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N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-(pyridin-3-yloxy)acetamide
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2-phenylimidazo[1,2-a]pyridine-6-carboxamide
1-(diethylamino)-3-(2-methoxy-4-{[methyl(quinolin-6-ylmethyl)amino]methyl}phenoxy)propan-2-ol
1-(2-ethoxyphenyl)-4-(3-methylpiperidine-3-carbonyl)piperazine
5-{4-hydroxy-1-[(3-methylphenyl)methyl]piperidin-4-yl}-N-(pyridin-3-ylmethyl)-1-benzofuran-2-carboxamide
N-{[2-(methylsulfanyl)pyrimidin-5-yl]methyl}-1-(3-phenylpropyl)piperidin-3-amine
2-(5-acetylthiophen-3-yl)-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-(1,2-benzoxazol-6-yl)-2-(dimethylamino)-4-oxo-1,3,8-triazaspiro[4.5]dec-1-ene-8-carboxamide
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[2-(2-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
2-amino-5-methyl-6-(5-methylfuran-2-yl)-4-(pyridin-3-yl)pyridine-3-carbonitrile
1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}azocane
N-methyl-5-({5-[(4-methylphenyl)sulfanyl]furan-2-yl}methyl)-2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
2,6-dimethyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}quinoline-4-carboxamide
2-(5-phenyl-1,2-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-4-ol
8-(1H-imidazol-2-ylmethyl)-2-methyl-2,8-diazaspiro[4.5]decan-3-one
1-butyl-4-(3,5-dichloro-4-methylbenzoyl)piperazin-2-one
(1R,5R)-6-[2-methyl-2-(morpholin-4-yl)propyl]-3-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
4-{[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]amino}-N-[2-(2-fluorophenyl)ethyl]-5-methylthieno[2,3-d]pyrimidine-6-carboxamide
8-[3-(2-methyl-1H-imidazol-1-yl)propanoyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
1-[(2-chlorophenyl)methyl]-N-(1-phenylcyclopropyl)-1H-1,2,3-triazole-4-carboxamide
N-cyclopropyl-N-[(2-ethoxyphenyl)methyl]-2-methylimidazo[1,2-a]pyridine-3-carboxamide
N-[(7R,8aS)-2-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-4-oxo-4H-chromene-3-carboxamide
N-cyclopropyl-5-[2-(phenylformamido)acetyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-(3-ethoxy-5-fluorophenyl)-2-[4-(pyridin-2-ylmethyl)piperazin-1-yl]acetic acid
3-{2-[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]ethyl}-6-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(1S,5R)-6-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
N-methyl-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[1-(pyridin-4-yl)ethyl]propanamide
4-[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
2-(3-butyl-4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-1-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]acetamide
4-[1-(1-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}piperidin-4-yl)ethyl]morpholine
N-(furan-2-ylmethyl)-1-methyl-2-oxo-N-(pyridin-2-ylmethyl)-1,2,3,4-tetrahydroquinoline-4-carboxamide
N-{1-[(2-chlorophenyl)methyl]-1H-pyrazol-5-yl}-4-methyl-1,4-diazepane-1-carboxamide
3-{[4-(5-fluoro-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]methyl}phenol
3-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methoxy}pyridin-2-amine
3-methyl-4-[3-(propan-2-yl)-5-[1-(1H-pyrazol-1-yl)propyl]-1H-1,2,4-triazol-1-yl]pyridine
N-[3-methyl-1-(pentan-3-yl)-1H-pyrazol-5-yl]-2-[3-(pyridin-2-yl)-1H-pyrazol-1-yl]acetamide
N-[(3R,4S)-1-acetyl-4-propylpyrrolidin-3-yl]-1-(2-fluorophenyl)methanesulfonamide
6-amino-N-[1-(piperidine-1-carbonyl)piperidin-4-yl]pyridine-2-carboxamide
methyl 1-[5-cyclohexaneamido-1-(2-methoxyethyl)-1H-1,3-benzodiazole-7-carbonyl]piperidine-4-carboxylate
2-hydroxy-N-[(3R,4S)-4-[(3-methyl-1,2-oxazol-5-yl)methyl]oxolan-3-yl]-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
[(3-ethoxyphenyl)methyl](methyl)[2-(oxan-2-yl)ethyl]amine
1-{[4-(2,3-dihydro-1-benzofuran-5-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}-N,N-diethylpiperidine-3-carboxamide
(2R,3S,6R)-3-(2-methoxyphenyl)-5-(1-methylpiperidin-4-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-[(2,6-difluorophenyl)methyl]-3-(4-hydroxybutyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxylic acid
1-(cyclohexylmethyl)-N-[(3-hydroxy-4-methoxyphenyl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
1-(4-{[(1S,5R)-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}thiophen-2-yl)ethan-1-one
4-{2-[4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-1-yl]ethyl}morpholine
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-3-phenyl-2-(1H-1,2,3,4-tetrazol-1-yl)propanamide
5-(oxolan-2-yl)-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]thiophene-2-carboxamide
(1-{3-[1-(2-fluoroethyl)-4-phenyl-1H-imidazol-5-yl]phenyl}ethyl)dimethylamine