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(3S)-N3-tert-butyl-N2-[(3-fluorophenyl)methyl]-1,2,3,4-tetrahydroisoquinoline-2,3-dicarboxamide
4-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-(6-methoxynaphthalen-2-yl)morpholine
N-cyclohexyl-1-cyclopropyl-4-oxo-5-[2-(pyridin-3-yl)piperidine-1-carbonyl]-1,4-dihydropyridine-3-carboxamide
2-[(4aS,8aR)-1-(3-aminopropyl)-2-oxo-decahydro-1,6-naphthyridine-6-carbonyl]benzonitrile
3-(2-ethylbutyl)-8-{pyrazolo[1,5-a]pyridine-3-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
(1S,5R)-3-[(4-methyl-1H-imidazol-5-yl)methyl]-6-{5-[(methylsulfanyl)methyl]furan-2-carbonyl}-3,6-diazabicyclo[3.2.2]nonane
1-({5-[(2-methoxy-3,5-dimethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
N-[(5-chlorothiophen-2-yl)methyl]-1-cyclopropyl-6-oxopiperidine-3-carboxamide
8-(1,3-benzothiazol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-[2-(1,4-oxazepan-4-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-{2-[4-(3-hydroxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]ethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(4-chlorophenyl)-2-[methyl(oxan-4-ylmethyl)amino]acetic acid
N-(cyclobutylmethyl)-2,6-dimethyl-N-(oxolan-2-ylmethyl)pyridine-4-carboxamide
3-(1H-imidazol-2-yl)-1-{1-[(4-phenylphenyl)methyl]-1H-1,2,3,4-tetrazol-5-yl}piperidine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-1-(2-methoxyethyl)piperidine-4-carboxamide
(1-{1-[(4-fluoro-3-methoxyphenyl)methyl]piperidin-4-yl}-2-phenylethyl)(2-methoxyethyl)(pyridin-2-ylmethyl)amine
4-(3-chloro-2-methylbenzoyl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(3,5-dimethylphenyl)-4-{trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}piperazin-2-one
2-(3-chlorothiophene-2-carbonyl)-7-(pyridin-3-ylmethyl)-2,7-diazaspiro[4.5]decan-6-one
[3-(cyclopropylmethyl)-1-(5-fluoro-2-methoxybenzoyl)piperidin-3-yl]methanol
1-methyl-8-[4-(methylsulfanyl)benzoyl]-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-[2-(azepan-1-yl)ethyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
benzyl({[4-(1H-pyrazol-1-yl)phenyl]methyl})(1,3-thiazol-2-ylmethyl)amine
2-(6-methoxynaphthalen-2-yl)-4-(pyrimidin-2-yl)morpholine
1-(2,2,3,3-tetramethylcyclopropanecarbonyl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-[(4-ethoxyphenyl)methyl]-N-(4,4,4-trifluorobutyl)cyclopropanamine
2-(4,5,6,7-tetrahydro-1H-indazol-5-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[(2-methyl-1H-imidazol-1-yl)methyl]-1-{2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidine
4-cyclopentyl-3-{[3-(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
2-ethyl-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-{3-cyclobutyl-6-oxo-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-4-yl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
methyl (2R,4S)-1-[4-(3,5-dimethyl-1H-pyrazol-1-yl)butanoyl]-4-hydroxypiperidine-2-carboxylate
1-({5-[(2-ethylphenyl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-3,3-dimethylurea
3-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-[1-(thiophen-2-yl)ethyl]benzamide
N-cyclohexyl-N-[2-(ethylsulfanyl)ethyl]-4-(4H-1,2,4-triazol-4-yl)benzamide
4-(3-hydroxy-4-methoxybenzoyl)-1-(4-methylphenyl)piperazin-2-one
4-(4-chlorophenyl)-N-[2-(4-methyl-6-oxo-1,6-dihydropyrimidin-2-yl)ethyl]butanamide
7-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carbonyl}-3,4-dihydro-2H-1,4-benzoxazin-3-one
2-[4-(5-fluoropentyl)phenoxy]propanamide
(3R,9aR)-3-(2-methylpropyl)-8-(2-phenylethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-{5-[3-(2,3-dimethoxyphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}-4-ethylpiperazine
1-(2-fluorophenyl)-4-[5-(oxolan-2-yl)thiophene-2-carbonyl]piperazine
(1S,5S,6S,7R)-6-(3-benzyl-1H-1,2,4-triazol-5-yl)-3-(pyridin-2-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-en-4-one
(2S,4S)-4-amino-N,N-diethyl-1-[6-(propan-2-yl)-1H-indole-2-carbonyl]pyrrolidine-2-carboxamide
3-{[(3S)-3-hydroxypyrrolidin-1-yl]methyl}-N-(2-methyl-1H-1,3-benzodiazol-6-yl)benzamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-1-(2-methoxyethyl)pyrrolidine-3-carboxamide
{[1-(2-fluorophenyl)-3-(4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}[2-(methylsulfanyl)ethyl]amine
3-[(1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-1,2,3-triazol-4-yl)methyl]-2,3-dihydro-1,3-benzoxazol-2-one
1-(2-methanesulfonylethyl)-4-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperazine