-1,6-dihydropyridin-2-yl)methyl]piperidine-3-carboxylate
3-({2-[(5-methylpyrazin-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-9-yl}methyl)benzonitrile
(1S,4R)-2-{[1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}-2-azabicyclo[2.2.1]heptan-3-one
N-[1-(3-methylpyridin-2-yl)propan-2-yl]-2,3-dihydro-1H-inden-2-amine
1-[1-(2-methyl-1-benzofuran-5-carbonyl)piperidin-4-yl]-N-(propan-2-yl)piperidine-4-carboxamide
methyl 2-[4-(2-phenylethyl)piperidine-1-carbonyl]piperidine-1-carboxylate
(4S,4aS,8aS)-4-phenyl-1-(pyridazine-4-carbonyl)-decahydroquinolin-4-ol
4,4-difluoro-N-[4-(1H-imidazol-1-yl)phenyl]piperidine-1-carboxamide
7-(2-hydroxyethyl)-2-[2-(methylsulfanyl)pyrimidin-4-yl]-2,7-diazaspiro[4.5]decan-6-one
2-amino-6-(1-methyl-1H-pyrrol-3-yl)-4-(3-methylthiophen-2-yl)pyridine-3-carbonitrile
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
8-[4-(dimethylamino)butanoyl]-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
4-({5-[(2H-1,3-benzodioxol-5-ylmethyl)carbamoyl]-6-oxo-1,6-dihydropyridin-2-yl}methyl)morpholine-2-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methyl-1-(piperidin-3-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
methyl (2S,4R)-1-[(3,5-dimethoxyphenyl)methyl]-4-[4-(trifluoromethyl)benzamido]pyrrolidine-2-carboxylate
N-{[5-(methylsulfanyl)-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl]methyl}thiophene-2-carboxamide
6-(azepane-1-carbonyl)-5-methyl-N-(prop-2-en-1-yl)thieno[2,3-d]pyrimidin-4-amine
2-(cyclopentylmethyl)-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
(1S,5S)-3-[(7-methoxy-2H-1,3-benzodioxol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
5-[3-(4-fluorophenoxymethyl)piperidine-1-carbonyl]-1H-1,2,3-benzotriazole
2-(2,4-difluorophenoxy)-1-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethan-1-one
N-[3-(3-fluorophenyl)phenyl]-1-[(4-hydroxyphenyl)methyl]piperidine-4-carboxamide
(3aS,6aS)-2-methyl-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(2-methyl-6-propylpyrimidin-4-yl)-N-[(3-methyloxetan-3-yl)methyl]piperidin-4-amine
1-methanesulfonyl-4-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-(1,3-dihydroxypropan-2-yl)-1-[(4-methylphenyl)methyl]piperazin-2-one
3,7-dimethyl-11-(pyrazine-2-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
4-({3-[2-hydroxy-3-(piperidin-1-yl)propoxy]-4-methoxyphenyl}methyl)piperazin-2-one
N-cyclopropyl-3-{methyl[3-(1-methyl-1H-imidazol-2-yl)propyl]sulfamoyl}benzamide
1-[1-(3-methylbutyl)-3-(morpholine-4-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(4-methylphenoxy)ethan-1-one
(3aS,6aS)-2-[(dimethyl-1H-1,2,4-triazol-5-yl)methyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-benzyl-5-[(2,2,2-trifluoro-1-phenylethoxy)methyl]-1H-1,2,4-triazole
N-[2-({[2-(3-methylphenyl)pyrimidin-5-yl]methyl}amino)ethyl]pyridine-3-carboxamide
N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methyl-3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamide
2-(6-aminopyridin-3-yl)-2-[methyl({[3-(trifluoromethyl)phenyl]methyl})amino]acetic acid
2-(dimethylamino)-8-[4-(1H-pyrazol-1-ylmethyl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
2-methyl-N-(4-pentanamidophenyl)-1H-1,3-benzodiazole-4-carboxamide
methyl({[1-(2-phenylethyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl})[1-(1,3-thiazol-2-yl)ethyl]amine
methyl[(3-phenyl-1,2-oxazol-5-yl)methyl][1-(pyrazin-2-yl)propan-2-yl]amine