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N-{2-[4-(quinolin-2-ylmethyl)morpholin-2-yl]ethyl}acetamide
2-[4-({[(5-cyclopropyl-1H-pyrazol-3-yl)methyl](methyl)amino}methyl)phenyl]-3,4,5,6,7,8-hexahydroquinazolin-4-one
N-[3-(dimethylamino)-1-phenylpropyl]-2-(ethylamino)pyrimidine-5-carboxamide
N-ethyl-2-methyl-6-(piperidin-4-yl)-N-(pyridin-4-ylmethyl)pyrimidin-4-amine
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
(furan-2-ylmethyl)(methyl)[(2,3,4-trimethoxyphenyl)methyl]amine
(2S)-4-methyl-2-{[2-(3-phenylpropyl)-1,3-benzoxazol-5-yl]formamido}pentanamide
2-{1-[1-(2-ethylhexyl)piperidin-4-yl]-1H-1,2,3-triazol-4-yl}propan-2-ol
2-methyl-N-(oxan-4-ylmethyl)pyrido[2,3-d]pyrimidin-4-amine
N-[(5-methyl-1H-imidazol-4-yl)methyl]-1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-amine
methyl 1-{4-[4-(3-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}cyclopropane-1-carboxylate
2-{1-[(4-methylphenyl)methyl]-3-oxopiperazin-2-yl}-N,N-dipropylacetamide
2,3-dimethyl-6-[(3R,5R)-5-(morpholine-4-carbonyl)piperidine-3-carbonyl]-3H,4H,5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-one
1-[4-(adamantan-1-yl)piperazin-1-yl]-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
N-ethyl-5-[4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine-1-carbonyl]pyrimidin-2-amine
5-{1-[2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetyl]pyrrolidin-2-yl}thiophene-2-carboxamide
9-(cyclohex-3-en-1-ylmethyl)-2-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-(3-aminopropyl)-1-[(4-methylphenyl)amino]cyclopentane-1-carboxamide
4-(1-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-1H-imidazol-2-yl)-1,5-dimethyl-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
N-ethyl-5-{[3-(pyridin-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}pyrimidin-2-amine
7-(5-chloropyridin-2-yl)-4-(pyrimidin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2-methoxyethyl)[(3-methylthiophen-2-yl)methyl](pyridin-2-ylmethyl)amine
5-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]furan-2-carboxamide
N-[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]-3-(methylsulfanyl)propanamide
N-{[3-cyclopropyl-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazol-5-yl]methyl}acetamide
N-ethyl-N-{[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}-4-(1H-1,2,3,4-tetrazol-1-yl)benzamide
5-{[(2S,4R)-4-amino-2-(ethylcarbamoyl)pyrrolidin-1-yl]methyl}-2-hydroxybenzoic acid
1-{5,7-dimethyl-[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}-4-(pyridin-3-yl)piperidin-4-ol
(4aS,8aR)-1-butyl-6-[(5-methoxy-1H-indazol-3-yl)methyl]-decahydro-1,6-naphthyridin-2-one
1-{[3-(cyclopropylmethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(4-methoxybenzoyl)piperazine
(2R,3R)-3-{[3-(1H-1,2,3-triazol-1-yl)propyl]amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
1-{dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-4-(furan-3-carbonyl)-1,4-diazepane
5-[4-(thiophen-2-ylmethyl)-1,4-diazepane-1-carbonyl]-1H-1,2,3-benzotriazole
2-(3-methoxypropyl)-9-(oxan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 3-{3-[(4-methoxyphenyl)methyl]-1-(2-methylpropyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-8-yl}propanoate
N,2-dimethyl-N-[1-(pyridin-3-yl)ethyl]pyridine-3-carboxamide
N-[(2-chlorophenyl)methyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-{1-[(3-methoxyphenyl)methyl]-5-(prop-2-en-1-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-3-ol
2-methyl-N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}oxane-2-carboxamide
N-(butan-2-yl)-N-(pyridin-4-ylmethyl)-4-(thiophen-2-yl)butanamide
N-[2-(6-hydroxy-2-methylpyrimidin-4-yl)ethyl]-4-(piperidin-3-yl)benzamide
5-(azepane-1-carbonyl)-1-(2-ethoxyethyl)-2,3-dihydro-1H-1,3-benzodiazol-2-one
1-(2-tert-butyl-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-5-yl)-3-(prop-2-en-1-yl)urea
(3R,4R)-4-amino-1-({4-[3-(1H-imidazol-1-yl)propoxy]phenyl}methyl)piperidin-3-ol
3-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-5-carbonyl]pyridin-2-ol
1'-(3-methyl-1H-pyrazole-5-carbonyl)-5-(2-methylpropyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]-1-(thian-4-yl)pyrrolidine-2-carboxamide
5-{1-[(2-chloro-6-fluorophenyl)methyl]-3-ethyl-1H-1,2,4-triazol-5-yl}-1-methyl-1H-pyrrole-3-carbonitrile
2-{1-[(2-fluorophenyl)methyl]-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl}-N-(2-hydroxyethyl)acetamide
5-(4-chloro-2-methoxyphenoxymethyl)-N-(3-hydroxypropyl)-N-methyl-1,2-oxazole-3-carboxamide