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1-[1-(4-chlorophenyl)cyclopropanecarbonyl]-4-[(4-methoxyphenyl)methyl]-1,4-diazepan-5-one
N-methyl-1-propyl-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
2-[2-(3-methoxypropyl)piperidine-1-carbonyl]-1,4-dimethyl-1H-indole
2-(2H-1,3-benzodioxol-5-yl)-2-(dimethylamino)-1-[(1R,2R,6S,7S)-10-oxa-4-azatricyclo[5.2.1.02,6]decan-4-yl]ethan-1-one
3-(2-hydroxybutyl)-6-phenyl-3H,4H-thieno[3,2-d]pyrimidin-4-one
N-({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)-N-methylimidazo[1,2-a]pyrimidine-2-carboxamide
2-{4-[2-amino-3-cyano-6-(1,3-dimethyl-1H-pyrazol-4-yl)pyridin-4-yl]phenoxy}acetamide
1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]-2-(1H-indol-3-yl)ethan-1-one
3-[(4-methoxyphenyl)methyl]-1-(3-methoxypropyl)-8-(1,2,3,4-tetrahydronaphthalen-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-cyclohexyl-3-(cyclopropylmethyl)-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
3-(3-hydroxy-3-methylbutyl)-N-[(2-methylphenyl)methyl]-N-(oxolan-2-ylmethyl)benzamide
methyl 5-(4,5,6,7-tetrahydro-2-benzothiophene-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
1-[benzyl(methyl)amino]-3-(5-{[(dicyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-methyl-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-4-(2-methylphenyl)piperazine
N-(2-methoxyethyl)-2-[2-(propan-2-yloxy)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
1-{[2-(2-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-3-(methoxymethyl)-1H-1,2,4-triazole
ethyl 1-(2-hydroxy-2-phenylethyl)-4-oxo-5-phenoxy-1,4-dihydropyridine-3-carboxylate
2-(5-{1-[2-(1H-pyrazol-1-yl)ethyl]-1H-1,2,3-triazol-4-yl}furan-2-yl)benzonitrile
N-cyclopentyl-1-(2-methylpropyl)-5-(pyridine-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-(1H-indol-4-ylmethyl)urea
4-(3-fluorophenyl)-6-methylpyrimidin-2-amine
2-{1-[(3,4-difluorophenyl)methyl]piperazin-2-yl}ethan-1-ol
N-(2,1,3-benzothiadiazol-5-ylmethyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
methyl 5-cyano-2-methyl-6-[methyl({[3-(pyridin-2-yl)-1,2,4-oxadiazol-5-yl]methyl})amino]pyridine-3-carboxylate
(4aS,7aR)-1-[2-(3,4-dimethyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[5-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]-1H-1,3-benzodiazole
N-[(1-ethylpyrrolidin-2-yl)methyl]-5-(2-fluorophenoxymethyl)-1H-pyrazole-3-carboxamide
(4aR,8aR)-4a-hydroxy-7-(1H-indol-5-ylmethyl)-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
(3S,5R)-N3-cyclohexyl-N5-(2,3-dihydro-1H-inden-5-yl)-1-(2-methylpropyl)piperidine-3,5-dicarboxamide
2-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-1,3-oxazole-4-carboxylic acid
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(2S,3S)-3-methyl-2-{[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}pentanamide
3-[2-(1H-imidazol-2-yl)-1H-imidazol-1-yl]-N-methylbenzamide
8-[2-(1-ethylpiperidin-3-yl)-1H-imidazol-1-yl]quinoline
1-(morpholin-4-yl)-3-[5-(pyridin-4-ylmethyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]propan-1-one
1-[2,2-bis(prop-2-en-1-yl)pyrrolidin-1-yl]-2-(morpholin-4-yl)ethane-1,2-dione
2-methyl-5-[(1R,5R)-6-methyl-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1-phenyl-1H-1,3-benzodiazole
4-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]morpholine
N-[2-(2-ethoxyphenoxy)ethyl]-N,6-dimethylpyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[(4S,6R)-6-methyl-2-sulfanylidene-1,3-diazinan-4-yl]-N-{5-[(2-methylphenyl)methyl]-1,3,4-thiadiazol-2-yl}acetamide
1-[(2R,3R)-3-amino-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]-2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)ethan-1-one
N-{2-[(2S)-pyrrolidin-2-yl]ethyl}-4-(1H-1,2,4-triazol-3-yl)benzamide
2-[methyl(pyridin-2-ylmethyl)amino]-1-[2-methyl-4-(4-methylphenyl)piperazin-1-yl]ethan-1-one
5-cyclopropyl-1-[4-(furan-2-yl)pyrimidin-2-yl]-N-methyl-N-(1-methylpiperidin-4-yl)-1H-pyrazole-4-carboxamide
1-(pyrimidin-2-yl)-4-{5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carbonyl}-1,4-diazepane
phenyl (7S,9aR)-7-(hydroxymethyl)-6,9-dioxo-octahydro-1H-pyrazino[1,2-a]piperazine-2-carboxylate
7-chloro-2-(1H-pyrazol-3-yl)quinoxaline
3-[1-(1-methyl-1H-pyrazol-5-yl)propyl]-1-(5,6,7,8-tetrahydronaphthalen-1-yl)urea
N-tert-butyl-5-[4-(3-chlorophenyl)piperazine-1-carbonyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxamide
7-(8-methylquinolin-5-yl)-[1,2,4]triazolo[4,3-c]pyrimidin-5-amine