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N-{4-[5-(furan-2-yl)-1,3,4-oxadiazol-2-yl]phenyl}-2-methyl-3-(1H-pyrazol-1-yl)propanamide
N-[(dimethyl-1,2-oxazol-4-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-{[3-ethyl-4-(propan-2-yl)piperazin-1-yl]methyl}-6-methyl-1,2-dihydroquinolin-2-one
3-{1-[1-(propan-2-yl)-1H-pyrazole-4-carbonyl]piperidin-4-yl}phenol
4-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-acetyl-6-methyl-3-[2-methyl-4-(4-methylphenyl)piperazine-1-carbonyl]-1,2-dihydropyridin-2-one
1-[4-({[(6-chloropyridin-3-yl)methyl](methyl)amino}methyl)phenyl]ethan-1-one
4-(4-{[4-methyl-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-1-yl)quinoline
10-methoxy-5-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
1-methyl-6-(pyridin-2-yl)-N-(1,2,3,4-tetrahydronaphthalen-1-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
N-(adamantan-1-yl)-3-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-oxopropanamide
4-ethyl-3-{1-[3-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}-4,5-dihydro-1H-1,2,4-triazol-5-one
methyl N-{2-[3-(3-methylphenoxymethyl)piperidin-1-yl]-2-oxoethyl}carbamate
N-{[2-(dimethylamino)-5,8-dimethoxyquinolin-3-yl]methyl}-N-[(4-methoxyphenyl)methyl]-4-methylbenzamide
(2S)-N2-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)pyrrolidine-1,2-dicarboxamide
6-fluoro-2-({4-[(pyridin-2-yl)amino]piperidin-1-yl}methyl)quinolin-4-ol
1-[(2S,4R)-1-benzyl-4-(1H-1,2,3,4-tetrazol-1-yl)pyrrolidine-2-carbonyl]azepane
3-{[(2H-1,3-benzodioxol-5-ylmethyl)[(3-fluorophenyl)methyl]amino]methyl}piperidin-3-ol
N-(2,5-dimethylphenyl)-N'-[2-(6-hydroxypyrimidin-4-yl)ethyl]propanediamide
5-[methyl(2-phenylethyl)amino]-2-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,3-dihydropyridazin-3-one
2-(dimethyl-1,2-oxazol-4-yl)-N-ethyl-N-({1-[2-(3-methoxyphenyl)ethyl]piperidin-3-yl}methyl)acetamide
2-(3-hydroxypiperidin-1-yl)-1-[4-(2-methoxybenzoyl)piperazin-1-yl]ethan-1-one
3-(prop-2-en-1-yl)-1-(2,3,4-trimethoxybenzoyl)piperidine-3-carboxylic acid
N-[3-(methylsulfanyl)propyl]-2,3-dihydro-1H-indene-1-carboxamide
3-[3-(furan-3-yl)phenyl]-1-(oxolan-2-ylmethyl)-1H-pyrazole
1'-[(5-ethylpyridin-2-yl)methyl]-1-methyl-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
7-cyclohexyl-2-[2-(diethylamino)ethyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)-3-(2-phenoxyethyl)piperidine-3-carboxylate
2-chloro-N-{1-[2-(4-methoxyphenyl)ethyl]-5-oxopyrrolidin-3-yl}benzamide
(2S,4S)-4-amino-N-ethyl-1-[(1-ethyl-3-methyl-1H-pyrazol-5-yl)sulfonyl]pyrrolidine-2-carboxamide
N-(dimethyl-1H-1,2,4-triazol-5-yl)-5-[1-(3,3,3-trifluoropropanoyl)pyrrolidin-2-yl]thiophene-2-carboxamide
[(1-ethenyl-1H-pyrazol-4-yl)methyl](methyl)[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
N-(2-chloro-4-fluorophenyl)-4-[5-(hydroxymethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidine-1-carboxamide
4-(3-tert-butyl-1H-pyrazol-1-yl)-1-(cyclohex-3-ene-1-carbonyl)piperidine-4-carboxylic acid
1-[2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
(2S,3S)-2-({1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-methylpentanamide
3-{[(3R,4S)-3-amino-4-(2-hydroxyethyl)pyrrolidin-1-yl]sulfonyl}-N-cyclopropylbenzamide
1-[2-(pyridin-2-yl)piperidin-1-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
4-[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]-N-[2-(pyrazin-2-yl)ethyl]pyrimidin-2-amine
(3R,4R)-3-methyl-1-{[4-(methylsulfanyl)phenyl]methyl}-4-(oxan-4-yl)piperidin-4-ol
N-cyclopropyl-2-{4-[(4-fluorophenyl)methyl]-5-oxo-3-(propan-2-yl)-1,4-diazepan-1-yl}acetamide
N-[2-(3-{[4-(3-chlorophenyl)piperazin-1-yl]methyl}phenoxy)propyl]-1,3-thiazole-5-carboxamide
[(3R,5R)-5-{[(2-methoxyethyl)(methyl)amino]methyl}-1-(2-methylfuran-3-carbonyl)piperidin-3-yl]methanol
(4aR,7aS)-1-(cyclopropylmethyl)-4-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]piperidine-1-carboxamide
3-[1-({5,7-dimethylpyrazolo[1,5-a]pyrimidin-3-yl}methyl)piperidin-4-yl]-4-ethyl-1-methyl-4,5-dihydro-1H-1,2,4-triazol-5-one
2-[(4aS,8aR)-1-(4-hydroxybutyl)-2-oxo-decahydro-1,6-naphthyridin-6-yl]-6-methylpyridine-3-carbonitrile
5-[(2-acetamidoethyl)amino]-1-propyl-4,5,6,7-tetrahydro-1H-indazole-3-carboxylic acid
N-(2,3-dihydro-1,4-benzodioxin-6-yl)-3-(1-{[3-(methylsulfanyl)phenyl]methyl}piperidin-4-yl)propanamide
2-fluoro-N-{3-[4-(3-methoxyphenyl)piperazin-1-yl]-3-oxopropyl}benzamide