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(2R,3S,6R)-3-(3,5-difluorophenyl)-N,N-dimethyl-1,5-diazatricyclo[5.2.2.02,6]undecane-5-sulfonamide
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-acetamidoacetamide
1-(2-methoxyphenyl)-3-[1-(1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]urea
(2R,3R)-3-(1H-imidazol-1-yl)-1'-(4-methoxypyrimidin-2-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-(2,4-dimethoxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(morpholin-4-ylmethyl)pyrrolidin-1-yl]ethan-1-one
5-cyclopropanecarbonyl-1'-[(2,2-dimethyloxan-4-yl)methyl]-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
2-{6-hydroxy-4-[2-(morpholin-4-yl)acetyl]-1,4-diazepan-1-yl}pyridine-3-carbonitrile
6-{[(4-methoxy-2,3,6-trimethylphenyl)methyl]amino}-2-methylheptan-2-ol
1-[(4aS,8aS)-4a-hydroxy-7-[(1-methyl-1H-imidazol-2-yl)methyl]-decahydro-2,7-naphthyridin-2-yl]-2-methoxy-2-methylpropan-1-one
(3aS,6aS)-2-(3-ethoxypropanoyl)-5-[(3-methylphenyl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-(but-2-yn-1-yl)-3-[5-(2-cyclohexylethyl)-1,3,4-oxadiazol-2-yl]-N-(furan-2-ylmethyl)propanamide
7-(2-{4H,5H,6H-cyclopenta[d][1,3]thiazol-2-yl}ethyl)-2-oxa-7-azaspiro[4.5]decan-8-one
3-({1-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]cyclopropyl}methyl)-1-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)urea
{1-[(2-chlorophenyl)methyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
N-butyl-2-{1-[2-(ethylamino)pyrimidin-5-yl]-N-methylformamido}acetamide
1-methyl-4-{1-[1-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]ethyl}piperazine
2-methoxy-4-[4-(3-methoxybenzoyl)piperazin-1-yl]pyridine-3-carbonitrile
N-cyclopropyl-4-{methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]sulfamoyl}benzamide
5-{4-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperazin-1-yl}-2-methyl-2,3-dihydropyridazin-3-one
N,1,7-trimethyl-N-(4,5,6,7-tetrahydro-1H-indazol-3-ylmethyl)-1H-indole-2-carboxamide
2-(2,3-difluorophenoxymethyl)-N-methyl-N-(pyridin-2-ylmethyl)-1,3-oxazole-4-carboxamide
N,4-dimethyl-5-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,3-thiazol-2-amine
1-(2-chloroprop-2-en-1-yl)-6,7-dimethoxy-3-{[({3-methylimidazo[2,1-b][1,3]thiazol-6-yl}methyl)amino]methyl}-1,2-dihydroquinolin-2-one
N-{[4-(4-methylphenyl)-5-(pyridin-2-yl)-1H-imidazol-2-yl]methyl}acetamide
3-(1,3-benzoxazol-2-yl)-N-{2-methyl-[1,2,4]triazolo[1,5-a]pyridin-8-yl}piperidine-1-carboxamide
methyl (2S)-1-{1-[(2-methoxyphenyl)methyl]-5-[(3-methylbutyl)carbamoyl]-4-oxo-1,4-dihydropyridine-3-carbonyl}pyrrolidine-2-carboxylate
3-(4-methanesulfonylphenyl)-6-methylpyridin-2-amine
1-(cyclopropylmethyl)-5-[(2,6-difluorophenyl)methyl]-N-(1,3-thiazol-2-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{4-[(2-chlorophenyl)methyl]-1-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]piperidin-4-yl}methanol
2-(4-methylpentyl)-4-{2,5,7-trimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}morpholine
1-ethyl-4-[3-(2-fluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1H-pyrazole
1-[(1s,4s)-4-aminocyclohexyl]-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
4-(3,5-dimethyl-1H-pyrazol-1-yl)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
2-amino-6-(2,4-dimethoxyphenyl)-4-[1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]pyridine-3-carbonitrile
N-(oxolan-2-ylmethyl)-3-(1-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperidin-4-yl)propanamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-(pyridin-3-ylmethyl)-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
5-chloro-2-(3,5-dimethoxyphenyl)pyrimidine
N-{[4-(2-methyl-1H-imidazol-1-yl)phenyl]methyl}-1H-pyrazole-4-carboxamide
3-[4-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]benzoic acid
N-[2-hydroxy-2-(thiophen-2-yl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
3-(3-methoxypropyl)-1-(3-methylbut-2-enoyl)piperidine-3-carboxylic acid
(3S,4R)-1-[(1-methyl-1H-pyrazol-4-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
3-(5-methylthiophen-2-yl)-5-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1H-pyrazole
N,N-dimethyl-3-{[2-(pyrrolidin-1-ylmethyl)piperidin-1-yl]sulfonyl}benzamide
N-[(3S,7S,8aS)-3-[(4-hydroxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-methoxybenzamide
2-[2-methyl-3-({7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}methyl)-1H-indol-1-yl]acetamide
1-{2-[1-(5-methoxy-1H-indazole-3-carbonyl)piperidin-4-yl]ethyl}pyrrolidin-2-one
3-[4-methoxy-3-(pyrrolidin-1-ylmethyl)phenoxy]-2,5-dimethylpyrazine
1-{2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidin-1-yl}-3-(trimethyl-1H-pyrazol-4-yl)propan-1-one
6-[3-(4-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]pyridine-2-carbonitrile