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3-(4-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}piperazin-1-yl)pyrazine-2-carbonitrile
1-[1-(4-fluorophenyl)-3,5-dimethyl-1H-pyrazole-4-carbonyl]-N,N-dimethylazepan-4-amine
1-[({[4-(3-chlorophenyl)-5-[(3-hydroxypropyl)sulfanyl]-4H-1,2,4-triazol-3-yl]methyl}(methyl)amino)methyl]naphthalen-2-ol
4-[3-(cyclopropylmethyl)-3-(hydroxymethyl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
({4-cyclopropyl-5-[1-(5-ethyl-1,3,4-thiadiazol-2-yl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
2-[5-(2-chloro-6-fluorophenoxymethyl)-1,2,4-oxadiazol-3-yl]pyridine
1-benzyl-8-(pyridin-2-ylmethyl)-3-[3-(pyridin-3-yl)propyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
ethyl 1-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
(4aS,7aR)-4-[(5-methylfuran-2-yl)methyl]-6,6-dioxo-N-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
1-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-methoxyethan-1-one
1-(furan-2-carbonyl)-4-{[3-(6-methoxynaphthalen-2-yl)-1H-pyrazol-4-yl]methyl}piperazine
({5-[1-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
benzyl N-[(3S,7S,8aS)-3-ethyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]carbamate
2-acetyl-8-(2,6-diaminopyrimidin-4-yl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}propan-1-one
(3aR,6aS)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(1H-1,3-benzodiazol-2-ylmethyl)-4-(furan-3-ylmethyl)-1,4-diazepan-6-ol
5-methyl-1-{[1-phenyl-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-(2-phenylpropyl)-8-(1,3-thiazol-4-ylmethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-(3-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-oxopropyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
4-(4-chlorophenyl)-N-(quinolin-3-ylmethyl)butanamide
1-{2-[1-(3,5-difluoropyridine-2-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
N-cyclopentyl-3-{[2-(1H-imidazol-1-yl)propyl]sulfamoyl}benzamide
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-5-(morpholin-4-yl)-2,3-dihydropyridazin-3-one
(2S,4S)-1-(2,3-dihydro-1H-inden-2-yl)-N-(2-methoxyethyl)-4-[(naphthalen-1-ylmethyl)amino]pyrrolidine-2-carboxamide
6-chloro-3-({2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}methyl)-4H-chromen-4-one
3-{[(1H-imidazol-2-ylmethyl)carbamoyl]methyl}-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-amino-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1H-1,2,4-triazole-5-carboxamide
(1H-indol-4-ylmethyl)(methyl){[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
1-[6-amino-2-(pyrrolidin-1-yl)pyrimidin-4-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-2-({[2-(methylsulfanyl)phenyl]formamido}methyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
4-(4-butyl-1H-1,2,3-triazol-1-yl)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)piperidine
2-[1-(4-fluorophenyl)-5-[5-(pyrrolidin-1-ylmethyl)furan-2-yl]-1H-1,2,4-triazol-3-yl]acetamide
3-ethoxy-1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}propan-1-one
N-cyclopropyl-3-[1-(1-propylpiperidin-4-yl)piperidin-3-yl]propanamide
1-benzyl-3-(2,3-dihydro-1H-inden-5-yl)-1-(1,1-dioxo-1λ6-thiolan-3-yl)urea
1-methyl-2-oxo-8-[2-(phenylsulfanyl)ethyl]-1,8-diazaspiro[4.5]decane-4-carboxylic acid
6-(2,5-dimethoxyphenyl)quinoline
2-amino-4-[2-(methoxymethyl)pyrimidin-5-yl]-5-methyl-6-(4-methylphenyl)pyridine-3-carbonitrile
[(4-chloro-1-methyl-1H-indazol-3-yl)methyl](methyl)[(4-methyl-1H-imidazol-2-yl)methyl]amine
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-4-(4-methylpiperazin-1-yl)pentanamide
3-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]-1-(2-propoxybenzoyl)piperidine
[4-benzyl-1-(2-chloro-4-fluorobenzenesulfonyl)piperidin-4-yl]methanol
N-ethyl-2-[(3-methoxyphenyl)amino]-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}butanamide
1-[3-(1H-pyrazol-1-yl)benzoyl]-4-(thiophen-2-ylmethyl)-1,4-diazepane
2-(3-hydroxypropyl)-8-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-2,8-diazaspiro[5.5]undecan-3-one
methyl (2S)-2-phenyl-2-({[(pyrazin-2-yl)carbamoyl]methyl}amino)acetate
N,N-dimethyl-6-(3-{[4-(propan-2-yl)phenyl]amino}piperidin-1-yl)pyrazine-2-carboxamide
(2S)-2-acetamido-3-{1-[6-(trifluoromethyl)pyridin-3-yl]-1H-imidazol-4-yl}propanoic acid
1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]-3-(1H-pyrazol-5-yl)piperidine