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(4aR,7aS)-1-(2-hydroxyethyl)-4-[5-(methoxymethyl)thiophene-2-carbonyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[(4aR,7aS)-4-(1H-1,3-benzodiazol-2-ylmethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
1-(1H-1,3-benzodiazole-2-carbonyl)-4-(1H-imidazol-1-yl)piperidine-4-carboxylic acid
N-(1-{1-[(4-fluorophenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-3-phenoxypropanamide
2-{1-[(3,5-dimethoxyphenyl)methyl]-4-{[3-(methylsulfanyl)phenyl]methyl}piperazin-2-yl}ethan-1-ol
2-(1-benzothiophen-7-yl)-1,3-thiazole-4-carboxamide
N-{[5-(furan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
N-[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]-2-(1H-pyrazol-1-yl)butanamide
[(3R,4S)-1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}pyrrolidin-3-yl]methanol
1-methyl-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-2-oxo-6-(propan-2-yl)-1,2-dihydropyridine-3-carboxamide
5-[3-(2-methylpropyl)-1H-pyrazol-5-yl]-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(2-methoxyphenyl)-3-[1-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
5-methyl-1-(oxan-4-yl)-5-phenylpiperidin-2-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
N-benzyl-N-(3-hydroxy-2-methylpropyl)-2-[1-(propan-2-yl)piperidin-4-yl]acetamide
2-{1-benzyl-4-[3-(1H-pyrazol-1-yl)propyl]piperazin-2-yl}ethan-1-ol
6-[3-(4-fluorophenoxymethyl)piperidin-1-yl]pyrimidin-4-amine
4-{3-[2-(3,4-difluorophenyl)ethyl]piperidine-1-carbonyl}-1,2-dihydroquinolin-2-one
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-phenyl-1,2-oxazole-4-carbonyl)piperidine
N-methyl-3-(5-methylthiophen-2-yl)-N-[2-(pyridin-2-yl)ethyl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[(1-propyl-1H-imidazol-2-yl)methyl]amine
4-ethyl-1-(3-phenyl-1,2-oxazole-5-carbonyl)-1,4-diazepan-5-one
N-(2-fluoro-4-{5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-6-yl}phenyl)acetamide
N-[3-(3-benzyl-1H-1,2,4-triazol-5-yl)propyl]acetamide
4-({1-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
5-(3-methyl-1-benzofuran-2-yl)-4-phenyl-1-(pyrrolidin-3-yl)-1H-imidazole
ethyl 1-{[2-(2-hydroxyethoxy)phenyl]methyl}-3-(2-phenoxyethyl)piperidine-3-carboxylate
1-ethyl-N-{[4-(2-phenylethyl)-4H-1,2,4-triazol-3-yl]methyl}-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
1-methyl-4-[3-(6-methylpyridazin-3-yl)-1,2,4-oxadiazol-5-yl]-1,2-dihydroquinolin-2-one
({3-[(3,4-dimethoxyphenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)(methyl){[1-(piperidin-1-yl)cyclohexyl]methyl}amine
1-tert-butyl-5-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-3-methyl-1H-1,2,4-triazole
N-[1-(1-methyl-1H-imidazol-2-yl)butyl]-2-(2,4,7-trimethyl-1H-indol-3-yl)acetamide
2-(2-hydroxyethyl)-9-[4-(trifluoromethyl)pyridin-2-yl]-2,9-diazaspiro[5.5]undecan-3-one
N,3,6-trimethyl-N-{[3-(1H-1,2,3,4-tetrazol-5-yl)phenyl]methyl}-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
4-{6-[4-(1H-imidazol-2-yl)piperidin-1-yl]pyrazine-2-carbonyl}morpholine
5,5-dimethyl-3-{2-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
6-[4-(2-hydroxyethyl)-1H-pyrazol-1-yl]-2-methylquinolin-4-ol
N,4-dimethyl-2-(4-methylpiperazin-1-yl)-N-[1-(pyridin-3-yl)propyl]pyrimidine-5-carboxamide
1-[2-(5-methyl-1H-pyrazol-1-yl)acetyl]-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
5-{1-[2-(3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
1-[3-(morpholine-4-carbonyl)-1-(3-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-2-(thiophen-2-yl)ethan-1-one
4-[4-(3-methoxybenzoyl)piperazin-1-yl]-6-(propan-2-yloxy)pyrimidin-2-amine
1-ethyl-3-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepin-2-ylmethyl}piperidine
N-[2-(3-carbamoylpiperidin-1-yl)ethyl]-7-fluoro-2-methylquinoline-4-carboxamide
8-(2-ethoxyacetyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3,3,3-trifluoro-1-[3-(hydroxymethyl)-3-(3-methoxypropyl)piperidin-1-yl]propan-1-one
N-[1-(4-methoxyphenyl)-6,6-dimethyl-4,5,6,7-tetrahydro-1H-indazol-4-yl]-4-(1H-1,2,4-triazol-1-yl)butanamide
(1R,3S)-3-ethoxy-7-{[2-(propylamino)pyrimidin-5-yl]methyl}-7-azaspiro[3.5]nonan-1-ol