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N-[(1-ethylpiperidin-3-yl)methyl]-1,6-dimethyl-4-oxo-1,4-dihydroquinoline-3-carboxamide
3-[methyl(1,2-oxazol-3-ylmethyl)sulfamoyl]-N-(oxan-4-ylmethyl)benzamide
N5-cyclooctyl-N3-[2-(diethylamino)ethyl]-N3-methyl-4-oxo-1-(pyridin-2-ylmethyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-{1-[(2-fluoro-4-methoxyphenyl)methyl]-4-[(5-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperazin-2-yl}ethan-1-ol
N-[(3S,4R)-4-propyl-1-{[3-(pyridin-2-yl)-1,2-oxazol-5-yl]methyl}pyrrolidin-3-yl]methanesulfonamide
3-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
methyl[(2-methyl-1,3-oxazol-4-yl)methyl]{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}amine
2-(2,4-dioxo-1,3-diazinan-1-yl)-N-methyl-N-[1-(pyrimidin-4-yl)ethyl]benzamide
7-chloro-N-{2-[2-(hydroxymethyl)piperidin-1-yl]ethyl}-3,5-dimethyl-1-benzofuran-2-carboxamide
N,N-dimethyl-4-{3-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]phenyl}benzamide
N-({1-[2-(1H-indol-3-yl)ethyl]-1,2,5,6-tetrahydropyridin-3-yl}methyl)acetamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-oxo-2-(piperazin-1-yl)ethyl]pyrrolidin-3-yl]acetamide
3-methyl-1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-4-yl]butan-1-ol
2-{3-[3-(3-chloropyridin-2-yl)phenyl]-1H-pyrazol-1-yl}-1-(morpholin-4-yl)ethan-1-one
3-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-1,5-dimethyl-1H-indazole
6-{3-[3-(1H-imidazol-2-yl)piperidin-1-yl]-3-oxopropyl}-2,3,4,5-tetrahydropyridazin-3-one
4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(oxan-4-yl)piperidine
2-[2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)ethyl]-3,4-dihydroquinazolin-4-one
N-{1-[1-(2-chloro-4-fluorobenzoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-methylbutanamide
N-[(3R,4S)-4-cyclopropyl-1-(2,2-dimethylpropanoyl)pyrrolidin-3-yl]-2-methyl-1H-1,3-benzodiazole-5-carboxamide
(3S,4S)-1-[3-(dimethyl-1,2-oxazol-4-yl)propanoyl]-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
2-[(1,3-benzothiazol-2-yl)amino]-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
N-{1-[7-(2-methoxypyridine-3-carbonyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]-2-methylpropyl}oxolane-3-carboxamide
1-(2-methoxy-4-{[(2-phenylethyl)amino]methyl}phenoxy)-3-(morpholin-4-yl)propan-2-ol
1-{[3-(2,5-dimethylthiophen-3-yl)-1-(2-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-4-ol
{[3-(2-chlorophenyl)-1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(pyridin-3-ylmethyl)amine
1-[6-(4-fluorophenyl)pyridine-3-carbonyl]-4-phenylazepane
(1S,5R)-6-[2-(4-chloro-1H-pyrazol-1-yl)ethyl]-3-[(4-methoxyphenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-4-{4-[(3-methoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-N-[2-(methylsulfanyl)phenyl]acetamide
1-methyl-4-[5-methyl-6-(3-phenylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]piperazine
1-(2-{[(3-chloro-2-methylphenyl)carbamoyl]amino}ethyl)piperidine-3-carboxamide
3-(dimethyl-1H-1,2,4-triazol-3-yl)-1-(1,4-dioxan-2-ylmethyl)urea
2,5-dimethoxy-N-(2-{4-methyl-5-[(oxolan-2-ylmethyl)sulfanyl]-4H-1,2,4-triazol-3-yl}ethyl)benzamide
[3-(3-phenylpropyl)-1-(9H-purin-6-yl)piperidin-3-yl]methanol
5-[(3-fluorophenyl)methyl]-3-(2-methylpropyl)-5-[1-(pyrazine-2-carbonyl)piperidin-4-yl]imidazolidine-2,4-dione
4-{[(2R,5S)-5-[(6-methoxypyridin-3-yl)methyl]oxolan-2-yl]methyl}thiomorpholine
3-methyl-1-[(4-methylphenyl)methyl]-4-{1H-pyrrolo[2,3-b]pyridin-6-yl}piperazin-2-one
3-(5-methyl-1H-pyrazol-1-yl)-1-[2-(morpholine-4-carbonyl)piperazin-1-yl]propan-1-one
3-(3-methoxyphenyl)-1-[(1S,5R)-3-(pyrazin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one
(3S,4R)-4-(pyridin-3-yl)-1-(quinolin-5-ylmethyl)pyrrolidine-3-carboxylic acid
8-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-8-azaspiro[4.5]decane-7,9-dione
N-[(2-ethyl-3,5-dimethyl-1H-indol-7-yl)methyl]-2-methylpyrimidine-5-carboxamide
N-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2-{2-methylimidazo[1,2-a]pyridin-3-yl}acetamide
1-{4-[(1R,9aR)-octahydro-1H-quinolizin-1-ylmethoxy]-2-methylphenyl}ethan-1-one
N-[4-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-1H-indazole-3-carboxamide
(1R,5R)-3-[3-(piperidine-1-carbonyl)pyrazine-2-carbonyl]-6-propyl-3,6-diazabicyclo[3.2.2]nonane
2-{5-[5-(3-hydroxy-3-methylbut-1-yn-1-yl)thiophen-2-yl]-4-phenyl-1H-imidazol-1-yl}acetamide
(2S)-2-amino-N-({6-cyclopentyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)butanamide
4-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-1H-imidazole