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N-[(5-chloro-2-methoxyphenyl)methyl]-N-methyl-5-(oxolan-2-yl)thiophene-2-carboxamide
N-(oxolan-3-ylmethyl)quinoxalin-6-amine
2-(2H-1,3-benzodioxol-5-yl)-N-[(3R,4S)-1-cyclopentanecarbonyl-4-cyclopropylpyrrolidin-3-yl]acetamide
N-({3-methyl-7-[(2E)-3-phenylprop-2-enoyl]-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-2-(phenylsulfanyl)acetamide
2-{9-[3-(4-hydroxyphenyl)propanoyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetamide
N-(3-chloro-4-fluorophenyl)-3-[1-(5-methyl-1,2-oxazole-3-carbonyl)piperidin-4-yl]propanamide
3-(cyclopropylmethyl)-1-(thiophen-2-ylmethyl)piperidine-3-carboxylic acid
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-2-(methylamino)pyridine-4-carboxamide
methyl({4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}){[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}amine
N-[(2-fluorophenyl)methyl]-4-[4-(2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)piperidin-1-yl]benzamide
methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]{[5-methyl-2-(thiophen-2-yl)-1,3-oxazol-4-yl]methyl}amine
2-ethyl-9-(5-fluoropyridine-3-carbonyl)-4-phenyl-2,9-diazaspiro[5.5]undecane
N-(furan-2-ylmethyl)-N,1-dimethyl-5-[methyl(1,3-thiazol-4-ylmethyl)amino]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
4-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
N-[2-(1,4-dioxo-1,2,3,4-tetrahydrophthalazin-2-yl)ethyl]-5-methyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
2-ethoxy-3-[3-(4-phenyl-1H-pyrazol-5-yl)piperidine-1-carbonyl]pyridine
2-[2-(1H-imidazol-4-yl)ethyl]-8-(5-methyl-1,3-oxazole-4-carbonyl)-2,8-diazaspiro[5.5]undecan-3-one
3,3-dimethyl-1-[(3S,4R)-1-(1-methyl-6-oxo-1,6-dihydropyridazine-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-yl]urea
ethyl 5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1-(3,3,3-trifluoropropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}-N-[4-(1,3-thiazol-4-yl)phenyl]piperidine-3-carboxamide
N-methyl-3-phenoxy-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
3-{3-cyclobutyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}-4,5,6,7-tetrahydro-1-benzofuran-4-one
1-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-3-yl)piperazine
1-[(6-methylquinolin-5-yl)methyl]piperidine-3-carbonitrile
3-chloro-N-[(2-fluorophenyl)methyl]-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzamide
N-[4-({methyl[1-(2-phenylethyl)piperidin-3-yl]amino}methyl)phenyl]acetamide
N-(1,3-benzothiazol-2-ylmethyl)-2-(dimethylamino)-N,4-dimethylpyrimidine-5-carboxamide
1-(2-phenylquinazolin-4-yl)-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
2-{2-ethyl-3-oxo-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}-N-(propan-2-yl)acetamide
N-{[7-methoxy-2-(3-methylphenyl)quinolin-3-yl]methyl}-N-(2-methoxyethyl)-2H-1,3-benzodioxole-5-carboxamide
2-{4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]piperidine-1-carbonyl}pyridine
1'-{[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]methyl}-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{5-[3-(1H-pyrazol-1-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}pyridine
4-(2,4-dimethoxyphenyl)-2-methyl-5H,6H,7H-cyclopenta[d]pyrimidine
2-[3-(1H-imidazol-1-ylmethyl)piperidin-1-yl]-N-methylpyrimidin-4-amine
4-[(3R,4S)-3-amino-4-(4-methoxyphenyl)pyrrolidine-1-carbonyl]-6-ethyl-1,2-dihydropyridin-2-one
1-{[(3R,4R)-1-(4-chloro-3-fluorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
1-ethyl-8-(1-methoxypropan-2-yl)-3-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]-1-[4-(methylsulfanyl)butan-2-yl]piperidine
(4aR,8aR)-2-(pyrrolidine-1-carbonyl)-7-(quinoxalin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
1-[(1-methyl-1H-pyrazol-4-yl)methyl]-3-(4-phenoxybenzoyl)piperidine
N-(2-methoxyethyl)-1,3-dimethyl-N-(1,3-thiazol-2-ylmethyl)-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(1R,5R)-6-(cyclopropylmethyl)-3-[3-(1H-imidazol-2-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-1-({2-[(propan-2-yl)amino]pyrimidin-5-yl}methyl)-4-propylpyrrolidin-3-yl]methanesulfonamide
(4aS,8aR)-1-[2-(methylamino)ethyl]-6-(1,3-thiazole-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-(1,1-dioxo-2,3-dihydro-1λ6-thiophen-3-yl)-4-methyl-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
2-(3-fluorophenyl)-N-[1-(pyrrolidine-1-carbonyl)azepan-3-yl]acetamide
N-(2-{4-methyl-5H,6H,7H-cyclopenta[d]pyrimidin-2-yl}ethyl)-3-(trimethyl-1H-pyrazol-4-yl)propanamide
N-[2-hydroxy-3-(pyrrolidin-1-yl)propyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-(2-chloro-4-fluorophenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-hydroxypiperidin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one