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4-{2-[1-(2,5-dichlorophenyl)-3-methyl-1H-1,2,4-triazol-5-yl]propyl}morpholine
1-acetyl-N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]piperidine-3-carboxamide
2-(2-chlorophenoxy)-1-(7-{[3-(methoxymethyl)piperidin-1-yl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)ethan-1-one
2-amino-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-2-methylpropanamide
5,6-dimethyl-3-[4-(1H-pyrazol-1-yl)phenyl]-1,2-dihydropyridin-2-one
3-({1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
(2S,4S)-4-amino-1-(2-cyclopentylacetyl)-N,N-diethylpyrrolidine-2-carboxamide
N-{[4-(dimethylamino)oxan-4-yl]methyl}-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methyl-1-(thiomorpholin-4-yl)propan-1-one
N-{[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-2-(2,6,6-trimethyl-4-oxo-1-propyl-4,5,6,7-tetrahydro-1H-indol-3-yl)acetamide
N-[(1,5-dimethyl-1H-pyrazol-3-yl)methyl]-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
2-(butylsulfanyl)-N4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]pyrimidine-4,6-diamine
1-[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]-3-(pyridin-4-yl)propan-1-one
2-(3-acetyl-7-ethyl-1H-indol-1-yl)-1-[4-(dimethylamino)azepan-1-yl]ethan-1-one
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-N-(propan-2-yl)-N-[(trimethyl-1H-pyrazol-4-yl)methyl]acetamide
1-[(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepane
2-{3-[1-(4-chlorophenyl)-1H-pyrazol-4-yl]-1H-pyrazol-1-yl}-N-(1,3-dimethyl-1H-pyrazol-5-yl)acetamide
5-fluoro-2-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)pyrrolidin-2-yl]-1H-1,3-benzodiazole
1-[4-ethoxy-3-(trifluoromethyl)phenyl]-3-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]urea
(4aS,8aR)-1-(2-aminoethyl)-6-(oxane-4-carbonyl)-decahydro-1,6-naphthyridin-2-one
5-(1-benzyl-1H-pyrazol-4-yl)-1,3-dimethyl-1H-1,2,4-triazole
2-methyl-1-[2-(4-methylpentyl)morpholin-4-yl]propan-1-one
2-(2-ethyl-4-methyl-6-oxo-1,6-dihydropyrimidin-5-yl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}acetamide
2-(1-cyclopentyl-4-{[4-(propan-2-yl)-1,3-thiazol-2-yl]methyl}piperazin-2-yl)ethan-1-ol
N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)quinoxaline-5-carboxamide
(4aR,7aS)-1-(2-methoxyethyl)-4-[2-oxo-2-(piperidin-1-yl)ethyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-methyl-N-[2-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]pyrido[2,3-d]pyrimidin-4-amine
1-[(1S,3R)-1-ethoxy-3-hydroxy-7-azaspiro[3.5]nonan-7-yl]-2-[3-(trifluoromethyl)phenyl]ethan-1-one
5-{2-[2-(4-hydroxyphenyl)ethyl]piperidine-1-carbonyl}-1-methyl-1,2-dihydropyridin-2-one
(1S,5R)-6-(1H-indole-2-carbonyl)-3-(3-phenylpropyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(3R,4S)-4-cyclopropyl-1-(2-hydroxyethyl)pyrrolidin-3-yl]-2-methyl-1H-pyrrole-3-carboxamide
1-[4-(3-chloro-4-fluorophenyl)piperazin-1-yl]-2-[methyl(piperidin-4-yl)amino]ethan-1-one
1-{2-[(2,4-dimethoxyphenyl)formamido]ethyl}-N-(thiophen-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
4-[5-chloro-2-(piperidine-1-carbonyl)phenoxy]-1-(thiophen-3-ylmethyl)piperidine
9-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-6-oxa-9-azaspiro[4.5]decane
N-[(3R,4S)-4-cyclopropyl-1-(pyridin-4-yl)pyrrolidin-3-yl]oxane-4-carboxamide
(2S)-2-amino-1-[3-(3-ethylphenoxy)azetidin-1-yl]-4-(methylsulfanyl)butan-1-one
1-[benzyl(methyl)amino]-3-[4-({[(3-fluorophenyl)methyl]amino}methyl)phenoxy]propan-2-ol
1,7-dimethyl-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]-1H-indole-2-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]ethan-1-one
1-{[1-(2-hydroxybutyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]methyl}-4-methyl-1,2-dihydroquinolin-2-one
(3aR,6aR)-2-methanesulfonyl-5-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-{[(1-hydroxybutan-2-yl)(thiophen-3-ylmethyl)amino]methyl}-2,6-dimethylphenyl acetate
3-{3-[(1-methylpiperidin-4-yl)methyl]-1,2,4-oxadiazol-5-yl}-1-phenylpropan-1-one
2-(2,5-dimethoxyphenyl)-2-[4-(pyridin-4-yl)piperazin-1-yl]acetic acid
2-(4-ethyl-1,3-thiazol-2-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
1-(6-{4-[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}pyridin-3-yl)ethan-1-one
1-{2-[1-(5-chloro-2-methoxyphenyl)-3-(2-methoxyethyl)-1H-1,2,4-triazol-5-yl]ethyl}-5-methyl-1H-1,2,3,4-tetrazole
N-(6-hydroxy-6-methylheptan-2-yl)-3-(4-methoxyphenyl)-1H-pyrazole-5-carboxamide
2-(2H-1,3-benzodioxol-5-yl)-1-[(2S)-2-(3-ethyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]ethan-1-one