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4,4,4-trifluoro-1-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]butan-1-one
[(5-fluoro-1-methyl-1H-indol-2-yl)methyl](methyl)[3-(1-methyl-1H-imidazol-2-yl)propyl]amine
1,4,6-trimethyl-N-[4-(5-methylfuran-3-amido)phenyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
7-[3-methyl-5-(phenoxymethyl)furan-2-carbonyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-{[3-(2H-1,3-benzodioxol-5-ylmethyl)-3-methylpiperidin-1-yl]methyl}-5-methoxypyridin-4-ol
4-{1-[4-(4-fluorophenyl)-5-methylpyrimidin-2-yl]-5-(thiophen-2-yl)-1H-pyrazole-4-carbonyl}thiomorpholine
3-ethyl-1-[(2-fluoro-5-methoxyphenyl)methyl]piperidine-3-carboxylic acid
2-[({5-[1-(3,6-dimethylpyrazin-2-yl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)(methyl)amino]ethan-1-ol
2-{3-cyclopropyl-5-[2-(pyrrolidin-1-ylmethyl)-1,3-thiazol-5-yl]-1H-1,2,4-triazol-1-yl}-3-methylpyridine
1-[(3-methoxyphenyl)methyl]-4-[3-(1H-pyrazol-1-ylmethyl)benzoyl]piperazine
(3S,4S)-4-cyclopropyl-1-[4-methyl-2-(methylamino)-1,3-thiazole-5-carbonyl]pyrrolidine-3-carboxylic acid
3-({[(4-fluorophenyl)methyl](1-hydroxybutan-2-yl)amino}methyl)phenol
N-({2-[4-(pyridin-2-yl)piperazin-1-yl]pyridin-3-yl}methyl)thiophene-2-carboxamide
[3-(3-methoxypropyl)-1-(oxan-4-yl)piperidin-3-yl]methanol
1-(2-{1-[(2,6-dichloro-3-hydroxyphenyl)methyl]piperidin-4-yl}ethyl)pyrrolidin-2-one
5-(3-methyl-1,2,4-oxadiazol-5-yl)-N-[1-(pyridin-3-yl)propan-2-yl]pyridin-2-amine
(4aR,7aS)-1-ethyl-4-(9H-fluoren-2-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-1H-indole
2-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-1,2,3,4-tetrahydroisoquinolin-4-ol
N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}-2,4,5-trimethylbenzamide
8-[(1-butyl-1H-1,3-benzodiazol-2-yl)methyl]-2-cyclopropyl-1,3,8-triazaspiro[4.5]dec-1-en-4-one
1-{[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-ol
5-(2-fluoro-3-methoxyphenyl)-1-(2-methanesulfonylethyl)-4-phenyl-1H-imidazole
1-(2,3-dihydro-1-benzofuran-2-carbonyl)-4-[2-(1H-1,2,4-triazol-1-yl)ethyl]piperazine
2-{[6-(4-chlorophenyl)imidazo[2,1-b][1,3]thiazol-3-yl]formamido}-N-(propan-2-yl)acetamide
3-{[1-(4-chlorophenyl)-3-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}pyridine
7-(morpholine-4-sulfonyl)-N-propyl-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
5-cyclopropyl-4-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1-methyl-1H-pyrazole
1-{2-[methyl(1,3-thiazol-2-ylmethyl)amino]ethyl}piperidin-2-one
N-(butan-2-yl)-3-(2-methylphenyl)-N-(pyridin-4-ylmethyl)propanamide
1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-4-ol
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(pyridin-2-ylmethyl)amino]methyl}piperidin-2-one
2-(3-methoxypropyl)-8-(3-methylpyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
2-[(5-methylpyrazin-2-yl)methyl]-8-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,8-diazaspiro[5.5]undecan-3-one
2-ethyl-5-[4-(pyridin-4-yl)piperidine-1-carbonyl]pyrimidine
3-[5-(1-ethyl-1H-pyrazol-3-yl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-{2-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2,3-dioxo-1,2,3,4-tetrahydroquinoxaline-6-carboxamide
N-methyl-6-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyridine-2-carboxamide
N-({2-[4-(2-methylphenyl)piperazin-1-yl]pyridin-3-yl}methyl)propane-1-sulfonamide
1-(1,2-oxazol-3-ylmethyl)-N-[3-(1H-pyrazol-5-yl)phenyl]piperidine-4-carboxamide
1,3-dimethyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-2-carboxamide
2,2-dimethyl-1-(3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)propan-1-one
6-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-ethyl-5-methylthieno[2,3-d]pyrimidin-4-amine
1,3-dimethyl-2,6-dioxo-N-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,2,3,6-tetrahydropyrimidine-4-carboxamide
N-(oxan-3-yl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
3-(oxolan-3-yl)-5-[3-(1H-pyrazol-1-yl)phenyl]-1,2,4-oxadiazole
6-({[2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)ethyl]amino}methyl)-1,4-oxazepan-6-ol
4-(benzyloxy)-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)butanamide
2-[(dimethylamino)methyl]-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]-1,3-thiazole-4-carboxamide
5-[3-(3-chlorophenyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-1,2,4-triazol-1-yl)propan-2-yl]pyridin-2-amine