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1-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-2-[ethyl(methyl)amino]ethan-1-one
1-(3-methoxyphenyl)-4-{4-oxo-4H-pyrido[1,2-a]pyrimidine-3-carbonyl}piperazin-2-one
3-(3-methoxyphenyl)-1-[(1S,5R)-3-(pyridin-3-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-[2-(azepan-1-yl)ethyl]-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-N-(propan-2-yl)propanamide
3-{1-[(8-fluoro-4-hydroxyquinolin-2-yl)methyl]piperidin-4-yl}-1,3-oxazolidin-2-one
2-(2-methyl-1H-imidazol-1-yl)-1-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}propan-1-one
2-(2,5-difluorophenyl)-2-[2-(1-propylpiperidin-4-yl)acetamido]acetic acid
3-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidin-3-yl)propanamide
5-methanesulfonyl-2-methyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]pyrimidine
1-[6-ethyl-2-(morpholin-4-yl)pyrimidin-4-yl]-N-(oxolan-3-ylmethyl)piperidin-4-amine
5-(3-methoxyphenoxymethyl)-N-(oxolan-2-ylmethyl)-N-propyl-1,2-oxazole-3-carboxamide
3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}[(4-fluorophenyl)methyl]amino)propan-1-ol
2-(adamantan-1-yl)-1-[4-(3-methylpyridin-2-yl)piperazin-1-yl]ethan-1-one
3,3-dimethyl-N-({3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)cyclohexan-1-amine
(3R,4R)-4-(azepan-1-yl)-1-[1-(2-fluorophenyl)piperidin-4-yl]piperidin-3-ol
6-{3,9-diazaspiro[5.6]dodecane-9-carbonyl}-2,3-dihydropyridazin-3-one
1-{3,5-diazatricyclo[9.4.0.02,7]pentadeca-1(11),2(7),3,5,12,14-hexaen-4-yl}-5-(methoxymethyl)-N-[(3-methyl-1,2-oxazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
N-({4-benzyl-5-[(pyridin-4-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}methyl)-4-methoxybenzamide
4-cyclobutaneamido-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methylbenzamide
N-[(3S,4R)-1-(1-acetylpiperidin-4-yl)-4-(4-methoxyphenyl)pyrrolidin-3-yl]acetamide
(2S)-2-[(heptan-4-yl)amino]-3-phenylpropan-1-ol
ethyl 2-{4-[(3-methylphenyl)methyl]piperazin-1-yl}-1,3-oxazole-4-carboxylate
(3R,5S)-5-[4-(2-methylphenyl)-1,4-diazepane-1-carbonyl]pyrrolidin-3-ol
1-(2-ethoxyethyl)-N-[(1-methylcyclohexyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]-1-(1,3-thiazol-2-yl)piperidine
3-[1-(adamantan-2-yl)piperidin-3-yl]-N-[(5-methylfuran-2-yl)methyl]propanamide
1-[1-(2-hydroxyethyl)piperidine-3-carbonyl]-4-phenylpiperidine-4-carbonitrile
5-{pyrazolo[1,5-a]pyridin-7-yl}furan-2-carboxylic acid
N-ethyl-2-(4-fluorophenoxymethyl)-4-hydroxy-N-(pyridin-2-ylmethyl)pyrimidine-5-carboxamide
3-{[1-(4-chlorophenyl)-3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
1-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidine-1-carbonyl}cyclopropane-1-carbonitrile
1-(1H-indazol-7-yl)-3-({1-[(2-methyl-1H-imidazol-1-yl)methyl]cyclopropyl}methyl)urea
(3S,4S)-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}-4-(propan-2-yloxy)pyrrolidin-3-ol
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(4,4,4-trifluorobutyl)piperidine
(2S,4S)-4-amino-1-[(3,5-dimethoxyphenyl)methyl]-N-methylpyrrolidine-2-carboxamide
9-[2-methyl-3-(1H-1,2,4-triazol-1-yl)propanoyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-methyl-2-(methylsulfanyl)-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}pyridine-3-carboxamide
1-(dimethyl-1,3-thiazole-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
(3S,4R)-3-ethyl-4-methyl-1-(2,3,4,9-tetrahydro-1H-carbazole-6-carbonyl)piperidin-4-ol
N-(3-cyano-4-ethoxyphenyl)-4-(thiomorpholin-4-yl)piperidine-1-carboxamide
5-(methoxymethyl)-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
N-{2H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-2-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methylacetamide
4-[3-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)propyl]-1,3-thiazol-2-amine
methyl 4-[6-(methoxymethyl)pyrimidin-4-yl]piperazine-1-carboxylate
2-{[3-(2,4-dimethoxybenzoyl)piperidin-1-yl]methyl}-1H-1,3-benzodiazole
N-[2-(ethanesulfonyl)ethyl]-4-(1H-pyrazol-3-yl)benzamide
N-[1-(2-methylpropyl)cyclopropyl]-1-[4-(1H-pyrazol-1-yl)phenyl]piperidin-4-amine
1-{3-[2-(2,6-difluorophenyl)ethyl]piperidin-1-yl}-2-(2-hydroxyphenoxy)ethan-1-one
N-{1-[1-(cyclohex-3-en-1-ylmethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-2,2-dimethylpropanamide