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7-ethyl-2-[5-(pyrrolidine-1-carbonyl)pyridin-2-yl]-2,7-diazaspiro[4.5]decan-6-one
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-[2-(1H-1,2,3,4-tetrazol-5-yl)benzoyl]-1,4-diazepane
4-(2-{1-[(2E)-2-methylbut-2-en-1-yl]piperidin-2-yl}ethyl)morpholine
2-[3-(1H-imidazol-1-yl)propyl]-9-(2-propoxypropanoyl)-2,9-diazaspiro[5.5]undecan-3-one
4-chloro-N-(2-hydroxyethyl)-N-[(2-methoxyphenyl)methyl]-1,5-dimethyl-1H-pyrazole-3-carboxamide
N3-[2-(4-oxo-3,4-dihydroquinazolin-2-yl)ethyl]piperidine-1,3-dicarboxamide
2,7,8-trimethyl-4-[4-(4H-1,2,4-triazol-4-yl)piperidine-1-carbonyl]quinoline
8-(quinolin-8-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
2-[methyl(1,2-oxazol-3-ylmethyl)amino]-2-{4-[(pyrrolidine-1-carbonyl)amino]phenyl}acetic acid
1-methyl-N-[(3-phenylphenyl)methyl]-3-(propan-2-yl)-1H-pyrazole-5-carboxamide
3-(3-methyl-1,2-oxazol-5-yl)-4-[(3-methylphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(pyridin-3-ylmethyl)-4-[(2R)-pyrrolidine-2-carbonyl]piperazine
[1-(5-fluoro-1H-indole-2-carbonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
5-{4-[4-(propan-2-yl)piperazin-1-yl]phenyl}-1H-indazol-3-amine
1-[4-hydroxy-4-(pyridin-3-yl)piperidin-1-yl]-2-[1-(propan-2-yl)piperidin-4-yl]ethan-1-one
4-methyl-2-propyl-6-{1H-pyrrolo[2,3-b]pyridin-4-yl}pyrimidine
1-(6-methyl-2-phenylpyrimidin-4-yl)-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)piperidin-4-amine
(3S,9aR)-3-(4-aminobutyl)-8-{[1-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
6-{2-[(adamantan-1-ylformamido)methyl]-5-methyl-2,3-dihydro-1-benzofuran-7-yl}pyridine-3-carboxamide
7-methyl-4-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-[4-(2,2-dimethylpropyl)-1-[(4-ethoxyphenyl)methyl]piperazin-2-yl]ethan-1-ol
1-(2-methoxyethyl)-3-(2-phenylethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(3aS,6aS)-2-cyclopentyl-5-(4-oxo-4-phenylbutanoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-[5-(5-acetylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propan-1-one
1-cyclopropanecarbonyl-3-({4-[4-(1H-pyrazol-1-yl)phenyl]-1H-1,2,3-triazol-1-yl}methyl)piperidine
6-(2-methylpropyl)-4-[3-(pyridin-2-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydropyrimidin-2-one
2-(4-methoxyphenyl)-5-{[2-(pyridin-3-yl)piperidin-1-yl]methyl}pyrimidine
[(4aS,8aR)-1-(furan-3-ylmethyl)-6-[(5-methylthiophen-2-yl)methyl]-decahydro-1,6-naphthyridin-4a-yl]methanol
(3S,4S)-4-(naphthalen-2-yl)-1-(oxane-4-carbonyl)piperidin-3-ol
2-(1-{7-methylpyrazolo[1,5-a]pyrimidine-6-carbonyl}pyrrolidin-2-yl)-1,3-benzothiazole
[(8-methoxy-3,4-dihydro-2H-1,5-benzodioxepin-7-yl)methyl](methyl){[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}amine
4-(1H-indol-3-yl)-N-[(1-methylpyrrolidin-3-yl)methyl]butanamide
N-cyclopropyl-1-{1-[(5-fluoro-2-methoxyphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(cyclohexylmethyl)-N-methyl-N-(oxan-4-ylmethyl)-6-oxopiperidine-3-carboxamide
2-{methyl[6-methyl-2-(pyridin-3-yl)pyrimidin-4-yl]amino}ethan-1-ol
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-2-(3-methoxyphenyl)pyrrolidine
9-(azepane-4-carbonyl)-2-cyclopropyl-2,9-diazaspiro[5.5]undecan-3-one
N-[(3S,4R)-1-[3-(hydroxymethyl)-8-methylquinolin-2-yl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
(2S)-1-({5-methyl-2-[3-(trifluoromethyl)phenyl]-1,3-oxazol-4-yl}methyl)pyrrolidine-2-carboxamide
N-[(3,4-difluorophenyl)methyl]-3-{1-[(4-methoxy-3-methylphenyl)methyl]piperidin-3-yl}propanamide
({1-[1-(5-fluoro-2-methoxybenzoyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}methyl)(methyl)amine
N-ethyl-N,7-dimethyl-2-[2-(pyridin-3-yl)pyrimidin-5-yl]quinoline-4-carboxamide
N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-4-methyl-N-(pyridin-4-ylmethyl)-1,3-thiazole-5-carboxamide
4-(4-ethyl-3,3-dimethylpiperazine-1-carbonyl)-2,3-dihydro-1H-imidazol-2-one
N-[3-({[3-(azepan-1-yl)propyl](methyl)carbamoyl}amino)-4-fluorophenyl]acetamide
5-(4-chloro-1-ethyl-1H-pyrazol-3-yl)-3-(oxolan-3-yl)-1,2,4-oxadiazole
[(8-fluoroquinolin-2-yl)methyl][1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]amine
N-[2-(4-fluorophenyl)-2-(pyrrolidin-1-yl)ethyl]-2-(8-methoxy-2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)acetamide
N-methyl-N-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}-2,3-dihydro-1-benzothiophene-2-carboxamide
2-{6-azaspiro[2.5]octane-1-carbonyl}-2,3-dihydro-1H-isoindole