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4-(naphthalen-2-yloxy)-1-(9H-purin-6-yl)piperidine-4-carboxylic acid
N-{1-[1-(3-cyclopentylpropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-fluorobenzamide
9-(6-methyl-4-oxo-4H-pyran-2-carbonyl)-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[(5-methylfuran-2-yl)methyl]-3-{5-[(3-methylphenyl)methyl]-1,3,4-oxadiazol-2-yl}propanamide
N3-(1-benzylpyrrolidin-3-yl)-N5-tert-butyl-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
4-(3,5-dimethyl-1-phenyl-1H-pyrazol-4-yl)-N-methyl-N-(pyridin-2-ylmethyl)pyrimidin-2-amine
6-(cyclohexylamino)-1-(pyridin-3-ylmethyl)-1H,4H,5H,8H-imidazo[4,5-e][1,3]diazepine-4,8-dione
N-[(3R,4R)-3-hydroxy-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidin-4-yl]pyridine-2-carboxamide
N,N-dimethyl-3-[4-(trifluoromethoxy)phenyl]-1H-1,2,4-triazol-5-amine
1-[3-(azetidin-1-ylmethyl)phenoxy]-3-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-2-ol
N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]-4-(3,3,3-trifluoropropyl)pyrimidin-2-amine
(3R,4R)-4-cyclobutyl-3-methyl-1-(quinoxalin-2-yl)piperidin-4-ol
3-fluoro-4-[3-(2-methoxyphenoxy)propyl]benzene-1-sulfonamide
(butan-2-yl)({[4-methoxy-3-(methoxymethyl)phenyl]methyl})(pyridin-3-ylmethyl)amine
1-[(4-propyl-4H-1,2,4-triazol-3-yl)methyl]-3-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]urea
N-[2-(4-fluorophenyl)ethyl]-2-phenyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
{[6-(cyclohexylmethoxy)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl}(pyridin-2-ylmethyl)amine
N-[3-(cyclohexylsulfanyl)propyl]-1,3-dimethyl-1H-pyrazole-5-carboxamide
1-[3-(1H-imidazol-2-yl)phenyl]-3,5-dimethyl-1H-pyrazole
(3S,5R)-1-[(4,5-dimethylfuran-2-yl)methyl]-5-[(pyridin-4-ylmethyl)carbamoyl]piperidine-3-carboxylic acid
methyl 2-(azepane-1-sulfonyl)-6-(3-fluorobenzoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
{4-[2-(trifluoromethyl)phenyl]-4H-1,2,4-triazol-3-yl}methanamine
1-[(2-chlorophenyl)methyl]-3-({[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]amino}methyl)-7-(methylsulfanyl)-1,2-dihydroquinolin-2-one
N-[1-(pyrrolidin-1-ylmethyl)cyclohexyl]-2-(trifluoromethyl)pyrimidin-4-amine
1-cyclopentyl-N-[4-(pyridin-3-yloxy)phenyl]piperidine-2-carboxamide
4-{4-[(3-methylpyridin-2-yl)methyl]piperazin-1-yl}pyrimidine-5-carboxylic acid
9-[2-(3-ethoxyphenoxy)ethyl]-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
3-{4-[2-(2-hydroxyethyl)piperidin-1-yl]-4-oxobutyl}-3,4-dihydroquinazolin-4-one
1-[(2-fluoro-5-methoxyphenyl)methyl]-3-({[(3-fluorophenyl)methyl]amino}methyl)-3-hydroxypiperidin-2-one
1-{4-[(3S,4R)-4-hydroxyoxolan-3-yl]-1,4-diazepan-1-yl}-2-(1-propylpiperidin-4-yl)ethan-1-one
8-[(4-carboxy-1,3-oxazol-2-yl)methyl]-2-cyclopropanecarbonyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
1-[1-(1-methyl-1H-imidazol-2-yl)butyl]-3-[1-(2-methylpropyl)-1H-pyrazol-5-yl]urea
1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-N-cyclopropyl-1H-1,2,3-triazole-4-carboxamide
4-(pyridin-3-yl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}pyrimidin-2-amine
N-[(3R,4S)-1-(3-hydroxypropyl)-4-propylpyrrolidin-3-yl]-1-methyl-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-carboxamide
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}(1,4-dioxan-2-ylmethyl)methylamine
(3S)-N-benzyl-3-(3-methoxyphenyl)piperidine-1-sulfonamide
N-[1-(cyclohexylmethyl)piperidin-3-yl]-3-(methylsulfanyl)propanamide
(4aS,8aR)-1-(2-aminoethyl)-6-[2-(dimethyl-1,2-oxazol-4-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
4-{[ethyl(pyridin-4-ylmethyl)amino]methyl}-N-(1,2,4-thiadiazol-5-yl)benzamide
N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
6-(4-{[4-(1H-pyrazol-1-ylmethyl)phenyl]methyl}piperazin-1-yl)pyridine-2-carbonitrile
N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethylpyrazine-2-carboxamide
2-{2-[4-(furan-2-carbonyl)-1,4-diazepan-1-yl]-2-oxoethyl}-1H,2H-pyrrolo[1,2-d][1,2,4]triazin-1-one
methyl 1-{[3-(3-fluorophenyl)-1-(3-methylphenyl)-1H-pyrazol-4-yl]methyl}piperidine-4-carboxylate
1-(but-2-ynoyl)-N-[3-(4-fluorophenyl)phenyl]piperidine-3-carboxamide
2-methyl-6-{3-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}pyridine
N-butyl-2-[2-(ethylsulfanyl)-1,3-thiazol-4-yl]-N-(pyridin-3-ylmethyl)acetamide
5-(cyclopentylamino)-1-ethyl-N-(pyridin-4-ylmethyl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[1-(2,2-dimethylpropanoyl)piperidin-4-yl]-N-(propan-2-yl)-1H-1,2,3-triazole-4-carboxamide