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N-ethyl-4-[2-(2-phenyl-1H-imidazol-1-yl)acetamido]piperidine-1-carboxamide
2-[(3-ethyl-1H-1,2,4-triazol-5-yl)sulfanyl]-1-[2-(1,3-thiazol-2-yl)piperidin-1-yl]ethan-1-one
2-(2,5-dimethylphenoxy)-N-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}propanamide
5-{4-[(3-fluorophenyl)methyl]piperazine-1-carbonyl}-2-phenyl-2,3-dihydro-1H-pyrazol-3-one
5-{4-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-6-hydroxy-1,4-diazepane-1-carbonyl}-1H-pyrrole-3-carbonitrile
3-{[(5-fluoro-1H-indol-2-yl)methyl](methyl)amino}-N-(pyridin-3-yl)propanamide
1-cyclopentyl-4-[5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-imidazol-2-yl]pyrrolidin-2-one
4-[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}butanamide
1-(2H-1,3-benzodioxol-5-ylmethyl)-4-[(1-propyl-1H-imidazol-2-yl)methyl]piperazin-2-one
4-[({1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}carbamoyl)amino]-N-(oxolan-2-ylmethyl)benzamide
2-[2-(2,6-dimethoxyphenyl)phenyl]-5-methyl-1,3,4-oxadiazole
N-[3-(azepan-1-yl)-2-hydroxypropyl]-3-(2-methylpropyl)-1,2-oxazole-5-carboxamide
4-(1H-imidazol-1-ylmethyl)-1-(6-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)piperidin-4-ol
2-[(5-methylpyrazin-2-yl)methyl]-8-propanoyl-2,8-diazaspiro[5.5]undecan-3-one
N-[2-(furan-2-ylmethyl)-3-hydroxypropyl]-2-(2,2,6,6-tetramethylpiperidin-4-yl)acetamide
(4aS,8aR)-1-(3-aminopropyl)-6-[3-(1-methyl-1H-pyrazol-4-yl)propanoyl]-decahydro-1,6-naphthyridin-2-one
6-(2-methoxyphenyl)-N-[(2-methyloxolan-2-yl)methyl]pyridazin-3-amine
7-(1,3-benzothiazol-2-yl)-4-(piperidine-4-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(2,3-dihydro-1-benzofuran-2-carbonyl)piperazin-1-yl]quinazoline
2-(2-{4-[(4-methylphenyl)sulfanyl]piperidin-1-yl}-2-oxoethyl)-1,2-dihydrophthalazin-1-one
2-{5-cyclopropyl-4-[4-(2-methoxyethyl)piperazine-1-carbonyl]-1H-pyrazol-1-yl}-5-methyl-4-(thiophen-2-yl)pyrimidine
4-(3-ethoxy-2-hydroxyphenyl)-3-methyl-2-propyl-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-{4-[1-(propan-2-yl)-1H,4H-pyrazolo[3,4-d]imidazol-5-yl]phenyl}-1H-pyrazole
1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-N5-[2-(4-phenyl-1,3-thiazol-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
N-{[1-(4-methoxyphenyl)cyclopentyl]methyl}oxane-2-carboxamide
ethyl 1-({3-[3-(4-ethylpiperazin-1-yl)-2-hydroxypropoxy]phenyl}methyl)piperidine-4-carboxylate
[(2S,4R)-1-(3-chloro-5-methoxybenzoyl)-4-(dimethylamino)pyrrolidin-2-yl]methanol
5-{[benzyl(methyl)amino]methyl}-N-[2-hydroxy-1-(pyridin-3-yl)ethyl]-1,2-oxazole-3-carboxamide
N-[(3S,4R)-1-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-(3-hydroxypropyl)-9-{2-methylthieno[3,2-d]pyrimidin-4-yl}-2,9-diazaspiro[5.5]undecan-3-one
3,5-difluoro-2-[3-(3-methoxyphenoxymethyl)piperidine-1-carbonyl]pyridine
4-[2-(2-chlorophenyl)-3-methyl-3H-imidazo[4,5-b]pyridine-6-carbonyl]thiomorpholine
2-(2-{1-[3-(2H-1,3-benzodioxol-5-yl)propanoyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
8-(2-hydroxyacetyl)-3-{2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
4-(2H-1,3-benzodioxol-5-yl)-3-(1-methylpiperidin-3-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
(2S,4S)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-1-[(2,4-dimethylphenyl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
2-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]-5-(1,2,3,4-tetrahydroisoquinolin-2-yl)-2,3-dihydropyridazin-3-one
3-{[(1,3-dihydroxy-2-methylpropan-2-yl)amino]methyl}-1-[(2-fluoro-5-methoxyphenyl)methyl]-3-hydroxypiperidin-2-one
1-{[3-(2-butyl-2,5-dihydro-1H-pyrrole-1-carbonyl)-1,2-oxazol-5-yl]methyl}-4-ethylpiperazine
1-(2-{1-[2-(3,4-dimethylphenyl)acetyl]piperidin-2-yl}ethyl)pyrrolidin-2-one
2-{3,5-dimethyl-4-[2-(1H-pyrazol-1-yl)butanamido]-1H-pyrazol-1-yl}acetic acid
5-[1-(4-chloro-2-methylphenyl)-3-methyl-1H-1,2,4-triazol-5-yl]-2-(4H-1,2,4-triazol-4-yl)pyridine
N-[2-(dimethylamino)ethyl]-N-({1-[(2-methoxyphenyl)methyl]piperidin-3-yl}methyl)-2-(1H-pyrazol-1-yl)acetamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(2-methyl-1,3-oxazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-ethyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1,2,3,4-tetrahydronaphthalene-2-carboxamide
6-[4-(2-phenoxyethyl)piperazin-1-yl]-9H-purin-2-amine
2-(4-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-6-hydroxy-1,4-diazepan-1-yl)acetamide
2-{4-[(4-methoxy-3-methylphenyl)methyl]-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl}ethan-1-ol
N-{2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}-2-(pyridin-3-yl)-2-(pyrrolidin-1-yl)acetamide
1-ethyl-5-[2-methyl-5-(propan-2-yl)furan-3-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid