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8-[2-(2,4,7-trimethyl-1H-indol-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}propan-1-one
1-[7-(hydroxymethyl)-9-(2-methoxyethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-(methylsulfanyl)ethan-1-one
4-(3-hydroxy-3-methylbutyl)-N-(4,5,6,7-tetrahydro-1H-indazol-5-yl)benzamide
3-[(3R,4S)-1-(5-chloro-3-fluoropyridin-2-yl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2S,4R)-4-amino-1-{2-[(2R,6S)-2,6-dimethylpiperidin-1-yl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-[2-(1,3-benzoxazol-2-yl)ethyl]-1-[3-(1,3-thiazol-4-yl)phenyl]piperidin-4-amine
1-({1-[(3,5-dichlorophenyl)methyl]pyrrolidin-3-yl}methyl)-3-ethylurea
2-(dimethylamino)-N-[(3R,4R)-3-hydroxypiperidin-4-yl]-4-methylpyrimidine-5-carboxamide
2-(2,3-dihydro-1H-indol-1-yl)-N-[(3S,4R)-4-ethoxyoxolan-3-yl]-2-oxoacetamide
4-[(2,3-difluorophenyl)methyl]-3-[2-(4-hydroxypiperidin-1-yl)-2-oxoethyl]piperazin-2-one
2-chloro-N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-5-(trifluoromethyl)benzamide
N-[(5-fluoro-1H-indol-2-yl)methyl]-N-methyl-2-(methylamino)acetamide
1-[4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)piperidin-1-yl]-2-ethylbutan-1-one
9-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-amino-1-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
2-[({6-chloro-2-methylimidazo[1,2-a]pyridin-3-yl}methyl)(furan-2-ylmethyl)amino]butan-1-ol
7-{[3,3-bis(hydroxymethyl)piperidin-1-yl]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
5-(2-methoxypyridin-3-yl)pyridine-2-carbonitrile
1-{2-[2-(dimethylamino)ethyl]morpholin-4-yl}-4-(4-fluorophenyl)butan-1-one
N-[2-(1-methylpiperidin-2-yl)ethyl]-6-[(oxan-4-yl)amino]pyridine-3-carboxamide
(2S,4S)-N-ethyl-4-(5-methoxyfuran-2-amido)-1-(pyridin-3-ylmethyl)pyrrolidine-2-carboxamide
2-[5-(2-ethylpyrimidin-4-yl)-4-phenyl-1H-imidazol-1-yl]-1-phenylethan-1-ol
(4aR,7aS)-1-acetyl-4-[(4-fluorophenyl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(3,5-difluorophenyl)ethyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
1-{[3,5-dimethyl-1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}-3-(4-methoxy-3,5-dimethylbenzoyl)piperidine
6-methyl-N-(2-{2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}ethyl)imidazo[2,1-b][1,3]thiazole-5-carboxamide
1-[(3S,5R)-3-(hydroxymethyl)-5-(pyrrolidin-1-ylmethyl)piperidin-1-yl]-4-(1H-pyrazol-4-yl)butan-1-one
N-({3-[2-(4-fluorophenyl)ethoxy]phenyl}methyl)-N-(pyridin-4-ylmethyl)cyclopropanecarboxamide
2-{8-butyl-9-oxo-2,8-diazaspiro[5.5]undecan-2-yl}pyridine-3-carboxamide
N-[1-(morpholine-4-carbonyl)piperidin-4-yl]pyrazine-2-carboxamide
5-[({2-methylpyrido[2,3-d]pyrimidin-4-yl}amino)methyl]-1,3,4-thiadiazol-2-amine
7-fluoro-2-methyl-N-[1-(pyrazin-2-yl)piperidin-4-yl]quinoline-4-carboxamide
5-[1-(piperidin-1-yl)ethyl]-N-[2-(pyridin-2-ylsulfanyl)ethyl]furan-2-carboxamide
2-{4-[(4-ethyl-6-hydroxy-1,4-diazepan-1-yl)methyl]phenoxy}acetamide
3-chloro-N-cyclopentyl-4-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-(3-methoxyphenyl)-3-[1-(pyridin-3-ylmethyl)piperidin-4-yl]propanamide
1-[(1R,2S,3S,4R,5S)-tricyclo[3.2.1.02,4]octane-3-carbonyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N,N-dimethyl-4-[1-(2-phenylethyl)pyrrolidin-3-yl]piperidine-1-sulfonamide
3-oxo-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-3,4-dihydroquinoxaline-2-carboxamide
N-[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]-2-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
(1R,3S)-N1,N1,2,2,3-pentamethyl-N3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]cyclopentane-1,3-dicarboxamide
N-{[5-(dimethylcarbamoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}quinoxaline-6-carboxamide
3-(azepane-1-carbonyl)-5-(2-ethylpiperidine-1-carbonyl)-1-(2-methylpropyl)-1,4-dihydropyridin-4-one
N-[2-methoxy-2-(thiophen-2-yl)ethyl]-4-methyl-2-phenylpyrimidine-5-carboxamide
methyl (2S,4R)-4-(dimethylamino)-1-{2-[(4-methylphenyl)carbamoyl]acetyl}pyrrolidine-2-carboxylate
({5-methyl-2-[4-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)(oxolan-2-ylmethyl)(pyridin-4-ylmethyl)amine
3-{[(1R,2R,4S)-bicyclo[2.2.1]heptan-2-yl]sulfamoyl}-N-methyl-N-[2-(methylsulfanyl)ethyl]benzamide
1-[6-(4-methoxy-3,5-dimethylphenyl)pyridin-3-yl]ethan-1-one
N-(2H-1,3-benzodioxol-5-ylmethyl)-5-propyl-N-(pyridin-3-ylmethyl)-1,2-oxazole-3-carboxamide