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2-(1H-imidazol-1-yl)-1-[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
1-[(3ar,6ar)-octahydropyrrolo[3,4-c]pyrrole-3a-carbonyl]-4-phenylpiperidine-4-carbonitrile
2-{1-[(6-methylpyridin-2-yl)methyl]-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
N-ethyl-1,3-dimethyl-N-[(2-methylphenyl)methyl]-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N-ethyl-3-(3-fluorophenyl)-N-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1H-pyrazole-4-carboxamide
1-[4-(3,6-dimethylpyrazin-2-yl)piperazin-1-yl]-3-[(2-methoxyethyl)(methyl)amino]propan-1-one
1-benzyl-8-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-3-(2-methoxyethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-cyclobutyl-5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
4-(1-benzofuran-2-ylmethyl)-1-[(3-methoxyphenyl)methyl]piperazin-2-one
3-(2-methoxyethyl)-1-[2-(4-methoxyphenyl)ethyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
5-{2-[4-(dimethylamino)piperidin-1-yl]pyrimidin-4-yl}-2-ethoxybenzoic acid
4-[3-(1-ethyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2-methyl-6-(2-methylpropyl)pyrimidine
1-methyl-1'-[2-(morpholin-2-yl)acetyl]-1,2-dihydrospiro[indole-3,4'-piperidine]-2-one
[benzyl(methyl)sulfamoyl]({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl})amine
2-(5-cyano-4,6-dimethylpyridin-2-yl)-N,N-bis(propan-2-yl)benzamide
3-{5-[1-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-1-methyl-1H-1,2,4-triazol-3-yl}pyridine
methyl 3-{[(3-fluorophenyl)formamido]methyl}-5-(furan-2-amido)benzoate
N-[(4-fluoro-3-methylphenyl)methyl]-7-(pyridine-3-carbonyl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
(3S,4S)-4-propyl-1-(1H-1,2,3-triazol-4-ylmethyl)pyrrolidine-3-carboxylic acid
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-methyl-1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
7-methyl-4-(2-{1-oxa-7-azaspiro[3.5]nonan-7-yl}-2-oxoethyl)-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-({4-[(2-ethoxyphenyl)methyl]-3-(2-hydroxyethyl)piperazin-1-yl}methyl)-5-methoxyphenol
2-methyl-6-[4-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]-2H,3H,5H,6H,7H,8H-[1,2,4]triazolo[4,3-a]pyridin-3-one
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-4-phenylbutanamide
1-({4-[2-(4-fluorophenyl)azetidine-1-carbonyl]phenyl}methyl)-3,5-dimethyl-1H-pyrazole
N-[2-(4-amino-6-hydroxypyrimidin-2-yl)ethyl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
N,N-dimethyl-2-[(1S,5R)-6-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]acetamide
3-[4-(adamantan-1-yl)piperazine-1-carbonyl]-1-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-2,6-dimethyl-1,4-dihydropyridin-4-one
N-[3-(4-fluorophenyl)propyl]-3-(1-methylpiperidin-2-yl)propanamide
(3S,9aR)-3-benzyl-8-(3,5-difluorobenzoyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-[(2-methoxyphenyl)methyl]-5-methyl-6-(morpholine-4-carbonyl)thieno[2,3-d]pyrimidin-4-amine
(butan-2-yl)({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl})(pyridin-3-ylmethyl)amine
1-[(1S,5R)-3-acetyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-(5-fluoro-2-methyl-1H-indol-3-yl)ethan-1-one
(4aS,8aR)-1-(2-aminoethyl)-6-(2-methyl-1-benzofuran-5-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{[(3-ethyl-1,2-oxazol-5-yl)methyl](methyl)amino}-N-phenylbutanamide
N-[(3R,5S)-5-[(1R,3s,6r,8S)-4-azatricyclo[4.3.1.13,8]undecane-4-carbonyl]pyrrolidin-3-yl]furan-2-carboxamide
N-(furan-3-ylmethyl)-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(1s,4s)-4-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}cyclohexan-1-ol
methyl 4-[({1-[1-(2,4-difluorophenyl)-5-methyl-1H-pyrazol-4-yl]ethyl}amino)methyl]benzoate
(2S)-2-{2-[3-(2-hydroxyethoxy)phenyl]-1H-imidazol-1-yl}-3-methylbutanamide
3-[1-(1,3-oxazole-5-carbonyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
(4aS,8aR)-6-(2-aminopyridine-4-carbonyl)-1-propyl-decahydro-1,6-naphthyridin-2-one
1-{7-[(4-fluorophenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-2-{5H,6H-imidazo[2,1-b][1,3]thiazol-3-yl}ethan-1-one
4-{1-[(2-butyl-5-chloro-1H-imidazol-4-yl)methyl]pyrrolidin-2-yl}-3,5-dimethyl-1,2-oxazole
(1R)-2-{3-[3-(2-methylpyridin-4-yl)phenyl]-1H-pyrazol-1-yl}-1-phenylethan-1-ol
3-[(2R,3R,6R)-3-(4-methylphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecane-5-carbonyl]-1H-pyrazol-5-amine
1-[2-(3-methyl-1,2-oxazol-5-yl)ethyl]-3-[(2-methyl-1H-imidazol-1-yl)methyl]piperidine
2-[4-benzyl-3-(2-hydroxyethyl)piperazin-1-yl]-1,3-thiazole-4-carboxamide
2-[4-(1H-pyrazol-5-yl)phenyl]-3-(pyrrolidin-1-yl)pyrazine