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N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-1-(thiophene-3-sulfonyl)piperidin-3-amine
methyl[(4-methyl-1H-imidazol-5-yl)methyl]{[3-(2-methylpropyl)-1,2,4-oxadiazol-5-yl]methyl}amine
2-(3,4-dimethoxyphenyl)-1-[3-(3-methoxyphenoxy)azetidin-1-yl]ethan-1-one
2-methoxy-N-[1-(1-{[4-(propan-2-yl)phenyl]methyl}piperidin-4-yl)-1H-pyrazol-5-yl]benzamide
[(2S,4R,5R)-4-({[(6-fluoro-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-5-(2-fluorophenyl)-1-methylpyrrolidin-2-yl]methanol
4-[2-({6-tert-butyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)ethyl]phenol
N-[(2S,4R,6S)-2-(5-chloro-1,3-dimethyl-1H-pyrazol-4-yl)-6-(2-phenylethyl)oxan-4-yl]acetamide
N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-4,6-dimethylpyrimidin-2-amine
({1-[2-(4-methoxyphenyl)ethyl]piperidin-3-yl}methyl)(methyl)[(2,4,6-trimethoxyphenyl)methyl]amine
N-methyl-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}oxane-4-carboxamide
(4aR,8aR)-7-(2-amino-6-methylpyrimidin-4-yl)-4a-hydroxy-N,N-dimethyl-decahydro-2,7-naphthyridine-2-sulfonamide
6-amino-1-[2-(3,4-dichlorophenyl)morpholin-4-yl]hexan-1-one
5-[4-(benzyloxy)piperidine-1-carbonyl]pyrrolidin-2-one
3-{1-[(1-methyl-1H-imidazol-2-yl)methyl]piperidin-3-yl}-N-[4-(trifluoromethyl)phenyl]propanamide
2-{[4-cyclohexyl-3-(2-hydroxyethyl)piperazin-1-yl]methyl}-6-ethoxyphenol
N-[2-(1H-imidazol-4-yl)ethyl]-4-(1,2,3,4-tetrahydroisoquinolin-2-yl)pyridine-2-carboxamide
{2-[(3S,4R)-3-(dimethylamino)-4-(4-methoxyphenyl)pyrrolidin-1-yl]-2-oxoethyl}urea
1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}-3-(5,6,7,8-tetrahydronaphthalen-2-ylmethyl)urea
4-[(4-methoxy-2-methylphenyl)methyl]-3-propylmorpholine
2-(2H-1,3-benzodioxol-5-yloxy)-N-[1-(pyridin-2-ylmethyl)piperidin-3-yl]acetamide
6-[2-(aminomethyl)-2,3-dihydro-1-benzofuran-7-yl]-2H-1,3-benzodioxole-5-carboxamide
2-(2-methanesulfonylethyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
2-(2-methyl-6-{4-[1-(4-methylpiperazin-1-yl)ethyl]piperidin-1-yl}pyrimidin-4-yl)ethan-1-amine
2-amino-4-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
2-{3-[(3-hydroxyazetidin-1-yl)methyl]phenyl}-6-(4-methoxyphenyl)-3,4-dihydropyrimidin-4-one
1-(4-{3-[3-(propan-2-yloxy)benzoyl]piperidin-1-yl}piperidin-1-yl)ethan-1-one
1-benzyl-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-methanesulfonamido-2-methyl-1H-1,3-benzodiazole-7-carboxamide
6-(1-benzofuran-2-carbonyl)-N-[(6-methylpyridin-2-yl)methyl]-6-azaspiro[2.5]octane-1-carboxamide
6,8-dimethoxy-4-methyl-2-(oxan-2-ylmethyl)quinoline
1-(4-methanesulfonylphenyl)isoquinoline
N-(1H-indol-4-ylmethyl)-6-methyl-2-(morpholin-4-yl)pyrimidin-4-amine
1-(4-methylphenyl)-4-(quinoline-5-carbonyl)piperazin-2-one
1-{imidazo[1,2-b]pyridazin-6-yl}-4-[2-(methylsulfanyl)-1,3-thiazole-4-carbonyl]piperazine
1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidine
4-hydroxy-N-{[5-(2-methoxyethyl)-1,2,4-oxadiazol-3-yl]methyl}-2-(2-methyl-1,3-thiazol-4-yl)pyrimidine-5-carboxamide
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-3-(2-methoxyphenyl)-N-methyl-1H-pyrazole-5-carboxamide
5-{1-[(2,3-difluoro-6-methoxyphenyl)methyl]pyrrolidin-2-yl}-3-(propan-2-yl)-1,2,4-oxadiazole
1-[4-(2-chlorophenoxy)piperidin-1-yl]-6-methoxyhexan-1-one
(2S,4R)-1-benzyl-N-methyl-4-{[2-(2,6,6-trimethylcyclohex-1-en-1-yl)ethyl]amino}pyrrolidine-2-carboxamide
7-{[4-(benzyloxy)piperidin-1-yl]methyl}-4-(cyclopropylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
N-[2-(4-ethyl-4H-1,2,4-triazol-3-yl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
methyl (1R,3S,3aR,6aS)-3-(3-ethenylphenyl)-1,5-diethyl-4,6-dioxo-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
(2S,4S)-4-amino-1-methyl-N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}pyrrolidine-2-carboxamide
N-{[4-(3-methylpiperidin-1-yl)phenyl]methyl}-5-(1H-pyrazol-1-ylmethyl)furan-2-carboxamide
2-methoxy-2-phenyl-1-{3-phenyl-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl}ethan-1-one
(2-ethoxy-5-{[2-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-4-yl]methyl}phenyl)methanol
3-[9-oxo-8-(2-phenylethyl)-2,8-diazaspiro[5.5]undecan-2-yl]propanamide
ethyl 4-[(4-chlorophenyl)methyl]-1-(3-methyl-2-oxopentanoyl)piperidine-4-carboxylate
3-[(3R,7S,8aS)-3-(hydroxymethyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
1-(4-methyl-1,3-oxazole-5-carbonyl)-3-[2-(2-methylphenyl)ethyl]piperidine