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7-(cyclobutylmethyl)-2-[2-(1H-1,2,4-triazol-1-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one
ethyl 4-[(4-cyclobutanecarbonyl-1,4-diazepane-1-carbonyl)amino]benzoate
2-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-1-methylazepane
N-[(3S,5S)-1-cyclopentyl-5-(diethylcarbamoyl)pyrrolidin-3-yl]-2-methylpyrimidine-5-carboxamide
7-(2-methylphenyl)-4-(piperidin-4-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-(2-hydroxyethyl)-4-methyl-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-phenylpyrimidine-5-carboxamide
2-[2-(2,3-dihydro-1,4-benzodioxin-6-yl)-2-oxoethyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
9-[(5-fluoro-2-methoxyphenyl)methyl]-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
2-{3-oxo-9-[(5-propylfuran-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
4-(2,5-difluorobenzoyl)-1-[(3,5-dimethylphenyl)methyl]piperazin-2-one
N-[(2-chloro-6-fluorophenyl)methyl]-6-(methoxymethyl)pyrimidin-4-amine
N,2-dimethyl-6-(piperidin-4-yl)-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-4-amine
2-[(1-benzylpiperidin-4-yl)amino]-N,N-dimethylethane-1-sulfonamide
9-(2-chlorophenyl)-15-methyl-12-(pyrrolidine-1-carbonyl)-8-thia-1-azatricyclo[9.4.0.02,7]pentadeca-2(7),3,5,11,14-pentaen-13-one
1,3-dimethyl-N-[3-(propan-2-yloxy)propyl]-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-({5,7-dimethylpyrido[2,3-d]pyrimidin-4-yl}amino)-3-(pyrrolidin-1-yl)propan-2-ol
2-(4-chlorophenyl)-1-{3-[(dimethylsulfamoyl)amino]azepan-1-yl}ethan-1-one
1-benzyl-5-{[(5-methoxy-1H-1,3-benzodiazol-2-yl)methyl]amino}azepan-2-one
2-methyl-4-phenyl-9-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-{2-[3-(methoxymethyl)piperidin-1-yl]-2-oxoethyl}-3-phenyl-1-(thiophen-2-ylmethyl)pyrrolidine-2,5-dione
3-[(3R,4S)-1-[(3-ethylphenyl)carbamoyl]-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
(3R,5S)-N3-methyl-N5-(4-methylphenyl)-N3-[(3-methylpyridin-2-yl)methyl]piperidine-3,5-dicarboxamide
(3aR,5R,6S,7aS)-2-{[3-(4-methylphenyl)-1,2-oxazol-5-yl]methyl}-octahydro-1H-isoindole-5,6-diol
N-[2-(3-methoxyphenyl)-1-{1-[2-(2-methyl-1,3-thiazol-4-yl)acetyl]piperidin-4-yl}ethyl]-N-methyl-3-(methylsulfanyl)propanamide
5-[1-ethyl-3-(pyrrolidine-1-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole
1-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}-4-(pyridin-3-ylmethyl)piperazine
N-benzyl-N-methyl-3-(morpholine-4-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-{3-methyl-3,9-diazaspiro[5.6]dodecane-9-carbonyl}pyridin-3-ol
1-cycloheptyl-5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidin-2-one
N-{[1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}-2-methylpyrido[2,3-d]pyrimidin-4-amine
4-(thiophen-3-ylmethyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
(3R,9aR)-8-(4-chlorobenzoyl)-3-[(4-hydroxyphenyl)methyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-{9-[(1-methyl-1H-imidazol-2-yl)methyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}propanoic acid
6-[1-(2,3-dihydro-1-benzothiophene-2-carbonyl)piperidin-4-yl]-2-methylpyrimidin-4-ol
3-{4-[(3-methylphenyl)sulfanyl]piperidine-1-carbonyl}-1H-indazole
methyl (1R,3S,3aR,6aS)-1,5-dimethyl-4,6-dioxo-3-[1-(prop-2-en-1-yl)-1H-1,3-benzodiazol-2-yl]-octahydropyrrolo[3,4-c]pyrrole-1-carboxylate
2-(8-methoxy-2-methylquinolin-5-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
3-(1-{2-[3-(pyridin-4-yl)-1H-1,2,4-triazol-5-yl]ethyl}-1H-imidazol-2-yl)-1,2-dihydroquinolin-2-one
2,6-dimethyl-4-[3-(pyridin-3-yloxy)azetidine-1-carbonyl]quinoline
3,5-dimethoxy-2-[(3-oxopiperazin-1-yl)methyl]benzoic acid
N-[(2,3-dimethylphenyl)methyl]-3-(4H-1,2,4-triazol-4-yl)benzamide
(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-3-(2-methyl-6-propylpyrimidin-4-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
{4-[6-(pyrrolidine-1-carbonyl)pyrazin-2-yl]phenyl}methanol
5-[2,2-bis(prop-2-en-1-yl)pyrrolidine-1-carbonyl]-1-[(4-chlorophenyl)methyl]piperidin-2-one
N-{[4-(1H-1,3-benzodiazol-2-yl)cyclohexyl]methyl}-2-methyl-1,3-thiazole-4-carboxamide
N-[1-(1H-indol-5-yl)ethyl]-3-(pyridin-4-yl)-1H-pyrazole-5-carboxamide
2-{1-[2-(1-methylpyrrolidin-2-yl)ethyl]-1H-imidazol-2-yl}-1H-1,3-benzodiazole
4-(5-acetylthiophen-3-yl)-3-(propan-2-yl)-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
(1R,5R)-6-[2-(2H-indazol-2-yl)acetyl]-N,N-dimethyl-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
N,N-dimethyl-6-(3-methyl-3-phenylpiperidin-1-yl)pyridine-3-carboxamide