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N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]pyrazin-2-amine
2-methyl-1-[1-(3-propyl-1H-pyrazole-5-carbonyl)azetidin-3-yl]piperidine
4-(2-phenylethyl)-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
N'-(2-ethoxyphenyl)-N-methyl-N-[(5-phenyl-1,2-oxazol-3-yl)methyl]propanediamide
1-[4-(dimethylamino)-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]-2,2-dimethylpropan-1-one
3-{1-[2-(2-methoxyphenyl)acetyl]piperidin-3-yl}-N-methyl-N-[2-(pyridin-2-yl)ethyl]propanamide
N-ethyl-N-({1-[2-(3-fluorophenyl)ethyl]piperidin-3-yl}methyl)-2-(1-methylpiperidin-4-yl)acetamide
3-(4-{[3-(hydroxymethyl)-3-methylpiperidin-1-yl]methyl}-1H-pyrazol-1-yl)propanoic acid
2-chloro-N-{[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]methyl}benzamide
(4aR,8aR)-2-[(2-chloro-5-fluorophenyl)methyl]-7-cyclobutanecarbonyl-decahydro-2,7-naphthyridin-4a-ol
4-{1-[1-(1,3-thiazole-4-carbonyl)piperidin-4-yl]piperidine-3-carbonyl}morpholine
4-(1H-imidazol-1-yl)-1-[3-(trimethyl-1H-pyrazol-1-yl)propanoyl]piperidine-4-carboxylic acid
N,N-dimethyl-4-(2-methyl-4-phenylpyrimidine-5-carbonyl)piperazine-1-sulfonamide
1-benzyl-4-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1,4-diazepan-6-ol
ethyl 4-[3-(azocan-1-yl)propanamido]piperidine-1-carboxylate
2-cyclopropyl-5-{3-[(2-fluorophenyl)methoxy]azetidin-1-yl}-1,3,4-oxadiazole
4-{4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}benzene-1-sulfonamide
N-{[7-(9H-fluoren-2-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}-5-(methoxymethyl)furan-2-carboxamide
2-({[(3R,4R)-4-(hydroxymethyl)-1-[7-(propan-2-yl)-[1,2,4]triazolo[1,5-a]pyrimidine-5-carbonyl]pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
4-{[2-(propan-2-yl)pyrimidin-4-yl]methyl}-1λ6-thiomorpholine-1,1-dione
6,7-dimethyl-2-({2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}methyl)-1H-1,3-benzodiazole
(4aS,7aR)-1-(3,4-difluorobenzoyl)-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
{1-[5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carbonyl]piperidin-2-yl}methanol
2-[(2-{2-cyano-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl}phenyl)amino]acetic acid
N-{[4-(cyclohex-3-en-1-ylmethoxy)phenyl]methyl}-3-fluoro-N-(pyridin-4-ylmethyl)benzamide
1-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-[5-(2-methylphenyl)-1,3,4-thiadiazol-2-yl]urea
4-hydroxy-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]piperidine-4-carboxylic acid
1,3-dimethyl-N-[1-(1-methyl-1H-pyrazol-4-yl)ethyl]-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methyl-4-({[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]carbamoyl}amino)-N-(propan-2-yl)benzamide
1-[(4aR,8aS)-1-(adamantane-1-carbonyl)-decahydro-1,6-naphthyridin-6-yl]-2-methoxyethan-1-one
N-{1-[(3-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-2-(3-methoxyphenoxy)acetamide
({5-[1-(2H-1,3-benzodioxol-5-ylmethyl)piperidin-3-yl]-4-methyl-4H-1,2,4-triazol-3-yl}methyl)dimethylamine
N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-2-hydroxybutanamide
1-(2-aminopyridine-4-carbonyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
4-benzyl-1-[2-(1-methylpyrrolidin-2-yl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
benzyl({[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl})methylamine
3-[(3S,4R)-1-benzyl-4-(pyrrolidin-1-yl)piperidin-3-yl]-N-(morpholin-4-yl)propanamide
1-(2-chloro-6-fluoro-3-methylbenzoyl)-4-[1-(cyclobutylmethyl)-1H-imidazol-2-yl]piperidine
2-(3-fluoro-4-hydroxyphenyl)-1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]ethan-1-one
4-methyl-7-(methylsulfanyl)-2-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}quinoline
N-[3-(1,3-benzothiazol-2-yl)propyl]-3-methyl-4,5-dihydro-1,2-oxazole-5-carboxamide
3-[4-(pyrimidin-2-yl)-1,4-diazepane-1-carbonyl]piperidine-1-carboxamide
2-[(propan-2-yl)amino]-N-(thiolan-3-yl)pyrimidine-5-carboxamide
(1-{[3-(3-methylphenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-yl)methanol
3-[1-(6-ethyl-5-fluoropyrimidin-4-yl)piperidin-3-yl]-N-methyl-N-(1-methylpiperidin-4-yl)propanamide
N-{1-[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-4-yl}methanesulfonamide
2-(1-ethylpiperidin-4-yl)-N-[2-(5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)ethyl]acetamide
4-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-7-(phenoxathiin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]-1-[4-(propan-2-yl)phenyl]pyrrolidin-2-one
{[5-(1-{imidazo[1,2-a]pyridine-2-carbonyl}piperidin-3-yl)-4-methyl-4H-1,2,4-triazol-3-yl]methyl}dimethylamine