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4-[2-(3-chloro-4-hydroxyphenyl)acetyl]-1-(4-methoxyphenyl)piperazin-2-one
5-acetyl-N-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}thiophene-3-carboxamide
5-{[(2S)-4-methyl-2-phenylpiperazin-1-yl]methyl}-2-(pyridin-2-yl)pyrimidine
2-[(dimethylcarbamoyl)amino]-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
[7-(3,4,5-trimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methanamine
2-{[4-(2-phenylethyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}phenol
1-[2-(2-ethoxyphenyl)ethyl]-3-[4-(2-methyl-5-oxopyrrolidin-1-yl)phenyl]urea
(3S,4R)-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
(3S,4S)-1-(dimethyl-1,2-oxazole-4-carbonyl)-4-(propan-2-yl)pyrrolidine-3-carboxylic acid
5-(3,4-dihydro-2H-1-benzopyran-3-ylmethyl)pyridin-2-amine
{3-[(2-fluorophenyl)methyl]-1-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)piperidin-3-yl}methanol
1-{[(3R,4R)-1-(2,2-diphenylethyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}piperidin-4-ol
(2,1,3-benzoxadiazol-5-ylmethyl)(oxolan-2-ylmethyl)(thiophen-3-ylmethyl)amine
2-(2,4-difluorophenyl)-1-[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]ethan-1-one
4-[(2S)-1-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}pyrrolidine-2-carbonyl]morpholine
1-(2H-1,3-benzodioxole-5-carbonyl)-3-(prop-2-en-1-yl)piperidine-3-carboxylic acid
1-{[2-(4-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2-methylphenyl)-1,4-diazepane
7-(cyclobutylmethyl)-2-(2-methylfuran-3-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
N-{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-N-methyl-1H-1,2,3-benzotriazole-5-carboxamide
methyl 3-(cyclobutylmethoxy)-5-[3-hydroxy-3-(hydroxymethyl)pyrrolidine-1-carbonyl]benzoate
(4aS,7aR)-1-(4-methylpyridine-3-carbonyl)-4-pentanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-4-cyclopropyl-1-(4-propylpyrimidine-5-carbonyl)pyrrolidin-3-yl]methanesulfonamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-2-(pyridin-2-yl)pyrimidine-5-carboxamide
2-[3-(2,3-dimethoxyphenyl)pyrrolidine-1-carbonyl]-3,5-dimethyl-1H-indole
3-(4-ethylphenyl)-5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-pyrazole
methyl 3-(3-{[(dimethylsulfamoyl)amino]methyl}piperidine-1-carbonyl)benzoate
N-methyl-4-({4-[2-(methylsulfanyl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)benzamide
3-[6-hydroxy-4-(pyridin-4-yl)-1,4-diazepan-1-yl]pyrazine-2-carbonitrile
3-(morpholin-4-yl)-N-[2-(trifluoromethyl)phenyl]piperidine-1-carboxamide
[2-(1H-1,3-benzodiazol-6-yl)phenyl]methanol
[(3-chloro-4-methoxyphenyl)methyl][(1-methyl-1H-imidazol-2-yl)methyl](propan-2-yl)amine
5-methyl-1-(2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}-2-oxoethyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
6-(2,5-dimethylfuran-3-yl)-N-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-({2-methylimidazo[2,1-b][1,3,4]thiadiazol-6-yl}methyl)-3-[5-(thiophen-3-yl)-1,3,4-oxadiazol-2-yl]propanamide
N-({1-[(3-fluoro-2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)piperidine-4-carboxamide
3-[(1S,4R)-2-azabicyclo[2.2.1]heptan-2-yl]-N-[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]-N-methylpropanamide
(3aS,6aR)-3-[2-(3-chlorophenyl)ethyl]-5-[1-(propan-2-yl)piperidin-4-yl]-hexahydro-2H-pyrrolo[3,4-d][1,3]oxazol-2-one
N-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]-4-(piperidin-3-yl)benzamide
N-ethyl-2-{4-[2-(2-hydroxyethyl)-4-methyl-1H-1,3-benzodiazol-1-yl]phenyl}acetamide
3-(1-methyl-1H-imidazole-2-carbonyl)-1-(3-methylbut-2-en-1-yl)piperidine
N-methyl-1-{1-[1-(2-phenylethyl)piperidin-4-yl]piperidine-3-carbonyl}piperidin-4-amine
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[(5-methyl-1H-pyrazol-3-yl)methyl]amino}pyridine-3-carboxamide
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
1-(6-chloropyridin-3-yl)-3-methyl-3-[3-(1H-pyrazol-1-yl)propyl]urea
(3S,4R)-1-{4-[(2-hydroxyethyl)(methyl)amino]benzoyl}-4-phenylpyrrolidine-3-carboxylic acid
N-(3-chloro-2-fluorophenyl)-4-(pyrrolidin-3-yl)piperazine-1-carboxamide
(3-{furo[3,2-c]pyridin-4-yl}phenyl)methanol
5-methyl-1'-(2-methyl-1,3-benzoxazole-6-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-5-methyl-N-[(3S)-2-oxoazepan-3-yl]thiophene-2-carboxamide
1-methyl-4-phenyl-3-[1-(pyrazin-2-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one