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N-cyclopentyl-N-({3-[2-(thiophen-2-yl)ethoxy]phenyl}methyl)imidazo[2,1-b][1,3]thiazole-6-carboxamide
N-[(4,6-dimethylpyridin-2-yl)methyl]-N-methyl-5-oxo-1-(pyridin-3-ylmethyl)pyrrolidine-3-carboxamide
3-{1-[5-(2,4-dimethoxyphenyl)-1,2,4-triazin-3-yl]piperidin-3-yl}propan-1-ol
2-(dimethylamino)-2-(3-fluorophenyl)-N-{[3-(trifluoromethyl)phenyl]methyl}acetamide
2-({[1-(2-methoxyethyl)piperidin-4-yl]methyl}(methyl)amino)-2-[4-(propan-2-yloxy)phenyl]acetic acid
N-[2-(3-methoxyphenyl)ethyl]-8-methyl-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(3R,4R)-3-cyclobutyl-4-methyl-1-(1,3,7-trimethyl-1H-indole-2-carbonyl)pyrrolidin-3-ol
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
methyl N-{2-[3-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-2-oxoethyl}carbamate
N-(4-{[ethyl({[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl})amino]methyl}phenyl)acetamide
7-(2-{[1,2,4]triazolo[4,3-b]pyridazin-6-yloxy}acetyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]-4-methylpentane-1,2-dione
(3-{3-[(1R,4S)-2-azabicyclo[2.2.1]heptane-2-carbonyl]pyridin-2-yl}phenyl)methanol
methyl (2S,4R)-4-(2-phenylbenzamido)-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxylate
2-cyclopropyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-1,3-benzodiazole
{[1-(1H-imidazol-1-ylmethyl)cyclopropyl]methyl}(1-methoxypropan-2-yl)amine
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(2-phenylquinazolin-4-yl)pyrrolidin-3-yl]methanol
1-(3-cyclopropyl-1H-pyrazole-5-carbonyl)-2-[2-(thiophen-2-yl)ethyl]piperidine
1-[(4-fluorophenyl)methyl]-3-hydroxy-3-{[methyl(2-methylprop-2-en-1-yl)amino]methyl}piperidin-2-one
2-methanesulfonamido-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]acetamide
[(dimethyl-1,2-oxazol-4-yl)methyl]({imidazo[1,2-a]pyridin-3-ylmethyl})methylamine
1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]-N-(thiophen-3-ylmethyl)piperidine-3-carboxamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}-1,3-oxazole
[(3R,4R)-1-(2-butoxybenzoyl)-4-(morpholin-4-ylmethyl)pyrrolidin-3-yl]methanol
3-[2-(morpholine-4-carbonyl)piperazine-1-carbonyl]-1,2-dihydroquinolin-2-one
N-benzyl-5-(cyclopropylamino)-N,1-dimethyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
(2S,4R)-4-amino-1-[4-(4-methoxyphenyl)butanoyl]-N-methylpyrrolidine-2-carboxamide
2-[(4-chlorophenyl)methyl]-8-[2-(2-hydroxyethoxy)ethyl]-2,8-diazaspiro[4.5]decan-3-one
3-hydroxy-1-(2-methoxyethyl)-3-(1,2,3,4-tetrahydroisoquinolin-2-ylmethyl)piperidin-2-one
N-[(3-chlorophenyl)methyl]-5-[1-(piperidin-1-yl)ethyl]furan-2-carboxamide
(3aS,6aR)-3-[(3,4-dimethoxyphenyl)methyl]-N-ethyl-2-oxo-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazole-5-carboxamide
2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)-N-[1-(cyclohexylmethyl)piperidin-3-yl]acetamide
(2S,4R)-1-benzyl-4-{[(2-chlorophenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-{5-chloro-2-[(1S,6R)-3-methyl-4-oxo-3,9-diazabicyclo[4.2.1]nonane-9-carbonyl]phenyl}propanamide
(1R,5R)-6-benzyl-3-(3,5-difluoropyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
(2S,4R)-4-amino-1-(1-benzothiophene-2-carbonyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
3-(3,5-dimethyl-1H-pyrazol-1-yl)-N-[2-(dimethylamino)ethyl]-N-(oxolan-2-ylmethyl)benzamide
N-[1-(3-methyl-1H-pyrazol-5-yl)propan-2-yl]-2-(pyridin-3-yl)pyrimidine-5-carboxamide
methyl 6-{[4-(2-hydroxyethoxy)phenyl]methyl}-2-[(3-methylbutyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-[4-({3-[2-(methylsulfanyl)benzoyl]piperidin-1-yl}methyl)phenoxy]ethan-1-ol
3,5-dichloro-4-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)azetidin-1-yl]methyl}pyridine
6-(3-fluorophenyl)-N-(3-hydroxy-3-methylbutyl)-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
7-(cyclopropylmethyl)-6-(4-methoxyphenyl)-2-(piperidine-1-carbonyl)-7H,8H-imidazo[1,2-a]pyrazin-8-one
ethyl 2-[4-(2-amino-1,3-benzothiazole-5-carbonyl)piperazin-1-yl]acetate
1-[4-(3-{[(7-methoxy-4-methylquinolin-2-yl)amino]methyl}pyridin-2-yl)piperazin-1-yl]ethan-1-one
[1-(1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-4-yl)piperidin-3-yl]methanol
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
1-methyl-2-[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]azepane
5-(1H-imidazol-4-yl)-4-phenyl-1-[2-(pyrrolidine-1-sulfonyl)ethyl]-1H-imidazole