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N-{[1-(2-methylpropyl)cyclobutyl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(4aR,7aS)-4-[(3-hydroxyphenyl)methyl]-N,N-dimethyl-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxamide
(4aR,7aS)-1-cyclobutanecarbonyl-4-(4-methyl-1H-pyrrole-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(2-{[2-(methylcarbamoyl)piperidin-1-yl]methyl}phenoxy)acetic acid
8-(4-hydroxybenzoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-cyclopentyl-1-{4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}ethan-1-one
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-2-[1-(3-methylbut-2-en-1-yl)-3-oxopiperazin-2-yl]acetamide
3-{1-[3-(3-hydroxy-3-methylbutyl)benzoyl]piperidin-3-yl}propanamide
2-(4-{1-[(3-chlorophenyl)methyl]-1H,4H-pyrazolo[3,4-d]imidazol-5-yl}-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-ol
N-(1-cyclohexyl-3-methyl-1H-pyrazol-5-yl)-2-(7-fluoro-1H-indol-1-yl)acetamide
6-({[(8-methoxyquinolin-5-yl)methyl](methyl)amino}methyl)-1,4-oxazepan-6-ol
8-(5-acetyl-4-methylpyrimidin-2-yl)-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-amino-4-(isoquinolin-5-yl)-5-methyl-6-(1-methyl-1H-pyrazol-4-yl)pyridine-3-carbonitrile
2-chloro-6-methoxy-3-({[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl](prop-2-en-1-yl)amino}methyl)phenol
N-(cyclopent-3-en-1-yl)-2-ethyl-7-(oxolane-2-carbonyl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
6-(cyclopropylmethoxy)-1-[(3-methoxyphenyl)methyl]-4-[(3-phenyl-1H-pyrazol-4-yl)methyl]-1,4-diazepan-2-one
3-fluoro-6-methyl-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)imidazo[1,2-a]pyridine-2-carboxamide
1-[4-(morpholin-4-yl)-3-(1,2,3,6-tetrahydropyridin-4-yl)phenyl]ethan-1-one
6-methyl-2-(2-phenylethyl)-3-(4-propylpiperazine-1-carbonyl)-1-(pyridin-4-ylmethyl)-1,4-dihydropyridin-4-one
(2R,3R)-3-{[2-(5-methylthiophen-2-yl)ethyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[7-(3,6-dimethylpyrazin-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanamide
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(cyclopropylmethyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-{[6-(dimethylamino)pyridin-3-yl]methyl}-2,7-diazaspiro[4.5]decan-6-one
(1R,7S)-6-(azepane-1-carbonyl)-3-[(3-methoxyphenyl)methyl]-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
3-[5-(2-oxo-1,2,3,4-tetrahydroquinoline-4-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanoic acid
1-[(2-chlorophenyl)methyl]-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{1-[2-(dimethylamino)ethyl]-5-oxopyrrolidin-2-yl}ethyl)-2-methyl-1,3-benzothiazole-6-carboxamide
3-hydroxy-3-{[4-(methylamino)piperidin-1-yl]methyl}-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-[(4-chlorophenyl)methyl]-N-methyl-N-[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
6-ethyl-3-[(3S,4R)-3-ethyl-4-hydroxy-4-methylpiperidine-1-carbonyl]-1,5-dimethyl-1,2-dihydropyridin-2-one
(1-{[1-(2-methylpropyl)-1H-1,3-benzodiazol-2-yl]methyl}pyrrolidin-3-yl)methanamine
N-{[(2R,3R,5S)-2-(2-fluorophenyl)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
2-amino-4-(2H-1,3-benzodioxol-5-yl)-6-(1H-pyrrol-2-yl)pyridine-3-carbonitrile
N-cyclopentyl-1-ethyl-3-methyl-N-[(2-methylphenyl)methyl]-1H-pyrazole-4-carboxamide
2-{1-[(2-chloro-4-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-cyclooctylacetamide
N-{[4-(2-methylpropoxy)phenyl]methyl}-2-(1H-pyrazol-1-yl)-N-(pyridin-4-ylmethyl)acetamide
N3-cyclopentyl-1-(2-methylpropyl)-4-oxo-N5-(prop-2-en-1-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-[(4-methyl-5-{[(2-methyl-1,3-thiazol-4-yl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)methyl]piperidine
(3S,9aR)-3-benzyl-8-(2-fluorobenzenesulfonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(1-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2H-1,3-benzodioxole-5-carboxamide
(1S,5R)-6-[5-(ethylsulfanyl)thiophene-2-carbonyl]-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
[(1R,3S,3aS,6aR)-5-benzyl-3-[4-(1H-imidazol-1-yl)phenyl]-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
2-{4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-6-methylpyridine-3-carboxamide
(3S,4R)-4-(2-methoxyphenyl)-1-{[(1s,4s)-4-aminocyclohexyl]methyl}pyrrolidine-3-carboxylic acid
4-[2-(1H-1,2,3-benzotriazol-1-yl)ethyl]-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2(7),5-trien-3-one
N-[(2S)-1-hydroxy-3-(1H-indol-3-yl)propan-2-yl]-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
3,3,3-trifluoro-1-(3-{[4-(thiophen-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)propan-1-one
1-(2-aminoethyl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-1,2,3-triazole-4-carboxamide
2,6-dimethyl-4-{1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}quinoline
N-[(4,6-dimethylpyrimidin-2-yl)methyl]-2-(morpholin-4-yl)-2-(pyridin-3-yl)acetamide