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1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(2-methoxyphenoxy)piperidine-4-carboxylic acid
2-[5-(6,6-dimethyl-5-oxothiomorpholin-3-yl)-3-methyl-1H-1,2,4-triazol-1-yl]acetic acid
methyl 6-({cyclopropyl[(trimethyl-1H-pyrazol-4-yl)methyl]amino}methyl)-3-(furan-2-amido)thieno[2,3-b]pyridine-2-carboxylate
2-(4-{[(2S)-1-hydroxy-4-(methylsulfanyl)butan-2-yl]amino}-6-methylpyrimidin-2-yl)phenol
3-({[2-(diethylamino)ethyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-methyl-4-(2-oxo-5,5-diphenylpiperidin-1-yl)butanamide
4-methyl-1-{pyrazolo[1,5-a]pyrimidin-3-yl}-1H-pyrazole
(4aS,7aR)-1-[(2,6-dimethylphenyl)methyl]-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(2-fluorophenyl)methyl]-2-{[(4-methanesulfonylmorpholin-2-yl)methyl]amino}acetamide
4-(1,3-benzothiazol-2-yl)-1-(1H-imidazol-4-ylmethyl)piperazine-2-carboxylic acid
1-methyl-4-[1-(5-phenoxyfuran-2-carbonyl)pyrrolidin-3-yl]piperazine
1-[(4-methoxyphenyl)methyl]-4-(4-phenylbutanoyl)piperazin-2-one
1-[cyclohexyl(methyl)amino]-3-[4-({[(3-fluoro-4-methylphenyl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
N-[2-({[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)amino}methyl)quinolin-6-yl]acetamide
2-methoxy-6-[2-(oxan-3-yl)ethyl]-5-oxo-5,6-dihydro-1,6-naphthyridine-3-carbonitrile
5-({4-[4-(4-fluorophenyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-2-methylpyrimidine
N-(2-methylpropyl)-2-[3-oxo-1-(3-phenylpropyl)piperazin-2-yl]acetamide
2-[methyl(piperidin-4-yl)amino]-N-{1-[(4-methylphenyl)methyl]cyclopropyl}acetamide
dimethyl({[(1R,5S,6R)-3-[4-(1,3-oxazol-5-yl)benzenesulfonyl]-3-azabicyclo[3.1.0]hexan-6-yl]methyl})amine
2-{1-[(2-ethoxyphenyl)methyl]-4-(3-methyl-1H-pyrazole-5-carbonyl)piperazin-2-yl}ethan-1-ol
4-(2-methoxyphenoxy)-1-{[2-(2-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
(1S,5R)-6-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
5-(1-{[4-(1H-imidazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
7-(cyclopropylmethyl)-2-{[3-(prop-2-en-1-yloxy)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
2-(2,6-difluorophenyl)-1-[(3R,4S)-3-(3-hydroxypropyl)-4-(4-methylpiperazin-1-yl)piperidin-1-yl]ethan-1-one
N-(1-{2-[cyclohexyl(methyl)amino]-4-methylpyrimidin-5-yl}ethyl)cyclopropanecarboxamide
1-(3-methoxyphenoxy)-3-{[1-(1-methylcyclopropyl)propan-2-yl]amino}propan-2-ol
6-oxo-N-(quinolin-6-ylmethyl)-1-{[3-(trifluoromethyl)phenyl]methyl}piperidine-3-carboxamide
2-({6-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]quinazolin-4-yl}amino)ethan-1-ol
1-(3,3-diphenylpiperidin-1-yl)-3-methanesulfonylpropan-1-one
4-[(2-methyl-1H-imidazol-1-yl)methyl]-1-[1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]piperidine
5-cyclopropanecarbonyl-1'-(1-ethylpyrrolidine-2-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
4-(2-ethoxyethyl)-1-[(4-fluorophenyl)methyl]-2-(propan-2-yl)-1,4-diazepane
{[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]methyl}[1-(1H-1,2,4-triazol-5-yl)ethyl]amine
4-acetyl-N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)benzamide
5-(1H-1,3-benzodiazol-1-ylmethyl)-N-[2-(propan-2-ylsulfanyl)ethyl]-1H-pyrazole-3-carboxamide
1-{4-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]phenyl}piperidine-3-carboxylic acid
4-(5-chloro-2-methylphenyl)-3-(pyridin-3-ylmethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
2-{4-[(2-fluoro-5-methoxyphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
3,7-dimethyl-11-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)-3,7,11-triazaspiro[5.6]dodecane
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(2-oxopiperidin-1-yl)acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-(3-methyl-3-phenylpiperidin-1-yl)butan-1-one
4-(cyclopropylmethyl)-1-[3-(3-hydroxy-1,2-oxazol-5-yl)propanoyl]-3-(propan-2-yl)-1,4-diazepan-5-one
6-methyl-1-[3-oxo-3-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)propyl]-1,2-dihydropyridin-2-one
[(3R,4R)-4-{[ethyl(methyl)amino]methyl}-1-(6-ethyl-2-methylpyrimidin-4-yl)pyrrolidin-3-yl]methanol
1-[(2-fluorophenyl)methyl]-4-[(3-phenyl-1,2-oxazol-5-yl)methyl]-1,4-diazepane
(1S,5R)-3-(pyrazine-2-carbonyl)-6-(pyridine-3-sulfonyl)-3,6-diazabicyclo[3.2.2]nonane
4-[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-(propan-2-yl)-1,3-oxazole
3-(2,5-dimethylphenyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}-1H-pyrazole
3-[(3R,4S)-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol