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N-[4-(3-methoxyphenoxy)phenyl]-3-(propoxymethyl)pyrrolidine-1-carboxamide
3-[5-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-2-yl]pyridine
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[4-(morpholin-4-ylmethyl)piperidin-1-yl]ethan-1-one
N4-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-2,4-diamine
2-{1-[2-(2-oxo-1,3-oxazinan-3-yl)ethyl]-4-phenyl-1H-imidazol-5-yl}benzonitrile
2-{5-[2-(3-methyl-1,2,4-oxadiazol-5-yl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
[2-(azepan-1-yl)ethyl](ethyl){[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]methyl}amine
8-methyl-4-{octahydro-1H-pyrrolo[1,2-a][1,4]diazepine-2-carbonyl}-2-(1H-pyrazol-4-yl)quinoline
1-[2-(2-oxopyrrolidin-1-yl)acetyl]-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-cyclopentyl-N-{[(2S,4S)-4-fluoro-1-(1H-pyrrole-2-carbonyl)pyrrolidin-2-yl]methyl}acetamide
1-{4-[(2-hydroxy-3-methoxypropyl)amino]-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}ethan-1-one
2-methyl-3-(2-{[6-(piperidin-4-yl)pyrimidin-4-yl]amino}ethyl)-1H-indole-5-carbonitrile
1-[(1S,6R)-3,9-diazabicyclo[4.2.1]nonan-3-yl]-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]ethan-1-one
4-{2-[4-(furan-2-ylmethyl)piperazin-1-yl]-2-oxoethyl}-3-methyl-1-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N'1-[(3R,4S)-1-(furan-2-ylmethyl)-4-(propan-2-yl)pyrrolidin-3-yl]cyclopropane-1,1-dicarboxamide
3-[(3R,4S)-1-[(6-chloropyridin-3-yl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propanoic acid
(2S)-2-amino-4-methyl-1-[3-(4-phenylphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]pentan-1-one
(1R,5R)-N,N-dimethyl-6-({9-methyl-4-oxo-4H-pyrido[1,2-a]pyrimidin-2-yl}methyl)-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-{[4-(1H-imidazol-1-yl)phenyl]methyl}-4-(oxan-4-yl)piperazine
2-[3-methyl-5-oxo-4-(2-phenylethyl)-4,5-dihydro-1H-1,2,4-triazol-1-yl]-N-[2-(5-methylfuran-2-yl)ethyl]acetamide
3-{[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-4-yl]methyl}-6-methoxy-1,2-dihydroquinolin-2-one
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-4-(4H-1,2,4-triazol-3-yl)piperidine
N-[1-(4-chlorophenyl)cyclobutyl]-2-oxo-1-oxaspiro[4.5]decane-4-carboxamide
1-(4-{2-[4-(3-{[methyl(thiophen-3-ylmethyl)amino]methyl}phenoxy)piperidin-1-yl]-2-oxoethyl}phenyl)imidazolidin-2-one
N-[1-(1H-imidazol-2-yl)ethyl]-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridin-2-amine
N-{2-chloro-4-[2-(trimethyl-1H-pyrazol-1-yl)acetamido]phenyl}propanamide
N-(4-methanesulfonylphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
4-(1-methylpyrrolidin-3-yl)-1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}piperidine
[(3R,4R)-1-(4-methoxy-3-methylbenzoyl)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]pyrrolidin-3-yl]methanol
3-(3-hydroxy-3-methylbutyl)-N-[1-(morpholin-4-ylmethyl)cyclopentyl]benzamide
3-(1-{[1-methyl-3-(4-phenoxyphenyl)-1H-pyrazol-4-yl]methyl}piperidin-2-yl)propan-1-ol
N-{1-[1-(4,5,6,7-tetrahydro-1-benzothiophene-3-carbonyl)piperidin-4-yl]-1H-pyrazol-5-yl}cyclopropanecarboxamide
N-{[5-chloro-7-(pyridin-4-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carboxamide
N-{1-[1-(4-methoxyphenyl)-1H-pyrazol-4-yl]ethyl}-3-(1H-pyrazol-1-yl)benzamide
3-[(3R,4S)-1-[(3-methoxyphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
N-({7-[4-(4-fluorophenyl)-4-oxobutanoyl]-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl}methyl)-3-methylthiophene-2-carboxamide
[(1-ethyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)[3-(methylsulfanyl)propyl]amine
10-methoxy-5-[(3-methyl-1,2-oxazol-5-yl)methyl]-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
4-{5-[3-(trifluoromethyl)phenoxymethyl]-1H-pyrazole-3-carbonyl}thiomorpholine
1-{[6-(azocane-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}piperidine-3-carboxamide
(4aS,7aR)-1-(5-chloro-2-methylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
4-(5-methoxyfuran-2-carbonyl)-2-(naphthalen-1-ylmethyl)morpholine
N-methyl-4-[(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]-1,3-thiazol-2-amine
3-{[5-(1-phenyl-1H-pyrazol-4-yl)-1H,4H-pyrazolo[3,4-d]imidazol-1-yl]methyl}pyridine
N-(9H-fluoren-9-yl)-2-propyl-1,3-thiazole-4-carboxamide
N-[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-7-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
N-[(3R,5S)-1-(cyclohexylmethyl)-5-(ethylcarbamoyl)pyrrolidin-3-yl]-1-methyl-1H-pyrazole-3-carboxamide
1-(3-{[(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)amino]methyl}phenyl)ethan-1-one
(4aS,8aR)-1-[3-(1H-imidazol-1-yl)propyl]-6-[(3-methyl-1,2-oxazol-5-yl)methyl]-decahydro-1,6-naphthyridin-2-one
7-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide