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(4aR,7aS)-1-ethyl-4-{[3-(3-fluorophenyl)-1H-pyrazol-4-yl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[(1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}piperidin-4-yl)oxy]pyrimidine
2-methyl-4-{5-[3-methyl-1-(quinolin-8-yl)-1H-1,2,4-triazol-5-yl]furan-2-yl}but-3-yn-2-ol
2-methyl-N-[2-phenyl-2-(piperidin-1-yl)ethyl]-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-{6-[4-(dimethylamino)azepan-1-yl]pyridin-3-yl}ethan-1-one
8-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)-3-methyl-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-(methoxymethyl)-N-methyl-N-(2-phenylethyl)-1-[4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}-4-(pyridin-2-yl)piperazine
N-[(2-ethoxyphenyl)methyl]-N-methyl-2-[(4S)-2-oxo-4-(propan-2-yl)-1,3-oxazolidin-3-yl]acetamide
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
1-(2-methoxyethyl)-2-{[3-(2-methylpropyl)pyrrolidin-1-yl]methyl}-1H-imidazole
4-ethyl-1-methyl-3-(1-{4H-thieno[3,2-b]pyrrole-5-carbonyl}piperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidine-6-carbonyl}-1,3-oxazolidin-2-one
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}propanamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-3-(methylsulfanyl)propan-1-one
N-(cyclohex-1-en-1-ylmethyl)-1-[1-(pyridin-3-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
1-ethyl-N-(2-phenylethyl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
ethyl({[4-(piperidin-1-ylmethyl)thiophen-2-yl]methyl})(pyridin-4-ylmethyl)amine
3-(3-methoxyphenyl)-N-[2-(3-methylthiophen-2-yl)ethyl]-1H-pyrazole-4-carboxamide
2-(1-{4-[2-(furan-2-yl)phenyl]-1H-1,2,3-triazol-1-yl}ethyl)-3-methylpyridine
2-{4-[5-methoxy-2-(pyrrolidine-1-carbonyl)phenoxy]piperidine-1-carbonyl}pyridine
1-[(4-fluorophenyl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
4-methyl-2-{2-[(1-methyl-3-propyl-1H-pyrazol-5-yl)formamido]ethyl}-1,3-thiazole-5-carboxylic acid
5-[3-(2-fluorophenoxymethyl)piperidine-1-carbonyl]quinoxaline
methyl 3-(cyclobutylmethoxy)-5-{[(6-hydroxypyrimidin-4-yl)methyl]carbamoyl}benzoate
9-[6-(4-methylpiperazine-1-carbonyl)pyrazin-2-yl]-3-oxa-9-azaspiro[5.5]undecane
1-[(3R,4R)-3-(azepan-1-ylmethyl)-4-(hydroxymethyl)pyrrolidin-1-yl]-2-[methyl(pyridin-4-ylmethyl)amino]ethan-1-one
5-[(2S)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
N-(1,1-dioxo-1λ6-thiolan-3-yl)-N-ethyl-2H,3H-thieno[3,4-b][1,4]dioxine-5-carboxamide
(2E)-N-{2-[2-(2-fluorophenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]ethyl}-4-methylpent-2-enamide
1-[(3S,4R)-3-[(dimethylsulfamoyl)amino]-4-(propan-2-yl)pyrrolidin-1-yl]-3-(1H-1,2,4-triazol-1-yl)propan-1-one
4-(4-tert-butyl-1H-1,2,3-triazol-1-yl)-1-(thiophene-2-sulfonyl)piperidine
2-(furan-2-yl)-1-{5-methylimidazo[1,2-a]pyridine-2-carbonyl}azepane
(2R,6R)-11-methoxy-4-[(6-methylpyridin-2-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
5-(2-fluorophenoxymethyl)-N-[(4-hydroxy-3,5-dimethylpyridin-2-yl)methyl]-1H-pyrazole-3-carboxamide
2-[4-({4-[methyl(phenyl)amino]phenyl}methyl)-1-(1-methylpiperidin-4-yl)piperazin-2-yl]ethan-1-ol
2-{4-phenyl-5-[2-(pyrrolidin-1-yl)-1,3-thiazol-5-yl]-1H-imidazol-1-yl}acetic acid
4-benzyl-3-ethyl-1-(quinoline-2-carbonyl)-1,4-diazepan-5-one
1-(6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidine-1-carbonyl}-5-methylthieno[2,3-d]pyrimidin-4-yl)azepane
4-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)morpholine
3-(2-methylpropyl)-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1,2-oxazole-5-carboxamide
(3S,4R)-4-(2H-1,3-benzodioxol-5-yl)-1-[2-(methylsulfanyl)acetyl]pyrrolidine-3-carboxylic acid
3-(1H-1,3-benzodiazol-2-yl)-1-[4-(5-chloropyridin-2-yl)piperazin-1-yl]propan-1-one
N-[(1S,2R)-2-[(1-ethylpiperidin-4-yl)amino]cyclobutyl]-3-(3-fluorophenyl)-1H-pyrazole-4-carboxamide
2-[4-cyclobutyl-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]amine
8-(3-ethoxypropanoyl)-2-(2-methylpropyl)-2,8-diazaspiro[4.5]decan-3-one
2-{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]piperidine-3-carbonyl}pyridine
(3R,5S)-5-[(2,3-dihydro-1H-inden-5-yloxy)methyl]-N-[(2-methoxyphenyl)methyl]-1-(2-methylpropyl)piperidine-3-carboxamide
6-ethyl-N-{3-[ethyl(methyl)amino]butyl}-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine