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8-(3,6-dimethyl-1-benzofuran-2-carbonyl)-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
N-{2-[(3,5-dimethyl-1H-pyrazol-4-yl)sulfanyl]phenyl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)acetamide
5-[1-(2-methyl-1,3-thiazole-4-carbonyl)pyrrolidin-2-yl]-3-phenyl-1,2,4-oxadiazole
4-phenyl-1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidine-4-carbonitrile
(4aS,8aR)-1-(2-aminoethyl)-6-(1,2,3,4-tetrahydroquinoline-8-carbonyl)-decahydro-1,6-naphthyridin-2-one
N-methyl-4-(2-methyl-1H-imidazol-1-yl)-N-(quinolin-5-ylmethyl)butanamide
2-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[2-(4,5,6,7-tetrahydro-2H-indazol-3-yl)ethyl]acetamide
1,3-dimethyl-N-{[1-(pyrrolidin-1-yl)cyclopentyl]methyl}-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3S,4S)-4-cyclopropyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}pyrrolidine-3-carboxylic acid
1-(azocan-1-yl)-3-[4-({[(3-ethyl-1,2-oxazol-5-yl)methyl]amino}methyl)-2-methoxyphenoxy]propan-2-ol
1-[3-({[(5-methylfuran-2-yl)methyl]amino}methyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
1-butyl-5-(pentan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazole
6-[(2R,6S)-6-phenyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridine-1-carbonyl]-2,3-dihydropyridazin-3-one
5-[1-(2-ethoxyacetyl)pyrrolidin-2-yl]-N-[(3-fluorophenyl)methyl]thiophene-2-carboxamide
1,6-dimethyl-N-[3-(1H-1,2,3,4-tetrazol-5-yl)propyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-(1,4-diazepane-1-carbonyl)-2,6-dimethylquinoline
1-(2-{5-butyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-4-methylphenyl)-1H-pyrazole
N-(oxan-4-yl)-3-[5-(4-phenylphenyl)-1,3,4-oxadiazol-2-yl]propanamide
(3S,9aR)-3-[(2S)-butan-2-yl]-8-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
[4-({[(2,2-diphenylcyclopropyl)methyl](methyl)amino}methyl)oxan-4-yl]methanol
N-butyl-3-({4-[(dimethylcarbamoyl)methyl]piperazin-1-yl}methyl)-N-methylimidazo[1,2-a]pyridine-2-carboxamide
{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]-3-(2-methoxyethyl)piperidin-3-yl}methanol
N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-3-[(3-methylbutyl)amino]-5-[(propan-2-yl)sulfamoyl]benzamide
4-(4-{[(1-benzyl-1H-pyrazol-4-yl)methyl]amino}piperidin-1-yl)-N-[(2-fluorophenyl)methyl]benzamide
N-[2-(5-ethyl-1,2,4-oxadiazol-3-yl)ethyl]-1-{2-methylthieno[2,3-d]pyrimidin-4-yl}piperidin-4-amine
1-(cyclohexylmethyl)-N-cyclopropyl-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]-4-oxo-1,4-dihydropyridine-3-carboxamide
2,5,6-trimethyl-N-{[4-(piperidine-1-carbonyl)phenyl]methyl}pyrimidin-4-amine
2-(3-fluorophenoxymethyl)-N-(2-hydroxypropyl)-N-methyl-1,3-oxazole-4-carboxamide
3-butanamido-N-(2-methoxyethyl)-4-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
2-(2-{[(3R,4R)-4-(piperidin-1-yl)oxolan-3-yl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
N-[2-(benzyloxy)ethyl]-8-methoxy-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
6-(aminomethyl)-N-(2-{[3-methyl-5-(trifluoromethyl)-1H-pyrazol-1-yl]methyl}propyl)pyrimidin-4-amine
N-({3-[(2-fluorophenyl)methoxy]-4-methoxyphenyl}methyl)-N-(pyridin-4-ylmethyl)-4-(trifluoromethyl)benzamide
ethyl({[1-(1-methylpiperidin-4-yl)piperidin-4-yl]methyl}){[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}amine
4-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-3-yl)pyrimidine
7-(cyclopropylmethyl)-2-(2,3-dimethoxybenzoyl)-2,7-diazaspiro[4.5]decan-6-one
4-[(3,5-dimethoxyphenyl)methyl]-7-(thiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
1-(2-methoxybenzoyl)-4-(2-methylquinolin-6-yl)piperidin-4-ol
4-{1-[3-(1-methyl-1H-pyrazol-5-yl)propanoyl]piperidin-3-yl}benzoic acid
1-(2-aminopyrimidin-4-yl)-4-[3-(furan-2-yl)-1H-pyrazol-1-yl]piperidine-4-carboxylic acid
9-(1H-imidazol-2-ylmethyl)-3-oxa-9-azaspiro[5.5]undecane
5-(1-{[2,4-dimethyl-6-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-2-yl)-3-methyl-1H-1,2,4-triazole
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2-(3-phenylpropyl)-1,3-benzoxazole-5-carboxamide
7-fluoro-3-[2-(4-methylpiperazin-1-yl)ethyl]-3,4-dihydroquinazolin-4-one
1-(azocan-1-yl)-4-[3-(1-methoxypropan-2-yl)-3H-imidazo[4,5-b]pyridin-2-yl]butan-1-one
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-2-(4-fluoro-2-methylphenyl)ethan-1-one
3-{4-[(5-cyclopropyl-1,2,4-oxadiazol-3-yl)methyl]piperidine-1-carbonyl}-2,8-diazaspiro[4.5]decane
4-[(4-fluorophenyl)methyl]-7-(pyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
6-fluoro-2-[({[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}amino)methyl]quinolin-4-ol
[1-(1-benzofuran-5-carbonyl)-3-(cyclopropylmethyl)piperidin-3-yl]methanol