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[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]({[2-(4-methoxyphenyl)pyrimidin-5-yl]methyl})methylamine
6-methyl-3-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-1,2-dihydropyridin-2-one
3-{5-[(2-fluorophenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
2-ethyl-8-(2-methyl-4-phenylpyridine-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
2,3,5-trimethyl-N-[2-(1H-1,2,3-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
1-{3-[5-(4-fluorophenyl)-2-methylpyrimidin-4-yl]piperidin-1-yl}-2-(thiophen-2-yl)ethan-1-one
1-{[1-(4-methoxyphenyl)-1H-imidazol-2-yl]methyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
(4aR,7aS)-1-[(5-methylfuran-2-yl)methyl]-4-(5-methylthiophene-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[4-({4-[(2-chlorophenyl)methyl]-5-oxo-1,4-diazepan-1-yl}methyl)phenyl]acetamide
N-(1-cyclopentyl-1H-pyrazol-5-yl)-2-{4-[6-(dimethylamino)pyrimidin-4-yl]-1H-pyrazol-1-yl}acetamide
N-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]propan-2-yl}thiophene-2-carboxamide
N-[(3S,4R)-1-(1,3-dihydroxypropan-2-yl)-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
1-[(3aS,6aS)-5-(2-{5H,6H,7H-[1,3]thiazolo[3,2-a]pyrimidin-3-yl}acetyl)-octahydropyrrolo[3,4-b]pyrrol-1-yl]pentan-1-one
4-(3-methyl-1H-1,2,4-triazol-5-yl)-N-[3-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
4-{5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}-2-(2-methylpropyl)morpholine
N4-[(7-methoxy-2,3-dihydro-1,4-benzodioxin-6-yl)methyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
N-cyclooctyl-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidin-1-yl]-2-(3-methoxyphenyl)ethan-1-one
4-({9-hydroxy-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-5-methyl-1-(4-methylphenyl)piperazin-2-one
5-fluoro-N-[2-(pyrazin-2-yl)ethyl]quinazolin-4-amine
1-(3-chlorobenzoyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
4-(5-{[(2-hydroxyethyl)({[4-(methylsulfanyl)phenyl]methyl})amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
{4-[(4-chlorophenyl)methyl]-1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]piperidin-4-yl}methanol
4-[4-(2-phenylpropyl)piperazin-1-yl]-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
N-[(2-chlorophenyl)methyl]-3-{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]piperidin-3-yl}propanamide
propan-2-yl (4aS,7aR)-4-[(4-methyl-1H-imidazol-5-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazine-1-carboxylate
1-[(4-methanesulfonylphenyl)methyl]-2-methyl-1,4-diazepan-5-one
8-chloro-2-({[2-(pyridin-2-yl)ethyl]amino}methyl)quinolin-4-ol
N-[2-(dimethylamino)-1-phenylethyl]-N,1-dimethyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
N-benzyl-N-(2-hydroxyethyl)-1-(2-methoxyethyl)-6-oxopiperidine-3-carboxamide
1-[(3S,4R)-1-[1-(4-methoxyphenyl)cyclopropanecarbonyl]-4-(propan-2-yl)pyrrolidin-3-yl]-3,3-dimethylurea
1-[2-(8-fluoroquinolin-2-yl)-1H-imidazol-1-yl]propan-2-ol
4-(cyclopropylmethyl)-1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-3-(propan-2-yl)-1,4-diazepan-5-one
2-methyl-4-(4-{[(2S)-2-(piperidine-1-carbonyl)pyrrolidin-1-yl]methyl}phenyl)butan-2-ol
N-ethyl-N-[(4-methoxyphenyl)methyl]-5-(propan-2-yl)-1,2-oxazole-3-carboxamide
2-(2H-1,2,3-benzotriazol-2-yl)-N-[2-(pyridin-4-yl)ethyl]acetamide
2-[(4aS,7aR)-4-(2-methoxyacetyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-(1-methyl-1H-pyrazol-4-yl)acetamide
1-[(3-chloro-4-fluorophenyl)methyl]-4-(pyrrolidin-3-yl)piperazine
N-(3-chlorophenyl)-3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carboxamide
(3S,4R)-1-[2-(5-amino-3-methyl-1H-pyrazol-1-yl)acetyl]-4-phenylpyrrolidine-3-carboxylic acid
(3aR,6aR)-2-benzyl-N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
3-[4-(2-methoxyphenyl)-2-methylpiperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
6-methoxy-2-oxo-N-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
5,5-dimethyl-3-{2-oxo-2-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}imidazolidine-2,4-dione
2-{3-[({5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-yl}amino)methyl]piperidin-1-yl}ethan-1-ol
2-(1-methyl-1H-pyrazol-4-yl)-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]quinoline-4-carboxamide
2-[7-(hydroxymethyl)-9-(1H-pyrazole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-ol
5-(4-{1-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-1H-1,2,3-triazol-4-yl}phenyl)-2H-1,2,3,4-tetrazole
1-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]piperidine-3-carboxamide
6-fluoro-3-(1H-1,2,4-triazol-5-ylmethyl)-3,4-dihydroquinazolin-4-one