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(3S,4S)-1-(2-methoxypyridine-4-carbonyl)-4-(morpholin-4-yl)pyrrolidin-3-ol
1-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-3-(1H-imidazol-1-ylmethyl)piperidine
2-[(3R,4R)-3-hydroxy-4-(morpholin-4-yl)piperidin-1-yl]pyridine-4-carboxamide
5-methyl-6-(3-methylpiperidine-1-carbonyl)-N-[(6-methylpyridin-2-yl)methyl]thieno[2,3-d]pyrimidin-4-amine
methyl 2-{[4-(cyclopropylmethyl)-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl]methyl}-1,3-oxazole-4-carboxylate
N-[(8-methoxyquinolin-5-yl)methyl]-N-methyl-1-(propan-2-yl)piperidine-4-carboxamide
2,4-dimethyl-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]-1,3-thiazole-5-carboxamide
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-(prop-2-en-1-yl)-2-(2,5,7-trimethyl-1H-indol-3-yl)acetamide
N-{[3-(4-chlorophenyl)-1H-pyrazol-4-yl]methyl}-2-oxo-1,2-dihydroquinoline-4-carboxamide
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-(1H-imidazol-2-ylmethyl)piperidine-3-carboxamide
4-(ethanesulfonyl)-1-(4-methoxyphenyl)piperazin-2-one
1-[(3-fluorophenyl)methyl]-3-[4-methyl-5-(piperidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
4-[4-(2,1,3-benzoxadiazol-5-ylmethyl)piperazin-1-yl]quinazoline
(2Z)-2-fluoro-1-(3-{5-methyl-2-[(pyridin-3-ylmethyl)sulfanyl]pyrimidin-4-yl}piperidin-1-yl)-3-phenylprop-2-en-1-one
5-(hydroxymethyl)-N-({2-[3-(trifluoromethyl)phenoxy]pyridin-3-yl}methyl)furan-2-carboxamide
6-cyclopentyl-3-{[(6-ethyl-2-methylpyrimidin-4-yl)amino]methyl}-2-methoxy-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
4-[3-(3-methoxyphenoxy)azetidine-1-carbonyl]-1-oxaspiro[4.4]nonan-2-one
N-{4-[2-fluoro-4-(pyrrolidin-1-ylmethyl)phenoxy]phenyl}acetamide
3-{2-[4-(furan-2-carbonyl)piperazin-1-yl]-2-oxoethyl}-1-(3-methoxypropyl)-3-(2-methylphenyl)pyrrolidine-2,5-dione
3-(4-methylpiperazine-1-carbonyl)-1-propyl-N-{[4-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
6-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}pyridine-2-carbonitrile
[1-(1-{[3-(cyclopentyloxy)phenyl]methyl}piperidin-3-yl)piperidin-4-yl]methanol
N6-benzyl-N5-methyl-N5-(1-methylpiperidin-4-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
4-[(1S,5R)-3-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane-6-carbonyl]quinoline
2-methyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]imidazo[1,2-a]pyrimidine-3-carboxamide
2-{3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-3-ol
2-{2-[(4-aminoazepan-1-yl)methyl]phenoxy}ethan-1-ol
N-ethyl-6-[2-(6-methoxynaphthalen-2-yl)morpholin-4-yl]pyridine-3-carboxamide
N-ethyl-2-[(1S,4S)-5-(2-methoxy-5-phenylphenyl)-6-oxo-2,5-diazabicyclo[2.2.1]heptan-2-yl]-N-methylacetamide
3-[1-(1H-indole-6-carbonyl)piperidin-4-yl]-N-(pyridin-3-ylmethyl)propanamide
N-(1,3,4-thiadiazol-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole-2-carboxamide
2-(2-chlorophenyl)-3-methyl-N-(2,2,2-trifluoroethyl)-3H-imidazo[4,5-b]pyridine-6-carboxamide
2-[(3,3-diphenylpiperidin-1-yl)methyl]-5-methoxypyridin-4-ol
5-{[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-3-ethyl-4,5-dihydro-1,2-oxazole
N-(2-methanesulfonamidoethyl)-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
ethyl[(4-methyl-1H-imidazol-2-yl)methyl]{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
1-(carbamoylmethyl)-N-[1-(5-methyl-1,3,4-oxadiazol-2-yl)ethyl]piperidine-4-carboxamide
2-({methyl[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)quinolin-8-ol
1-[2-({2-[(prop-2-en-1-yl)amino]phenyl}formamido)ethyl]piperidine-3-carboxamide
2-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}benzamide
N-ethyl-2-{4-[2-(1H-imidazol-1-yl)acetyl]piperazin-1-yl}acetamide
N-{[3-methoxy-4-(oxolan-3-yloxy)phenyl]methyl}-2-(1H-pyrazol-1-yl)-N-(pyridin-3-ylmethyl)acetamide
1-{2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-2-oxoethyl}-4,6-dimethyl-1,2-dihydropyrimidin-2-one
(3R,4R)-1-cyclobutyl-4-[4-(2-phenylethyl)piperazin-1-yl]piperidin-3-ol
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-5-methyl-1-propyl-1H-pyrazole-4-carboxamide
8-[3-(1H-indol-3-yl)propanoyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
4,5-dimethyl-2-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]propyl}-1H-1,3-benzodiazole
6-(2-methoxyphenyl)-N2-(4-methylphenyl)-1,3,5-triazine-2,4-diamine
3-ethyl-N1-[2-(pyridin-3-yloxy)phenyl]piperidine-1,3-dicarboxamide
N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}-2-(piperidin-1-yl)acetamide