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1-[(3R,4S)-3-amino-4-(5-methylfuran-2-yl)pyrrolidin-1-yl]-4-phenylbutane-1,4-dione
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-[(1S,5R)-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
3-(2,4-dioxo-1,2,3,4-tetrahydropyrimidin-1-yl)-N-[(3-phenyl-1H-1,2,4-triazol-5-yl)methyl]propanamide
(3S,4S)-1-[2-(2,5-dimethyl-1H-pyrrol-1-yl)benzoyl]-4-(morpholin-4-yl)pyrrolidin-3-ol
(2S,4R)-4-amino-N-ethyl-1-[3-(1,2-oxazinan-2-yl)propanoyl]pyrrolidine-2-carboxamide
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidine-1-carbonyl]pyridine
N-[1-(2,4-dimethylphenyl)propyl]imidazo[1,2-a]pyridine-6-carboxamide
ethyl 5-(1-methyl-1H-1,3-benzodiazol-2-yl)-2-oxo-2,3-dihydro-1H-imidazole-4-carboxylate
N-[2-(2-fluorophenyl)ethyl]-1-(2-methylpropyl)-3-(morpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
2-(3-fluorophenyl)-5-[4-(pyridin-3-yloxy)piperidine-1-carbonyl]pyridine
2-{5-[6-amino-5-cyano-4-(1-ethyl-3-methyl-1H-pyrazol-4-yl)pyridin-2-yl]thiophen-3-yl}acetic acid
N-[2-(4-hydroxypiperidin-1-yl)ethyl]-3-(piperidin-3-yl)benzamide
1-(2-hydroxyethyl)-5-{imidazo[2,1-b][1,3]thiazole-6-carbonyl}-N-(1-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
3-{1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexan-6-ylmethyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
N-(1H-imidazol-2-ylmethyl)-N,1-dimethyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
(4aR,7aS)-1-[2-(4-aminopiperidin-1-yl)pyrimidin-4-yl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[(3R,4S)-4-cyclopropyl-1-(3-methoxypropyl)pyrrolidin-3-yl]benzenesulfonamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-(pyrazine-2-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
5-chloro-2-(4-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperazin-1-yl)pyrimidine
4-{1-[(2-carboxyethyl)carbamoyl]piperidin-3-yl}benzoic acid
N-methyl-N-[2-(oxan-4-yl)ethyl]-2-[5-(pyrrolidin-1-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]acetamide
8-(furan-3-ylmethyl)-1-methyl-3-(pyridin-3-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1'-(1-methyl-1H-pyrrole-2-carbonyl)-5-propyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-[4-(3-acetylphenyl)-3,5-dimethyl-1H-pyrazol-1-yl]propanamide
N-[(1-cyclopentylpiperidin-4-yl)methyl]-2-(morpholine-4-carbonyl)pyridin-4-amine
N3-[(4-fluorophenyl)methyl]-N5-methyl-4-oxo-1-(3-phenylpropyl)-1,4-dihydropyridine-3,5-dicarboxamide
2-[(4-chlorophenyl)methyl]-8-(cyclopropanesulfonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[(3S,4R)-3,4-dihydroxy-4-methylpiperidine-1-carbonyl]-6-methyl-1,2-dihydropyridin-2-one
N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
N-[(1-benzylpiperidin-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
3-cyclopentyl-5-(1,2-oxazol-3-yl)-1-(2-phenylethyl)-1H-1,2,4-triazole
(2R,3R)-3-methoxy-1'-(3-methoxypropyl)-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-[(4-benzylpiperazin-1-yl)methyl]-N-[2-(pyridin-2-yl)ethyl]-1,3-oxazole-4-carboxamide
7-methyl-N-{[2-(4-methylpiperazin-1-yl)pyridin-3-yl]methyl}-2-oxo-1H,2H-pyrazolo[1,5-a]pyrimidine-6-carboxamide
N-(3-hydroxy-1-{2-[(4-methoxyphenyl)methyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-1-oxopropan-2-yl)acetamide
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-6-methylpyrazolo[1,5-a]pyrimidine-3-carboxamide
N-[4-(1H-pyrazol-1-yl)phenyl]-1-(pyridin-3-ylmethyl)piperidine-2-carboxamide
2-(3-chlorophenyl)-N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}acetamide
4-(3,4-dichlorophenyl)-1-[1-(furan-2-yl)ethyl]-1H-1,2,3-triazole
5-(2-{2-[(3-chloropyridin-2-yl)amino]ethyl}morpholin-4-yl)-2-methyl-2,3-dihydropyridazin-3-one
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-2-hydroxy-2-methylpropanamide
4-ethyl-5-{3-[2-(4-fluorophenyl)ethyl]piperidine-1-carbonyl}-1,3-thiazol-2-amine
8-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[1-(carbamoylmethyl)piperidin-4-yl]formamido}-2-(2-fluorophenyl)acetic acid
6-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
1-[4-(furan-2-yl)pyrimidin-2-yl]-N,5-dimethyl-N-(quinolin-5-ylmethyl)-1H-pyrazole-4-carboxamide
1-(cyclohexylmethyl)-5-(4H-1,2,4-triazol-4-ylmethyl)-1H-1,2,4-triazole
2-(2-hydroxyethyl)-8-(pyrazin-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
4-chloro-N-[(3R,4S)-4-cyclopropyl-1-methanesulfonylpyrrolidin-3-yl]-1-methyl-1H-pyrazole-5-carboxamide