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ethyl 2-{4-[1-(3-phenylpropyl)-1H-1,2,3-triazole-4-carbonyl]morpholin-3-yl}acetate
2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)-N-(propan-2-yl)acetamide
2-[4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)-1-(thiophen-2-ylmethyl)piperazin-2-yl]ethan-1-ol
methyl[(1-methyl-1H-pyrazol-4-yl)methyl][(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-N-[(2-methylphenyl)methyl]pyridine-2-carboxamide
3-(4-methyl-1,2,3,6-tetrahydropyridine-1-carbonyl)-N-(oxan-4-yl)benzene-1-sulfonamide
2-(ethylsulfanyl)-1-[7-(pyrrolidine-1-sulfonyl)-1,2,3,4-tetrahydroisoquinolin-2-yl]propan-1-one
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-6-methylimidazo[1,2-a]pyridine-2-carboxamide
5-(isoquinolin-5-yl)-N-propylfuran-2-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-{[1-(oxan-4-yl)piperidin-4-yl]oxy}benzamide
3-(1-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}piperidin-3-yl)benzoic acid
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methoxyethyl)-8-(1-methoxypropan-2-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
(2S,4R)-4-amino-N-(4-phenylbutyl)pyrrolidine-2-carboxamide
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-2-(1H-1,2,3,4-tetrazol-1-yl)acetamide
(4aR,7aS)-1-propyl-4-(pyridine-3-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-{[2-(2-methylpropoxy)phenyl]methyl}acetamide
N-[(1R,2R)-2-(benzyloxy)cyclopentyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
2-(methoxymethyl)-1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)piperidine
2-[3-(4-methyl-1,4-diazepane-1-carbonyl)piperidin-1-yl]acetamide
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-[1,2,3,4]tetrazolo[1,5-a]pyridine-7-carboxamide
2-(3,4-dihydro-1H-2-benzopyran-1-yl)-7,7-dimethyl-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
(3R,4R)-3-cyclobutyl-4-methyl-1-[4-(4-methylpiperazin-1-yl)benzoyl]pyrrolidin-3-ol
1-[4-(4-methoxyphenoxy)piperidine-1-carbonyl]-6-azaspiro[2.5]octane
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(pyrrolidine-1-sulfonyl)piperazine
(1R,5R)-6-(cyclopropylmethyl)-N-[2-(trifluoromethyl)phenyl]-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N-(1-cyclohexyl-1H-pyrazol-5-yl)-2-cyclopropylacetamide
5-(methoxymethyl)-N-[4-(5-methyl-4-{[2-(2-methyl-1,3-thiazol-4-yl)acetamido]methyl}-1,3-oxazol-2-yl)phenyl]furan-2-carboxamide
5-[4-(thian-4-yl)piperazine-1-carbonyl]quinoxaline
2-(2,6-dimethoxypyridin-3-yl)-2-{methyl[2-(piperidin-1-yl)ethyl]amino}acetic acid
[(2S,6S)-4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(9),10,12-trien-6-yl]methanol
4-[2-(3-methoxypropyl)piperidine-1-carbonyl]benzene-1-sulfonamide
2-{4-[4-(methylsulfanyl)phenyl]-1H-1,2,3-triazol-1-yl}ethan-1-amine
1-methyl-2-oxo-8-{[4-(trifluoromethyl)phenyl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylic acid
{1-[3-(propan-2-yl)-1,2-oxazole-5-carbonyl]piperidin-4-yl}(pyridin-2-yl)methanol
2-[(3S,4R)-3-acetamido-4-(4-methylphenyl)pyrrolidin-1-yl]-6-methylpyridine-3-carboxylic acid
1-[4-(dimethylamino)-5-fluoropyrimidin-2-yl]-3-(hydroxymethyl)pyrrolidin-3-ol
N-[1-(3,5-difluorophenyl)cyclopropyl]-6-methoxy-1-methyl-1H-indole-2-carboxamide
N-{2-methyl-3-[(3-phenylprop-2-yn-1-yl)(propyl)carbamoyl]phenyl}oxolane-2-carboxamide
1-[1-ethyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
5-cyclopropyl-N-(2-hydroxyethyl)-N-methyl-1-[5-methyl-4-(thiophen-2-yl)pyrimidin-2-yl]-1H-pyrazole-4-carboxamide
5-[(4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}piperidin-1-yl)methyl]-2-methyl-1H-pyrrole-3-carbonitrile
4-{6-[1-(3-ethyl-1,2-oxazole-5-carbonyl)piperidin-3-yl]-2-methylpyrimidin-4-yl}morpholine
1-[(2,6-difluorophenyl)methyl]-N-(1-methoxybutan-2-yl)-1H-1,2,3-triazole-4-carboxamide
1-[3-(cyclohexylsulfanyl)propyl]-3-[2-fluoro-5-(4H-1,2,4-triazol-4-yl)phenyl]urea
1-{3-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]-3-phenylpropyl}-1H-1,2,4-triazole
1-[(2,4,5-trimethylphenyl)methyl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
4-(pyridin-3-yl)-2-[4-(1,3-thiazol-2-yl)piperazin-1-yl]pyrimidine
3-chloro-N-cyclopentyl-4-{[1-(3-methyl-1H-pyrazole-4-carbonyl)piperidin-4-yl]oxy}benzamide
[4-(2,3-dimethylquinoxaline-6-carbonyl)-1,4-oxazepan-6-yl]methanol
[2-(3-fluorophenyl)ethyl]({[6-(pyrrolidin-1-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine