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N3-[(4-fluorophenyl)methyl]-N5-methyl-4-oxo-1-(2-phenylethyl)-1,4-dihydropyridine-3,5-dicarboxamide
[1-(3,6-dimethylpyrazin-2-yl)-3-(2-phenoxyethyl)piperidin-3-yl]methanol
1-(cyclohexylmethyl)-N-methyl-5-{[(3-methyloxetan-3-yl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-methyl-2-{[4-(5-methylpyrimidin-4-yl)piperidin-1-yl]methyl}-1H-indole
N-[3-(4-methoxyphenyl)propyl]-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}-N-(2-fluorophenyl)piperidine-1-carboxamide
(3R,5S)-5-[4-(2-methoxyphenoxy)piperidine-1-carbonyl]pyrrolidin-3-ol
4-hydroxy-1-(8-methoxyquinolin-2-yl)piperidine-4-carboxylic acid
7-fluoro-3-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,2-dihydroquinolin-2-one
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-3-methoxypiperidine
4-({5-[(5-methylthiophen-2-yl)methyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)piperazin-2-one
2-[9-(1-benzofuran-2-ylmethyl)-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
N-{imidazo[1,2-a]pyrimidin-2-ylmethyl}-1-(propan-2-yl)piperidine-4-carboxamide
[1-(5-methyl-1,2-oxazole-4-carbonyl)-3-(prop-2-en-1-yl)piperidin-3-yl]methanol
(1R,7S)-3-[(3,4-dimethylphenyl)methyl]-6-(thiomorpholine-4-carbonyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]({[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl})amine
1-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-(5-{[methyl(propan-2-yl)amino]methyl}-1H-1,2,3,4-tetrazol-1-yl)ethan-1-one
N-{[7-(cyclopent-1-ene-1-carbonyl)-3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl]methyl}-3-ethyl-1-methyl-1H-pyrazole-5-carboxamide
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
1-[2-(1H-pyrazol-1-yl)benzoyl]-1H,2H,3H,4H,6H,10bH-pyrimido[2,1-a]isoindol-6-one
5-{2-[4-(4-methoxyphenoxy)piperidin-1-yl]-2-oxoethyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
3-hydroxy-2-methyl-N-[1-(4-methyl-1,3-thiazol-2-yl)ethyl]benzamide
N-[2-ethyl-1-methyl-5-(2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)-1H-1,3-benzodiazol-7-yl]-2-methoxybenzamide
1-[(dimethyl-1,2-oxazol-4-yl)methyl]-4-[(4-fluorophenyl)methyl]piperidine
(1S,5R)-3-methyl-6-(5-methyl-4-phenylthiophene-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
1-{4-[(2-hydroxy-6-methoxyquinolin-3-yl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
ethyl 1-[3-(1,2-oxazolidin-2-yl)propanoyl]-3-[(2E)-3-phenylprop-2-en-1-yl]piperidine-3-carboxylate
N-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
methyl 5-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-5-oxopentanoate
1-[1-(2-methoxyethyl)piperidine-3-carbonyl]-4-phenylpiperidine-4-carbonitrile
3-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-N-(4-methylphenyl)piperidine-1-carboxamide
4-(2,4-dioxoimidazolidin-1-yl)-N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}benzamide
5-cyclopropyl-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-1,3,4-oxadiazol-2-amine
2-[4-(propan-2-yl)morpholin-2-yl]-1-[4-(pyrimidin-2-yl)piperazin-1-yl]ethan-1-one
2-(4-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}piperazin-1-yl)pyrazine
N-{[2-(dimethylamino)-1,3-thiazol-4-yl]methyl}-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-(6-methyl-2-propylpyrimidin-4-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
4-[(2S,4R)-4-aminopyrrolidine-2-carbonyl]-1-cyclohexylpiperazin-2-one
2-methoxy-6-{[4-(4-methyl-5-{[2-(piperidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl)piperidin-1-yl]methyl}phenol
N,N-diethyl-4-[(1-methoxybutan-2-yl)amino]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-{2-[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}acetamide
7-{2-[4-(pyrimidin-2-yl)piperazin-1-yl]acetyl}-2,7-diazaspiro[4.4]nonane-1,3-dione
2-{imidazo[2,1-b][1,3]thiazol-6-yl}-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
8-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)-5-fluorophenyl]methyl}-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-methyl-N-[1-(3-methylpyridin-2-yl)propan-2-yl]thiophene-2-carboxamide
4-{[1-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)piperidin-3-yl]methyl}morpholine
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-5-[1-(2-methoxyacetyl)pyrrolidin-2-yl]thiophene-2-carboxamide
1-[2-(2-methylphenyl)acetyl]-4-[2-(piperidin-1-yl)ethyl]-1,4-diazepan-5-one
N-cyclopropyl-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide