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7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decane
4-(4-cyclohexylpiperazin-1-yl)-5,6-dimethylpyrimidine
(2S,4R)-4-{[(2-chlorophenyl)methyl]amino}-1-(2-methylpropyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
(3R,4R)-4-ethyl-1-[5-(methoxymethyl)thiophene-2-carbonyl]piperidine-3,4-diol
(4aS,8aR)-1-(2-aminoethyl)-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-decahydro-1,6-naphthyridin-2-one
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-1-{7-methylthieno[3,2-d]pyrimidin-4-yl}piperidin-4-amine
3-(2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)-N-[3-(1H-imidazol-1-yl)propyl]propanamide
5-{[4-(3-methylpyridin-2-yl)piperazin-1-yl]methyl}-2-(thiophen-2-yl)pyrimidine
4-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-N-methylpyrimidin-2-amine
1-(azepan-1-yl)-3-{3-[(2,2-dimethylmorpholin-4-yl)methyl]phenoxy}propan-2-ol
2-methyl-8-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)-2,8-diazaspiro[4.5]decane-3-carboxylic acid
3-(2-oxo-2-{3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}ethyl)-1,2,3-oxadiazol-3-ium-5-olate
1-(1-ethyl-1H-pyrazole-5-carbonyl)-4-[4-ethyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
(3aS,6aS)-2-acetyl-5-{2-[3-(trifluoromethyl)phenyl]acetyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
{[1-(4-chlorophenyl)-3-cyclopropyl-1H-1,2,4-triazol-5-yl]methyl}(methyl)(pyridin-3-ylmethyl)amine
2-[4-(5-methyl-4-{[1-(thiophen-2-yl)propyl]amino}thieno[2,3-d]pyrimidine-6-carbonyl)piperazin-1-yl]ethan-1-ol
4-methyl-6-(4-{[3-(6-methyl-1,3-benzoxazol-2-yl)propyl]amino}piperidin-1-yl)pyrimidin-2-amine
8-[(6-ethoxyquinolin-2-yl)methyl]-1-oxa-8-azaspiro[4.5]decan-3-ol
7-[(2,3-difluorophenyl)methyl]-2-(pyridine-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-2-(pyridin-3-yl)piperidine-1-carboxamide
3-methyl-N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(oxolan-2-ylmethyl)furan-2-carboxamide
2-methyl-N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-(thiophen-2-ylformamido)propanamide
(1S,5R)-6-methyl-3-[2-(4,6,7-trimethyl-1-benzofuran-3-yl)acetyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
7-(3,6-dimethylpyrazin-2-yl)-4-[2-(piperidin-1-yl)ethyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(3-phenyl-1H-pyrazole-4-carbonyl)-4-(1H-pyrrole-2-carbonyl)piperazine
1-[1-(1-methyl-1H-pyrazole-3-carbonyl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-3-carboxamide
1-[2-chloro-5-(morpholin-4-yl)phenyl]-3-ethyl-3-propylurea
2-(3,4-dimethylphenyl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-[2-(3-cyclopropyl-1-phenyl-1H-1,2,4-triazol-5-yl)pyrazolo[1,5-a]pyrimidin-6-yl]ethan-1-ol
9-(3-hydroxy-4-methoxybenzoyl)-2-(2-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(4-chlorophenyl)methyl]-1-(pyrimidin-2-yl)piperidin-3-amine
{2-[(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}urea
3-[5-(2H-1,3-benzodioxol-5-yl)-1,3,4-oxadiazol-2-yl]-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}propanamide
N,2-dimethyl-N-[1-(4-methylpyridin-2-yl)propan-2-yl]-1,8-naphthyridine-3-carboxamide
methyl 3-[(1S,9aR)-octahydro-1H-quinolizin-1-ylmethyl]-9-hydroxy-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
4-[5-(oxolan-2-yl)thiophene-2-carbonyl]thiomorpholine
2-tert-butyl-5-[4-(2-ethylphenyl)piperazine-1-carbonyl]pyrimidin-4-ol
1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-N-{[3-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,N-dimethyl-2-phenyl-2-{[4-(3,3,3-trifluoropropyl)pyrimidin-2-yl]amino}acetamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)thiophene-2-carboxamide
4-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}phenol
1,5,6-trimethyl-N-[4-(methylamino)butyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{2-methyl-4-[(oxolan-3-yl)amino]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl}-2-(1H-1,2,4-triazol-1-yl)ethan-1-one
5-{[4-(3-chloro-5-methylpyridin-2-yl)piperazin-1-yl]methyl}-N-(propan-2-yl)pyrimidin-2-amine
ethyl 2-(methylsulfanyl)-4-[3-(2-oxopyrrolidin-1-yl)piperidin-1-yl]pyrimidine-5-carboxylate
({5-[1-(1H-1,2,3-benzotriazole-5-carbonyl)piperidin-4-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
5-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-methyl-2-[(2-oxo-2-{2-[2-(1H-pyrazol-1-yl)ethyl]piperidin-1-yl}ethyl)sulfanyl]-3,4-dihydropyrimidin-4-one
2-(2-{[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]methyl}-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl)pyridine
5-(3-phenylpropyl)-5-(piperidin-4-yl)-3-(pyridin-3-ylmethyl)imidazolidine-2,4-dione