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3-fluoro-4-{3-[1-(pyridin-2-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine
(1S,2R)-2-{[(6-ethoxyquinolin-2-yl)methyl](methyl)amino}cyclohexan-1-ol
3-chloro-9-[2-(3,4-dimethylpiperazin-1-yl)ethyl]-9H-carbazole
8-{[4-(3-hydroxyprop-1-yn-1-yl)thiophen-2-yl]methyl}-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2,2-dimethyl-1-(4-methylphenyl)-N-{[6-(morpholin-4-yl)pyrimidin-4-yl]methyl}cyclopropane-1-carboxamide
2-(2-chloro-5-methylphenyl)-2-{methyl[(1-methyl-1H-pyrazol-4-yl)methyl]amino}acetic acid
N-[(5-chloro-1H-indol-2-yl)methyl]-5-(morpholin-4-ylmethyl)-1,2-oxazole-3-carboxamide
(1S,5R)-6-(3-methylbut-2-en-1-yl)-3-[2-(pyrrolidin-1-yl)benzoyl]-3,6-diazabicyclo[3.2.2]nonan-7-one
7-[(4-fluorophenyl)methyl]-2-(5-methoxyfuran-2-carbonyl)-2,7-diazaspiro[4.5]decane
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-2,3-dimethylbenzamide
8-benzoyl-2-[(5-methylpyrazin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-7-(1-methylpiperidine-3-carbonyl)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-[(5-amino-1H-1,2,4-triazol-3-yl)methyl]-8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carboxamide
1-{3-[2-(4-fluorophenyl)ethyl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
2-[({1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxy-2-oxopiperidin-3-yl}methyl)amino]-N-methylacetamide
N-(1,1-dioxo-1λ6-thian-4-yl)-N-methyl-2-(1H-pyrazol-1-yl)butanamide
3-(propan-2-yl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,2-oxazole-5-carboxamide
5-(1-ethyl-3-methyl-1H-pyrazol-4-yl)-8-methoxyquinoline
4-[4-(pyrrolidin-1-yl)piperidin-1-yl]-2-(trifluoromethyl)pyrimidine
2-[5-(5-methoxy-1-methyl-1H-indole-2-carbonyl)-1H,4H,5H,6H-pyrrolo[3,4-c]pyrazol-1-yl]ethan-1-ol
1-[(2-fluorophenyl)methyl]-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
3-(azocan-1-yl)-N-[(5-methoxy-1,3-benzoxazol-2-yl)methyl]propanamide
(1-{[2-(ethylsulfanyl)pyrimidin-5-yl]methyl}piperidin-4-yl)(1-methyl-1H-imidazol-2-yl)methanol
[1-(1-benzylpyrrolidin-3-yl)-4-(2-phenoxyethyl)piperidin-4-yl]methanol
methyl (2S,4R)-1-methyl-4-(1-methyl-1H-1,2,3-benzotriazole-5-amido)pyrrolidine-2-carboxylate
3-(2,4-difluorophenyl)-6-(oxolane-3-carbonyl)-1-(pyridin-2-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{1-[(8-methoxyquinolin-2-yl)methyl]piperidin-4-yl}-N-(propan-2-yl)piperidine-4-carboxamide
7-fluoro-N-{2-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}-2-methylquinoline-4-carboxamide
N-{2-[2-(3,6-dioxo-1,2,3,6-tetrahydropyridazin-1-yl)acetamido]-4-methylphenyl}pentanamide
3-({[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl](2-methoxyethyl)amino}methyl)-7-fluoro-1,2-dihydroquinolin-2-one
methyl (2S)-3-methyl-2-[(5-methyl-4-{[2-(piperidin-1-yl)ethyl]amino}thieno[2,3-d]pyrimidin-6-yl)formamido]butanoate
1-cyclohexyl-3-(cyclopropylmethyl)-N-(2-hydroxyethyl)-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
2-methyl-4-(5-{[(2-methylpropyl)(pyridin-2-ylmethyl)amino]methyl}thiophen-2-yl)but-3-yn-2-ol
3-[3-(2,5-dimethoxyphenyl)pyrrolidine-1-carbonyl]-1,4,6-trimethyl-1,2-dihydropyridin-2-one
N-ethyl-N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-1H-1,2,4-triazole-5-carboxamide
methyl 6-{[bis(prop-2-en-1-yl)amino]methyl}-3-(5-methylthiophene-2-amido)thieno[2,3-b]pyridine-2-carboxylate
N-[(3-ethoxyphenyl)methyl]-2-(2-hydroxyphenyl)-N-(prop-2-en-1-yl)acetamide
1-(cyclopropanesulfonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
4-{1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-2-methylpropan-2-yl}morpholine
4-(1-methyl-5-phenyl-1H-pyrrole-2-carbonyl)-1-(4-methylphenyl)piperazin-2-one
9-[2-(dimethylamino)-6-methylpyrimidin-4-yl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-hydroxy-2,2-dimethylpropyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
(1R,5R)-3-methanesulfonyl-6-(3-phenylbenzoyl)-3,6-diazabicyclo[3.2.2]nonane
2-methyl-6-[(thian-4-yl)amino]heptan-2-ol
4-[(4-fluorophenyl)sulfanyl]-1-{[2-(4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperidine
1-{1-[(2-fluorophenyl)methyl]-1H-1,2,3-triazole-4-carbonyl}-4-(2-phenylethyl)piperidine
N-[2-(4-methoxyphenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(1-oxo-2,3-dihydro-1H-isoindol-2-yl)-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}butanamide
ethyl 3-(2-phenylethyl)-1-(pyrazine-2-carbonyl)piperidine-3-carboxylate
N2-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]pyrimidine-2,4-diamine